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Target
Similar to alpha-tubulin isoform 1
Ligand
BDBM50081637
Substrate
n/a
Meas. Tech.
ChEMBL_1474254 (CHEMBL3424347)
IC50
7360±n/a nM
Citation
 Stepanov, AI; Astrat'ev, AA; Sheremetev, AB; Lagutina, NK; Palysaeva, NV; Tyurin, AY; Aleksandrova, NS; Sadchikova, NP; Suponitsky, KY; Atamanenko, OP; Konyushkin, LD; Semenov, RV; Firgang, SI; Kiselyov, AS; Semenova, MN; Semenov, VV A facile synthesis and microtubule-destabilizing properties of 4-(1H-benzo[d]imidazol-2-yl)-furazan-3-amines. Eur J Med Chem 94:237-51 (2015) [PubMed]  Article 
Target
Name:
Similar to alpha-tubulin isoform 1
Synonyms:
Similar to alpha-tubulin isoform 1
Type:
PROTEIN
Mol. Mass.:
10383.05
Organism:
Bos taurus
Description:
ChEMBL_104716
Residue:
99
Sequence:
CVSASPSTLARLVSRSAMPAGSSTAWNTAFSPMARCQVTKTIGGGDDSFNTFFSETGAGKHVPRAVFVDLEPTVIDEVRTGTYRSSSTLSSSSQAKKMP
  
Inhibitor
Name:
BDBM50081637
Synonyms:
CHEMBL3422177
Type:
Small organic molecule
Emp. Form.:
C17H13ClN6O2
Mol. Mass.:
368.777
SMILES:
Nc1nonc1-c1nc2ccccc2n1CC(=O)Nc1ccccc1Cl
Structure:
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