Compile Data Set for Download or QSAR
maximum 50k data
Found 64 Enz. Inhib. hit(s) with all data for entry = 50010228
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50024253(CHEMBL3334887)
Affinity DataIC50:  66nMAssay Description:Antagonist activity at PAR4 in human platelets after 10 mins by flow cytometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536645(CHEMBL4528799)
Affinity DataIC50: <100nMAssay Description:Inhibition of CYP2D6 in human liver microsomes incubated for 15 mins using dextromethorphan substrate in presence of NADPH by LC-MS/MS methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536646(CHEMBL4557930)
Affinity DataIC50:  120nMAssay Description:Inhibition of CYP2D6 in human liver microsomes incubated for 15 mins using dextromethorphan substrate in presence of NADPH by LC-MS/MS methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50024254(CHEMBL125021)
Affinity DataIC50:  130nMAssay Description:Antagonist activity PAR4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536642(CHEMBL4566669)
Affinity DataIC50:  132nMAssay Description:Antagonist activity against PAR4 activating peptide domain in in human platelets assessed as inhibition of P-selectin activationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536642(CHEMBL4566669)
Affinity DataIC50:  178nMAssay Description:Antagonist activity against PAR4 activating peptide domain in human platelets assessed as inhibition of alpha2bbeta3 activation level by PAC1 binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536642(CHEMBL4566669)
Affinity DataIC50:  180nMAssay Description:Antagonist activity against PAR4 activating peptide domain in human platelets assessed as inhibition of alpha2bbeta3 activation level by PAC1 binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536657(CHEMBL4586027)
Affinity DataIC50:  204nMAssay Description:Antagonist activity against PAR4 activating peptide domain in human platelets assessed as inhibition of alpha2bbeta3 activation level by PAC1 binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536657(CHEMBL4586027)
Affinity DataIC50:  210nMAssay Description:Antagonist activity against PAR4 activating peptide domain in human platelets assessed as inhibition of alpha2bbeta3 activation level by PAC1 binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536646(CHEMBL4557930)
Affinity DataIC50:  435nMAssay Description:Antagonist activity against PAR4 activating peptide domain in in human platelets assessed as inhibition of P-selectin activationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536646(CHEMBL4557930)
Affinity DataIC50:  450nMAssay Description:Antagonist activity against PAR4 activating peptide domain in human platelets assessed as inhibition of alpha2bbeta3 activation level by PAC1 binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536646(CHEMBL4557930)
Affinity DataIC50:  490nMAssay Description:Antagonist activity against PAR4 activating peptide domain in human platelets assessed as inhibition of alpha2bbeta3 activation level by PAC1 binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536645(CHEMBL4528799)
Affinity DataIC50:  490nMAssay Description:Antagonist activity against PAR4 activating peptide domain in human platelets assessed as inhibition of alpha2bbeta3 activation level by PAC1 binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536645(CHEMBL4528799)
Affinity DataIC50:  490nMAssay Description:Antagonist activity against PAR4 activating peptide domain in human platelets assessed as inhibition of alpha2bbeta3 activation level by PAC1 binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536659(CHEMBL4517009)
Affinity DataIC50:  813nMAssay Description:Antagonist activity against PAR4 activating peptide domain in human platelets assessed as inhibition of alpha2bbeta3 activation level by PAC1 binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536659(CHEMBL4517009)
Affinity DataIC50:  820nMAssay Description:Antagonist activity against PAR4 activating peptide domain in human platelets assessed as inhibition of alpha2bbeta3 activation level by PAC1 binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536642(CHEMBL4566669)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of CYP2D6 in human liver microsomes incubated for 15 mins using dextromethorphan substrate in presence of NADPH by LC-MS/MS methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536643(CHEMBL4567147)
Affinity DataIC50:  1.35E+3nMAssay Description:Antagonist activity against PAR4 activating peptide domain in human platelets assessed as inhibition of alpha2bbeta3 activation level by PAC1 binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536643(CHEMBL4567147)
Affinity DataIC50:  1.35E+3nMAssay Description:Antagonist activity against PAR4 activating peptide domain in human platelets assessed as inhibition of alpha2bbeta3 activation level by PAC1 binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536644(CHEMBL4537098)
Affinity DataIC50:  1.38E+3nMAssay Description:Antagonist activity against PAR4 activating peptide domain in human platelets assessed as inhibition of alpha2bbeta3 activation level by PAC1 binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536644(CHEMBL4537098)
Affinity DataIC50:  1.39E+3nMAssay Description:Antagonist activity against PAR4 activating peptide domain in human platelets assessed as inhibition of alpha2bbeta3 activation level by PAC1 binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536654(CHEMBL4570494)
Affinity DataIC50:  1.50E+3nMAssay Description:Antagonist activity against PAR4 activating peptide domain in human platelets assessed as inhibition of alpha2bbeta3 activation level by PAC1 binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536654(CHEMBL4570494)
Affinity DataIC50:  1.51E+3nMAssay Description:Antagonist activity against PAR4 activating peptide domain in human platelets assessed as inhibition of alpha2bbeta3 activation level by PAC1 binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536663(CHEMBL4483019)
Affinity DataIC50:  2.19E+3nMAssay Description:Antagonist activity against PAR4 activating peptide domain in human platelets assessed as inhibition of alpha2bbeta3 activation level by PAC1 binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536663(CHEMBL4483019)
