Reaction Details Report a problem with these data
Target
Poly [ADP-ribose] polymerase tankyrase-2 [873-1161]
Ligand
BDBM199181
Substrate
n/a
Meas. Tech.
Enzymatic Activity Assay
IC50
>1.00e+5±n/a nM
Citation
Venkannagari, H; Verheugd, P; Koivunen, J; Haikarainen, T; Obaji, E; Ashok, Y; Narwal, M; Pihlajaniemi, T; Lüscher, B; Lehtiö, L Small-Molecule Chemical Probe Rescues Cells from Mono-ADP-Ribosyltransferase ARTD10/PARP10-Induced Apoptosis and Sensitizes Cancer Cells to DNA Damage. Cell Chem Biol 23:1251-1260 (2016) [PubMed] Article
More Info.:
Target
Name:
Poly [ADP-ribose] polymerase tankyrase-2 [873-1161]
Synonyms:
Human diphtheria toxin-like ADP-ribosyltransferase (ARTD6 or PARP5b) | PARP5B | TANK2 | TNKL | TNKS2 | TNKS2_HUMAN
Type:
n/a
Mol. Mass.:
32865.54
Organism:
Homo sapiens (Human)
Description:
Q9H2K2[873-1161]
Residue:
289
Sequence:
GVDFSITQFVRNLGLEHLMDIFEREQITLDVLVEMGHKELKEIGINAYGHRHKLIKGVERLISGQQGLNPYLTLNTSGSGTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMKMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE