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Found 15 Enz. Inhib. hit(s) with all data for entry = 50030138
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291519(3-(3-Biphenyl-4-yl-but-2-enoylamino)-4-methoxy-ben...)
Affinity DataIC50:  16nMAssay Description:In vitro binding affinity towards LTB4 receptor determined by measuring the displacement of [3H]-LTB4 from isolated neutrophilsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291521((E)-3-Biphenyl-4-yl-N-[2-methoxy-5-(1H-tetrazol-5-...)
Affinity DataIC50:  17nMAssay Description:In vitro binding affinity towards LTB4 receptor determined by measuring the displacement of [3H]-LTB4 from isolated neutrophilsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291516(3-((E)-3-Biphenyl-4-yl-acryloylamino)-4-methoxy-be...)
Affinity DataIC50:  68nMAssay Description:In vitro binding affinity towards LTB4 receptor determined by measuring the displacement of [3H]-LTB4 from isolated neutrophilsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291512(3-((E)-3-Biphenyl-4-yl-acryloylamino)-4-ethoxy-ben...)
Affinity DataIC50:  190nMAssay Description:In vitro binding affinity towards LTB4 receptor determined by measuring the displacement of [3H]-LTB4 from isolated neutrophilsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291515(4-Methoxy-3-[3-(4'-methyl-biphenyl-4-yl)-acryloyla...)
Affinity DataIC50:  276nMAssay Description:In vitro binding affinity towards LTB4 receptor determined by measuring the displacement of [3H]-LTB4 from isolated neutrophilsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291507(3-(3-Biphenyl-4-yl-3-oxo-propionylamino)-4-methoxy...)
Affinity DataIC50:  784nMAssay Description:In vitro binding affinity towards LTB4 receptor determined by measuring the displacement of [3H]-LTB4 from isolated neutrophilsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291511(2-((E)-3-Biphenyl-4-yl-acryloylamino)-benzoic acid...)
Affinity DataIC50:  830nMAssay Description:In vitro binding affinity towards LTB4 receptor determined by measuring the displacement of [3H]-LTB4 from isolated neutrophilsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291509(3-((E)-3-Biphenyl-4-yl-acryloylamino)-4-chloro-ben...)
Affinity DataIC50:  908nMAssay Description:In vitro binding affinity towards LTB4 receptor determined by measuring the displacement of [3H]-LTB4 from isolated neutrophilsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291510(3-[((1S,2S)-2-Biphenyl-4-yl-cyclopropanecarbonyl)-...)
Affinity DataIC50:  932nMAssay Description:In vitro binding affinity towards LTB4 receptor determined by measuring the displacement of [3H]-LTB4 from isolated neutrophilsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291518(2-((E)-3-Biphenyl-4-yl-acryloylamino)-3-methoxy-be...)
Affinity DataIC50:  1.18E+3nMAssay Description:In vitro binding affinity towards LTB4 receptor determined by measuring the displacement of [3H]-LTB4 from isolated neutrophilsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291514(3-((E)-3-Biphenyl-4-yl-acryloylamino)-benzoic acid...)
Affinity DataIC50:  1.18E+3nMAssay Description:In vitro binding affinity towards LTB4 receptor determined by measuring the displacement of [3H]-LTB4 from isolated neutrophilsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291520(4-Methoxy-3-[3-(2-methyl-biphenyl-4-yl)-acryloylam...)
Affinity DataIC50:  1.22E+3nMAssay Description:In vitro binding affinity towards LTB4 receptor determined by measuring the displacement of [3H]-LTB4 from isolated neutrophilsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291517(3-(3-Biphenyl-4-yl-propionylamino)-4-methoxy-benzo...)
Affinity DataIC50:  1.51E+3nMAssay Description:In vitro binding affinity towards LTB4 receptor determined by measuring the displacement of [3H]-LTB4 from isolated neutrophilsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291513(4-Methoxy-3-[3-(2'-methyl-biphenyl-4-yl)-acryloyla...)
Affinity DataIC50:  4.57E+3nMAssay Description:In vitro binding affinity towards LTB4 receptor determined by measuring the displacement of [3H]-LTB4 from isolated neutrophilsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291508((E)-3-Biphenyl-4-yl-N-(2-methoxy-phenyl)-acrylamid...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro binding affinity towards LTB4 receptor determined by measuring the displacement of [3H]-LTB4 from isolated neutrophilsMore data for this Ligand-Target Pair
In DepthDetails Article