Affinity DataIC50:  2.19E+3nMAssay Description:Antagonist activity against PAR4 activating peptide domain in human platelets assessed as inhibition of alpha2bbeta3 activation level by PAC1 binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536645(CHEMBL4528799)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of CYP1A2 in human liver microsomes incubated for 15 mins using phenacetin substrate in presence of NADPH by LC-MS/MS methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536656(CHEMBL4571068)
Affinity DataIC50:  3.72E+3nMAssay Description:Antagonist activity against PAR4 activating peptide domain in human platelets assessed as inhibition of alpha2bbeta3 activation level by PAC1 binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536656(CHEMBL4571068)
Affinity DataIC50:  3.76E+3nMAssay Description:Antagonist activity against PAR4 activating peptide domain in human platelets assessed as inhibition of alpha2bbeta3 activation level by PAC1 binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536661(CHEMBL4516569)
Affinity DataIC50:  4.15E+3nMAssay Description:Antagonist activity against PAR4 activating peptide domain in human platelets assessed as inhibition of alpha2bbeta3 activation level by PAC1 binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536661(CHEMBL4516569)
Affinity DataIC50:  4.17E+3nMAssay Description:Antagonist activity against PAR4 activating peptide domain in human platelets assessed as inhibition of alpha2bbeta3 activation level by PAC1 binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536646(CHEMBL4557930)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of CYP1A2 in human liver microsomes incubated for 15 mins using phenacetin substrate in presence of NADPH by LC-MS/MS methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536642(CHEMBL4566669)
Affinity DataIC50:  4.35E+3nMAssay Description:Antagonist activity at PAR4 TL domain in human platelets assessed as gamma-thrombin-induced PAC1 binding response preincubated for 20 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536650(CHEMBL4544189)
Affinity DataIC50:  4.79E+3nMAssay Description:Antagonist activity against PAR4 activating peptide domain in human platelets assessed as inhibition of alpha2bbeta3 activation level by PAC1 binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536650(CHEMBL4544189)
Affinity DataIC50:  4.82E+3nMAssay Description:Antagonist activity against PAR4 activating peptide domain in human platelets assessed as inhibition of alpha2bbeta3 activation level by PAC1 binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536660(CHEMBL4514069)
Affinity DataIC50:  4.90E+3nMAssay Description:Antagonist activity against PAR4 activating peptide domain in human platelets assessed as inhibition of alpha2bbeta3 activation level by PAC1 binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536660(CHEMBL4514069)
Affinity DataIC50:  4.91E+3nMAssay Description:Antagonist activity against PAR4 activating peptide domain in human platelets assessed as inhibition of alpha2bbeta3 activation level by PAC1 binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536641(CHEMBL4514977)
Affinity DataIC50:  5.11E+3nMAssay Description:Antagonist activity against PAR4 activating peptide domain in human platelets assessed as inhibition of alpha2bbeta3 activation level by PAC1 binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536641(CHEMBL4514977)
Affinity DataIC50:  5.13E+3nMAssay Description:Antagonist activity against PAR4 activating peptide domain in human platelets assessed as inhibition of alpha2bbeta3 activation level by PAC1 binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536645(CHEMBL4528799)
Affinity DataIC50:  6.10E+3nMAssay Description:Inhibition of CYP2C9 in human liver microsomes incubated for 15 mins using diclofenac substrate in presence of NADPH by LC-MS/MS methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536646(CHEMBL4557930)
Affinity DataIC50:  6.80E+3nMAssay Description:Inhibition of CYP2C9 in human liver microsomes incubated for 15 mins using diclofenac substrate in presence of NADPH by LC-MS/MS methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536646(CHEMBL4557930)
Affinity DataIC50:  9.40E+3nMAssay Description:Antagonist activity at PAR4 TL domain in human platelets assessed as gamma-thrombin-induced PAC1 binding response preincubated for 20 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50024253(CHEMBL3334887)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of PAR1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536646(CHEMBL4557930)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at PAR4 TL domain in human platelets assessed as gamma-thrombin-induced P-selectin activation preincubated for 20 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536649(CHEMBL4577100)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity against PAR4 activating peptide domain in human platelets assessed as inhibition of alpha2bbeta3 activation level by PAC1 binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536648(CHEMBL4526529)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity against PAR4 activating peptide domain in human platelets assessed as inhibition of alpha2bbeta3 activation level by PAC1 binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536655(CHEMBL4517686)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity against PAR4 activating peptide domain in human platelets assessed as inhibition of alpha2bbeta3 activation level by PAC1 binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536653(CHEMBL4593803)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity against PAR4 activating peptide domain in human platelets assessed as inhibition of alpha2bbeta3 activation level by PAC1 binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536652(CHEMBL4544905)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity against PAR4 activating peptide domain in human platelets assessed as inhibition of alpha2bbeta3 activation level by PAC1 binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536662(CHEMBL4548807)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity against PAR4 activating peptide domain in human platelets assessed as inhibition of alpha2bbeta3 activation level by PAC1 binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50536651(CHEMBL4559153)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity against PAR4 activating peptide domain in human platelets assessed as inhibition of alpha2bbeta3 activation level by PAC1 binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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