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Target
Interleukin-1 receptor antagonist protein
Ligand
BDBM50570140
Substrate
n/a
Meas. Tech.
ChEMBL_2111177 (CHEMBL4820027)
IC50
100000±n/a nM
Citation
Laura, M; Ronan, G; Vy, LB; Valentin, G; Omar, CA; Virgyl, C; Piveteau, C; Melissa, R; Charlotte, F; Sandrine, W; Julie, C; Julie, DR; Damien, B; Florence, L; Peter, VE; Benoit, D; Rebecca, DP Modulators of hERAP2 discovered by high-throughput screening. Eur J Med Chem 211:0 (2021) [PubMed] Article
More Info.:
Target
Name:
Interleukin-1 receptor antagonist protein
Synonyms:
ICIL-1RA | IL-1RN | IL-1ra | IL1 inhibitor | IL1F3 | IL1RA | IL1RA_HUMAN | IL1RN | INN=Anakinra | IRAP | Interleukin-1 receptor antagonist protein
Type:
PROTEIN
Mol. Mass.:
20053.78
Organism:
Homo sapiens
Description:
ChEMBL_118941
Residue:
177
Sequence:
MEICRGLRSHLITLLLFLFHSETICRPSGRKSSKMQAFRIWDVNQKTFYLRNNQLVAGYLQGPNVNLEEKIDVVPIEPHALFLGIHGGKMCLSCVKSGDETRLQLEAVNITDLSENRKQDKRFAFIRSDSGPTTSFESAACPGWFLCTAMEADQPVSLTNMPDEGVMVTKFYFQEDE