Compile Data Set for Download or QSAR
maximum 50k data
Found 18 Enz. Inhib. hit(s) with all data for entry = 3220
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM29511(Pyranonaphthoquinone (PNQ) lactone, 11a)
Affinity DataIC50:  44nMpH: 7.4 T: 2°CAssay Description:AKT1 was assayed using constitutively active Myr-AKT1 in low-binding 96-well plates. The kinase reactions were initiated by the addition of assay mix...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM29512(Pyranonaphthoquinone (PNQ) lactone, 11b)
Affinity DataIC50:  57nMpH: 7.4 T: 2°CAssay Description:AKT1 was assayed using constitutively active Myr-AKT1 in low-binding 96-well plates. The kinase reactions were initiated by the addition of assay mix...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM29513(Pyranonaphthoquinone (PNQ) lactone, 11c)
Affinity DataIC50:  72nMpH: 7.4 T: 2°CAssay Description:AKT1 was assayed using constitutively active Myr-AKT1 in low-binding 96-well plates. The kinase reactions were initiated by the addition of assay mix...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM29514(Pyranonaphthoquinone (PNQ) lactone, 11d)
Affinity DataIC50:  80nMpH: 7.4 T: 2°CAssay Description:AKT1 was assayed using constitutively active Myr-AKT1 in low-binding 96-well plates. The kinase reactions were initiated by the addition of assay mix...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM29515(Pyranonaphthoquinone (PNQ) lactone, 11e)
Affinity DataIC50:  99nMpH: 7.4 T: 2°CAssay Description:AKT1 was assayed using constitutively active Myr-AKT1 in low-binding 96-well plates. The kinase reactions were initiated by the addition of assay mix...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM29516(Pyranonaphthoquinone (PNQ) lactone, 11f)
Affinity DataIC50:  122nMpH: 7.4 T: 2°CAssay Description:AKT1 was assayed using constitutively active Myr-AKT1 in low-binding 96-well plates. The kinase reactions were initiated by the addition of assay mix...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM29506(Lactoquinomycin | Lactoquinomycin A)
Affinity DataIC50:  149nMpH: 7.4 T: 2°CAssay Description:AKT1 was assayed using constitutively active Myr-AKT1 in low-binding 96-well plates. The kinase reactions were initiated by the addition of assay mix...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM29517(Pyranonaphthoquinone (PNQ) lactone, 11g)
Affinity DataIC50:  150nMpH: 7.4 T: 2°CAssay Description:AKT1 was assayed using constitutively active Myr-AKT1 in low-binding 96-well plates. The kinase reactions were initiated by the addition of assay mix...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM29518(Pyranonaphthoquinone (PNQ) lactone, 11h)
Affinity DataIC50:  163nMpH: 7.4 T: 2°CAssay Description:AKT1 was assayed using constitutively active Myr-AKT1 in low-binding 96-well plates. The kinase reactions were initiated by the addition of assay mix...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM29508(Frenolicin B)
Affinity DataIC50:  198nMpH: 7.4 T: 2°CAssay Description:AKT1 was assayed using constitutively active Myr-AKT1 in low-binding 96-well plates. The kinase reactions were initiated by the addition of assay mix...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM29519(Pyranonaphthoquinone (PNQ) lactone, 11i)
Affinity DataIC50:  295nMpH: 7.4 T: 2°CAssay Description:AKT1 was assayed using constitutively active Myr-AKT1 in low-binding 96-well plates. The kinase reactions were initiated by the addition of assay mix...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM29507(Kalafungin | Kalamycin | cid_283138)
Affinity DataIC50:  313nMpH: 7.4 T: 2°CAssay Description:AKT1 was assayed using constitutively active Myr-AKT1 in low-binding 96-well plates. The kinase reactions were initiated by the addition of assay mix...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM29520(Pyranonaphthoquinone (PNQ) lactone, 11j)
Affinity DataIC50:  350nMpH: 7.4 T: 2°CAssay Description:AKT1 was assayed using constitutively active Myr-AKT1 in low-binding 96-well plates. The kinase reactions were initiated by the addition of assay mix...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM29521(Pyranonaphthoquinone (PNQ) lactone, 11k)
Affinity DataIC50:  383nMpH: 7.4 T: 2°CAssay Description:AKT1 was assayed using constitutively active Myr-AKT1 in low-binding 96-well plates. The kinase reactions were initiated by the addition of assay mix...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM29510(Deoxyfrenolicin)
Affinity DataIC50:  424nMpH: 7.4 T: 2°CAssay Description:AKT1 was assayed using constitutively active Myr-AKT1 in low-binding 96-well plates. The kinase reactions were initiated by the addition of assay mix...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM29509(Frenolicin B analogue, 4)
Affinity DataIC50:  497nMpH: 7.4 T: 2°CAssay Description:AKT1 was assayed using constitutively active Myr-AKT1 in low-binding 96-well plates. The kinase reactions were initiated by the addition of assay mix...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM29522(Pyranonaphthoquinone (PNQ) lactone, 11l)
Affinity DataIC50:  850nMpH: 7.4 T: 2°CAssay Description:AKT1 was assayed using constitutively active Myr-AKT1 in low-binding 96-well plates. The kinase reactions were initiated by the addition of assay mix...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM29523(Pyranonaphthoquinone (PNQ) lactone, 11m)
Affinity DataIC50:  1.44E+3nMpH: 7.4 T: 2°CAssay Description:AKT1 was assayed using constitutively active Myr-AKT1 in low-binding 96-well plates. The kinase reactions were initiated by the addition of assay mix...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed