Compile Data Set for Download or QSAR
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Found 15 Enz. Inhib. hit(s) with all data for entry = 50006741
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50052975(CHEMBL118797 | Methyl-[2-(4-nitro-phenyl)-ethyl]-(...)
Affinity DataKi:  4.30nMAssay Description:Displacement of [3H]-(+)-pentazocine from Sigma opioid receptor type 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50052965(CHEMBL118405 | Methyl-[2-(3-nitro-phenyl)-ethyl]-(...)
Affinity DataKi:  6.40nMAssay Description:Displacement of [3H]-(+)-pentazocine from Sigma opioid receptor type 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50052968(CHEMBL324513 | Methyl-[2-(2-nitro-phenyl)-ethyl]-(...)
Affinity DataKi:  7.70nMAssay Description:Displacement of [3H]-(+)-pentazocine from Sigma opioid receptor type 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50052966(CHEMBL115956 | [2-(2-Methoxy-phenyl)-ethyl]-methyl...)
Affinity DataKi:  15.7nMAssay Description:Displacement of [3H]-(+)-pentazocine from Sigma opioid receptor type 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50052964(CHEMBL119104 | [2-(3-Methoxy-phenyl)-ethyl]-methyl...)
Affinity DataKi:  23.8nMAssay Description:Displacement of [3H]-(+)-pentazocine from Sigma opioid receptor type 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50052971(CHEMBL118297 | [2-(4-Methoxy-phenyl)-ethyl]-methyl...)
Affinity DataKi:  30.3nMAssay Description:Displacement of [3H]-(+)-pentazocine from Sigma opioid receptor type 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50052967(4-{2-[Methyl-(2-pyrrolidin-1-yl-ethyl)-amino]-ethy...)
Affinity DataKi:  276nMAssay Description:Displacement of [3H]-(+)-pentazocine from Sigma opioid receptor type 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50052977(2-{2-[Methyl-(2-pyrrolidin-1-yl-ethyl)-amino]-ethy...)
Affinity DataKi:  291nMAssay Description:Displacement of [3H]-(+)-pentazocine from Sigma opioid receptor type 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50052969(3-{2-[Methyl-(2-pyrrolidin-1-yl-ethyl)-amino]-ethy...)
Affinity DataKi:  579nMAssay Description:Displacement of [3H]-(+)-pentazocine from Sigma opioid receptor type 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50052973(CHEMBL119310 | N-Methyl-2-(2-nitro-phenyl)-N-(2-py...)
Affinity DataKi:  736nMAssay Description:Displacement of [3H]-(+)-pentazocine from Sigma opioid receptor type 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50052976(CHEMBL116773 | N-Methyl-2-(4-nitro-phenyl)-N-(2-py...)
Affinity DataKi:  869nMAssay Description:Displacement of [3H]-(+)-pentazocine from Sigma opioid receptor type 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50052972(CHEMBL326935 | N-Methyl-2-(3-nitro-phenyl)-N-(2-py...)
Affinity DataKi:  1.85E+3nMAssay Description:Displacement of [3H]-(+)-pentazocine from Sigma opioid receptor type 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50052974(2-(4-Methoxy-phenyl)-N-methyl-N-(2-pyrrolidin-1-yl...)
Affinity DataKi:  2.22E+3nMAssay Description:Displacement of [3H]-(+)-pentazocine from Sigma opioid receptor type 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50052970(2-(3-Methoxy-phenyl)-N-methyl-N-(2-pyrrolidin-1-yl...)
Affinity DataKi:  3.10E+3nMAssay Description:Displacement of [3H]-(+)-pentazocine from Sigma opioid receptor type 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50052963(2-(2-Methoxy-phenyl)-N-methyl-N-(2-pyrrolidin-1-yl...)
Affinity DataKi:  5.46E+3nMAssay Description:Displacement of [3H]-(+)-pentazocine from Sigma opioid receptor type 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed