Compile Data Set for Download or QSAR
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Found 30 Enz. Inhib. hit(s) with all data for entry = 50047502
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50117930((4-{1-[2-(6-Methyl-pyridin-2-yl)-ethyl]-piperidine...)
Affinity DataIC50:  70nMAssay Description:Inhibition of human ERG expressed in cell membranes after 4 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50171845(CHEMBL3805971)
Affinity DataEC50:  3.69E+3nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium influx assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50171849(CHEMBL3805668)
Affinity DataEC50:  1.52E+3nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium influx assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50171853(CHEMBL3805086)
Affinity DataEC50:  6.64E+3nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium influx assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50171855(CHEMBL3806055)
Affinity DataEC50:  1.77E+3nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium influx assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50171865(CHEMBL3805888)
Affinity DataEC50:  580nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium influx assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50171866(CHEMBL3805143)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium influx assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50171867(CHEMBL3806208)
Affinity DataEC50:  1.06E+3nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium influx assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50171868(CHEMBL3804883)
Affinity DataEC50:  1.79E+4nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium influx assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50171869(CHEMBL3805303)
Affinity DataEC50:  1.64E+3nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium influx assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50171870(CHEMBL3805879)
Affinity DataEC50:  1.28E+3nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium influx assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50171871(CHEMBL3805558)
Affinity DataEC50:  1.69E+3nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium influx assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50171872(CHEMBL3805328)
Affinity DataEC50:  760nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium influx assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50171873(CHEMBL3805952)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR120 (unknown origin) expressed in CHO cells by calcium influx assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50171865(CHEMBL3805888)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR120 (unknown origin) expressed in CHO cells by calcium influx assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50171870(CHEMBL3805879)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR120 (unknown origin) expressed in CHO cells by calcium influx assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50171872(CHEMBL3805328)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR120 (unknown origin) expressed in CHO cells by calcium influx assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50171873(CHEMBL3805952)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR43 (unknown origin) expressed in CHO cells by calcium influx assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50171865(CHEMBL3805888)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR43 (unknown origin) expressed in CHO cells by calcium influx assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50171870(CHEMBL3805879)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR43 (unknown origin) expressed in CHO cells by calcium influx assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50171872(CHEMBL3805328)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR43 (unknown origin) expressed in CHO cells by calcium influx assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 3(Homo sapiens (Human))
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50171873(CHEMBL3805952)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR41 (unknown origin) expressed in CHO cells by calcium influx assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 3(Homo sapiens (Human))
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50171865(CHEMBL3805888)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR41 (unknown origin) expressed in CHO cells by calcium influx assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 3(Homo sapiens (Human))
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50171870(CHEMBL3805879)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR41 (unknown origin) expressed in CHO cells by calcium influx assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 3(Homo sapiens (Human))
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50171872(CHEMBL3805328)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR41 (unknown origin) expressed in CHO cells by calcium influx assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50171874(CHEMBL3805377)
Affinity DataEC50:  1.06E+4nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium influx assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50171875(CHEMBL3805246)
Affinity DataEC50:  4.30E+3nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium influx assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50171873(CHEMBL3805952)
Affinity DataEC50:  580nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium influx assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50171876(CHEMBL3805670)
Affinity DataEC50:  4.68E+3nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium influx assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50171832(CHEMBL3805903)
Affinity DataEC50:  1.19E+3nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium influx assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed