Compile Data Set for Download or QSAR
maximum 50k data
Found 8 Enz. Inhib. hit(s) with all data for entry = 3171
LigandPNGBDBM28920((2S,3S)-N-(4-chlorophenyl)-1-hydroxy-3-methylpenta...)
Affinity DataEC50:  5.45E+3nMAssay Description:A Chinese Hamster Ovary cell line stably expressing human beta-APP were aliquoted into a 96-well plate, and after attachment the medium was replaced ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28921((2S,3S)-N-(4-bromophenyl)-1-hydroxy-3-methylpentan...)
Affinity DataEC50:  2.21E+3nMAssay Description:A Chinese Hamster Ovary cell line stably expressing human beta-APP were aliquoted into a 96-well plate, and after attachment the medium was replaced ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28922((2S)-N-(5-chlorothiophen-2-yl)-4,4,4-trifluoro-1-h...)
Affinity DataEC50:  15nMAssay Description:A Chinese Hamster Ovary cell line stably expressing human beta-APP were aliquoted into a 96-well plate, and after attachment the medium was replaced ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28927((2R)-N-(5-chlorothiophen-2-yl)-4,4,4-trifluoro-1-h...)
Affinity DataEC50:  1.07E+4nMAssay Description:A Chinese Hamster Ovary cell line stably expressing human beta-APP were aliquoted into a 96-well plate, and after attachment the medium was replaced ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28924((2S,3S)-N-(5-chlorothiophen-2-yl)-1-hydroxy-3-meth...)
Affinity DataEC50:  297nMAssay Description:A Chinese Hamster Ovary cell line stably expressing human beta-APP were aliquoted into a 96-well plate, and after attachment the medium was replaced ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28925((2S)-N-(5-chlorothiophen-2-yl)-3-ethyl-1-hydroxype...)
Affinity DataEC50:  25nMAssay Description:A Chinese Hamster Ovary cell line stably expressing human beta-APP were aliquoted into a 96-well plate, and after attachment the medium was replaced ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28926((2S)-N-(5-chlorothiophen-2-yl)-5,5,5-trifluoro-1-h...)
Affinity DataEC50:  16nMAssay Description:A Chinese Hamster Ovary cell line stably expressing human beta-APP were aliquoted into a 96-well plate, and after attachment the medium was replaced ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28923((2S)-N-(4-chlorophenyl)-3-ethyl-1-hydroxypentane-2...)
Affinity DataEC50:  294nMAssay Description:A Chinese Hamster Ovary cell line stably expressing human beta-APP were aliquoted into a 96-well plate, and after attachment the medium was replaced ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed