Found 2 Enz. Inhib. hit(s) with Target = 'Endoplasmic reticulum aminopeptidase 2' and Ligand = 'BDBM50570140'
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
Institut Pasteur De Lille
Curated by ChEMBL
Institut Pasteur De Lille
Curated by ChEMBL
Affinity DataIC50: 9.70E+3nMAssay Description:Inhibition of recombinant ERAP2 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using R-AMC as substrate preincubated for 30 min...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
Institut Pasteur De Lille
Curated by ChEMBL
Institut Pasteur De Lille
Curated by ChEMBL
Affinity DataIC50: 9.80E+4nMAssay Description:Inhibition of human ERAP2 assessed as hydrolysis of KSIINFEKL to SIINFEKL measured after 2 hrs by LC-MS analysisMore data for this Ligand-Target Pair