TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
Institut Pasteur De Lille
Curated by ChEMBL
Institut Pasteur De Lille
Curated by ChEMBL
Affinity DataIC50: 9.70E+3nMAssay Description:Inhibition of recombinant ERAP2 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using R-AMC as substrate preincubated for 30 min...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
Institut Pasteur De Lille
Curated by ChEMBL
Institut Pasteur De Lille
Curated by ChEMBL
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of human ERAP1More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
Institut Pasteur De Lille
Curated by ChEMBL
Institut Pasteur De Lille
Curated by ChEMBL
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of recombinant ERAP2 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using R-AMC as substrate preincubated for 30 min...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
Institut Pasteur De Lille
Curated by ChEMBL
Institut Pasteur De Lille
Curated by ChEMBL
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of human ERAP2More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
Institut Pasteur De Lille
Curated by ChEMBL
Institut Pasteur De Lille
Curated by ChEMBL
Affinity DataIC50: 3.70E+4nMAssay Description:Inhibition of human ERAP1More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
Institut Pasteur De Lille
Curated by ChEMBL
Institut Pasteur De Lille
Curated by ChEMBL
Affinity DataIC50: 4.30E+4nMAssay Description:Inhibition of human ERAP1More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
Institut Pasteur De Lille
Curated by ChEMBL
Institut Pasteur De Lille
Curated by ChEMBL
Affinity DataIC50: 8.90E+4nMAssay Description:Inhibition of human ERAP2 assessed as hydrolysis of KSIINFEKL to SIINFEKL measured after 2 hrs by LC-MS analysisMore data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
Institut Pasteur De Lille
Curated by ChEMBL
Institut Pasteur De Lille
Curated by ChEMBL
Affinity DataIC50: 9.80E+4nMAssay Description:Inhibition of human ERAP2 assessed as hydrolysis of KSIINFEKL to SIINFEKL measured after 2 hrs by LC-MS analysisMore data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
Institut Pasteur De Lille
Curated by ChEMBL
Institut Pasteur De Lille
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human ERAP2More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
Institut Pasteur De Lille
Curated by ChEMBL
Institut Pasteur De Lille
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant ERAP2 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using R-AMC as substrate preincubated for 30 min...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
Institut Pasteur De Lille
Curated by ChEMBL
Institut Pasteur De Lille
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant ERAP2 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using R-AMC as substrate preincubated for 30 min...More data for this Ligand-Target Pair
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
Institut Pasteur De Lille
Curated by ChEMBL
Institut Pasteur De Lille
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human IRAP expressed in HEK293 cells using L-AMC as substrate preincubated for 30 mins followed by substrate addition measu...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
Institut Pasteur De Lille
Curated by ChEMBL
Institut Pasteur De Lille
Curated by ChEMBL
Affinity DataIC50: 7.55E+5nMAssay Description:Inhibition of human ERAP2More data for this Ligand-Target Pair