Compile Data Set for Download or QSAR
maximum 50k data
Found 56 Enz. Inhib. hit(s) with all data for entry = 50033065
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339043(2-(2-((4-Pyridyl)methyl)aminophenyl)-5-(3,4-ethyle...)
Affinity DataIC50:  110nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339053(CHEMBL1688357 | N-(2,3-dihydrobenzo[b][1,4]dioxin-...)
Affinity DataIC50:  150nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addtion of substrate measur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339046(5-(2-((1H-imidazol-5-yl)methylamino)pyridin-3-yl)-...)
Affinity DataIC50:  160nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addtion of substrate measur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50179492(3-(5-(2,3-dihydrobenzo[b][1,4]dioxin-6-ylamino)-1,...)
Affinity DataIC50:  170nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addtion of substrate measur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339043(2-(2-((4-Pyridyl)methyl)aminophenyl)-5-(3,4-ethyle...)
Affinity DataIC50:  210nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addtion of substrate measur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339048(CHEMBL1688352 | N-(2,3-dihydrobenzo[b][1,4]dioxin-...)
Affinity DataIC50:  220nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339048(CHEMBL1688352 | N-(2,3-dihydrobenzo[b][1,4]dioxin-...)
Affinity DataIC50:  300nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addtion of substrate measur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339054(2-(2-((4-Pyridyl)methyl)aminophenyl)-5-(3,4-methyl...)
Affinity DataIC50:  830nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addtion of substrate measur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339046(5-(2-((1H-imidazol-5-yl)methylamino)pyridin-3-yl)-...)
Affinity DataIC50:  830nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339037(CHEMBL1688246 | N-(pyridin-4-ylmethyl)-3-(5-(3-(tr...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50179492(3-(5-(2,3-dihydrobenzo[b][1,4]dioxin-6-ylamino)-1,...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339037(CHEMBL1688246 | N-(pyridin-4-ylmethyl)-3-(5-(3-(tr...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addtion of substrate measur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339047(5-(2-((1H-indazol-5-yl)methylamino)pyridin-3-yl)-N...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addtion of substrate measur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50179495(3-(5-(benzo[d][1,3]dioxol-5-ylamino)-1,3,4-oxadiaz...)
Affinity DataIC50:  1.89E+3nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addtion of substrate measur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339040(3-(5-(benzo[d][1,3]dioxol-5-yl)-4H-1,2,4-triazol-3...)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addtion of substrate measur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339039(CHEMBL1688248 | N-(pyridin-4-ylmethyl)-3-(5-(3-(tr...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addtion of substrate measur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50179502(CHEMBL203642 | N-(benzo[d][1,3]dioxol-5-ylmethyl)-...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addtion of substrate measur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339050(CHEMBL1688354 | N-(2,3-dihydrobenzo[b][1,4]dioxin-...)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339052(5-(2-((1H-indazol-5-yl)methylamino)phenyl)-N-(2,3-...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addtion of substrate measur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339055(CHEMBL1688344 | N-(2,2-difluorobenzo[d][1,3]dioxol...)
Affinity DataIC50:  3.16E+3nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addtion of substrate measur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339050(CHEMBL1688354 | N-(2,3-dihydrobenzo[b][1,4]dioxin-...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addtion of substrate measur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339057(CHEMBL1688346 | N-(benzo[d][1,3]dioxol-5-yl)-5-(2-...)
Affinity DataIC50:  3.41E+3nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addtion of substrate measur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339041(CHEMBL1688250 | N-((1,4-dioxan-2-yl)methyl)-3-(5-(...)
Affinity DataIC50:  4.50E+3nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addtion of substrate measur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339051(5-(2-((1H-imidazol-5-yl)methylamino)phenyl)-N-(2,3...)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addtion of substrate measur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339049(CHEMBL1688353 | N-(2,3-dihydrobenzo[b][1,4]dioxin-...)
Affinity DataIC50:  5.10E+3nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addtion of substrate measur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339052(5-(2-((1H-indazol-5-yl)methylamino)phenyl)-N-(2,3-...)
Affinity DataIC50:  7.30E+3nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50179487(3-(5-(benzo[d][1,3]dioxol-5-ylamino)-1,3,4-oxadiaz...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addtion of substrate measur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50179498(3-(5-(benzo[d][1,3]dioxol-5-ylamino)-1,3,4-oxadiaz...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addtion of substrate measur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339056(CHEMBL1688345 | N-(benzo[d][1,3]dioxol-5-yl)-5-(2-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addtion of substrate measur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339053(CHEMBL1688357 | N-(2,3-dihydrobenzo[b][1,4]dioxin-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339051(5-(2-((1H-imidazol-5-yl)methylamino)phenyl)-N-(2,3...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339049(CHEMBL1688353 | N-(2,3-dihydrobenzo[b][1,4]dioxin-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339047(5-(2-((1H-indazol-5-yl)methylamino)pyridin-3-yl)-N...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339045(CHEMBL1688349 | N-(2,3-dihydrobenzo[b][1,4]dioxin-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339044(CHEMBL1688348 | N-(2,3-dihydrobenzo[b][1,4]dioxin-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50179502(CHEMBL203642 | N-(benzo[d][1,3]dioxol-5-ylmethyl)-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50179504(3-(5-(2,3-dihydrobenzo[b][1,4]dioxin-6-ylamino)-1,...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50179501(3-(5-(2,3-dihydrobenzo[b][1,4]dioxin-6-ylamino)-1,...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339042(CHEMBL1688347 | N-(benzo[d][1,3]dioxol-5-yl)-5-(2-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339057(CHEMBL1688346 | N-(benzo[d][1,3]dioxol-5-yl)-5-(2-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339056(CHEMBL1688345 | N-(benzo[d][1,3]dioxol-5-yl)-5-(2-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50179498(3-(5-(benzo[d][1,3]dioxol-5-ylamino)-1,3,4-oxadiaz...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50179487(3-(5-(benzo[d][1,3]dioxol-5-ylamino)-1,3,4-oxadiaz...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339055(CHEMBL1688344 | N-(2,2-difluorobenzo[d][1,3]dioxol...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339054(2-(2-((4-Pyridyl)methyl)aminophenyl)-5-(3,4-methyl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50179495(3-(5-(benzo[d][1,3]dioxol-5-ylamino)-1,3,4-oxadiaz...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339041(CHEMBL1688250 | N-((1,4-dioxan-2-yl)methyl)-3-(5-(...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339040(3-(5-(benzo[d][1,3]dioxol-5-yl)-4H-1,2,4-triazol-3...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339039(CHEMBL1688248 | N-(pyridin-4-ylmethyl)-3-(5-(3-(tr...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339038(CHEMBL1688247 | N-((1H-pyrazol-4-yl)methyl)-3-(5-(...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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