Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with all data for entry = 50013183
TargetChloroquine resistance transporter(Plasmodium falciparum)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50563441(CHEMBL4745810)
Affinity DataIC50:  1.25E+4nMAssay Description:Inhibition of Plasmodium falciparum Dd2 CRT expressed in Xenopus laevis oocyte assessed as inhibition of [3H]-CQ transport incubated for 1.5 hrs by m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChloroquine resistance transporter(Plasmodium falciparum)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50563442(CHEMBL4754685)
Affinity DataIC50:  1.56E+4nMAssay Description:Inhibition of Plasmodium falciparum Dd2 CRT expressed in Xenopus laevis oocyte assessed as inhibition of [3H]-CQ transport incubated for 1.5 hrs by m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChloroquine resistance transporter(Plasmodium falciparum)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50563440(CHEMBL4784051)
Affinity DataIC50:  5.50E+4nMAssay Description:Inhibition of Plasmodium falciparum Dd2 CRT expressed in Xenopus laevis oocyte assessed as inhibition of [3H]-CQ transport incubated for 1.5 hrs by m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChloroquine resistance transporter(Plasmodium falciparum)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50563439(CHEMBL4748649)
Affinity DataIC50:  6.40E+4nMAssay Description:Inhibition of Plasmodium falciparum Dd2 CRT expressed in Xenopus laevis oocyte assessed as inhibition of [3H]-CQ transport incubated for 1.5 hrs by m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed