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Target
Mu-type opioid receptor
Ligand
BDBM50027408
Substrate
n/a
Meas. Tech.
ChEBML_147111
IC50
7.2±n/a nM
Citation
 Gacel, G; Fournié-Zaluski, MC; Fellion, E; Roques, BP Evidence of the preferential involvement of mu receptors in analgesia using enkephalins highly selective for peripheral mu or delta receptors. J Med Chem 24:1119-24 (1982) [PubMed]  Article 
Target
Name:
Mu-type opioid receptor
Synonyms:
M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:
Enzyme Catalytic Domain
Mol. Mass.:
11165.58
Organism:
GUINEA PIG
Description:
P97266
Residue:
98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
  
Inhibitor
Name:
BDBM50027408
Synonyms:
2-[1-[1-[1-amino-2-(4-hydroxyphenyl)-(1S)-ethylcarboxamido]-(1S)-ethylcarboxamidomethyl(methyl)carboxamido]-2-phenyl-(1S)-ethylcarboxamido]-4-methylsulfinyl-(2S)-butanoic acid | CHEMBL274204
Type:
Small organic molecule
Emp. Form.:
C29H39N5O8S
Mol. Mass.:
617.714
SMILES:
C[C@H](NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)NCC(=O)N(C)[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCS(C)=O)C(O)=O
Structure:
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