Compile Data Set for Download or QSAR
Report error Found 40 Enz. Inhib. hit(s) with all data for entry = 8689
TargetHistone-lysine N-methyltransferase EHMT2(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 413399BDBM413399(US10407423, Compound 2-06)
Affinity DataIC50: 100nMAssay Description:The biochemical assay to measure G9a enzyme activity relies on time-resolved fluorescence energy transfer (TR-FRET) between europium cryptate (donor)...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase EHMT2(Human)
FundaciÓN Para La InvestigaciÓN MÉDica Aplicada

US Patent
LigandChemical structure of BindingDB Monomer ID 413400BDBM413400(US10407423, Compound 2-07)
Affinity DataIC50: 100nMAssay Description:The biochemical assay to measure G9a enzyme activity relies on time-resolved fluorescence energy transfer (TR-FRET) between europium cryptate (donor)...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase EHMT2(Human)
FundaciÓN Para La InvestigaciÓN MÉDica Aplicada

US Patent
LigandChemical structure of BindingDB Monomer ID 413396BDBM413396(US10407423, Compound 2-03)
Affinity DataIC50: 100nMAssay Description:The biochemical assay to measure G9a enzyme activity relies on time-resolved fluorescence energy transfer (TR-FRET) between europium cryptate (donor)...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase EHMT2(Human)
FundaciÓN Para La InvestigaciÓN MÉDica Aplicada

US Patent
LigandChemical structure of BindingDB Monomer ID 413405BDBM413405(US10407423, Compound 2-12)
Affinity DataIC50: 100nMAssay Description:The biochemical assay to measure G9a enzyme activity relies on time-resolved fluorescence energy transfer (TR-FRET) between europium cryptate (donor)...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase EHMT2(Human)
FundaciÓN Para La InvestigaciÓN MÉDica Aplicada

US Patent
LigandChemical structure of BindingDB Monomer ID 413398BDBM413398(US10407423, Compound 2-05)
Affinity DataIC50: 100nMAssay Description:The biochemical assay to measure G9a enzyme activity relies on time-resolved fluorescence energy transfer (TR-FRET) between europium cryptate (donor)...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase EHMT2(Human)
FundaciÓN Para La InvestigaciÓN MÉDica Aplicada

US Patent
LigandChemical structure of BindingDB Monomer ID 413406BDBM413406(US10407423, Compound 2-13)
Affinity DataIC50: 100nMAssay Description:The biochemical assay to measure G9a enzyme activity relies on time-resolved fluorescence energy transfer (TR-FRET) between europium cryptate (donor)...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase EHMT2(Human)
FundaciÓN Para La InvestigaciÓN MÉDica Aplicada

US Patent
LigandChemical structure of BindingDB Monomer ID 413403BDBM413403(US10407423, Compound 2-10)
Affinity DataIC50: 100nMAssay Description:The biochemical assay to measure G9a enzyme activity relies on time-resolved fluorescence energy transfer (TR-FRET) between europium cryptate (donor)...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase EHMT2(Human)
FundaciÓN Para La InvestigaciÓN MÉDica Aplicada

US Patent
LigandChemical structure of BindingDB Monomer ID 413404BDBM413404(US10407423, Compound 2-11)
Affinity DataIC50: 100nMAssay Description:The biochemical assay to measure G9a enzyme activity relies on time-resolved fluorescence energy transfer (TR-FRET) between europium cryptate (donor)...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase EHMT2(Human)
FundaciÓN Para La InvestigaciÓN MÉDica Aplicada

US Patent
LigandChemical structure of BindingDB Monomer ID 413401BDBM413401(US10407423, Compound 2-08)
Affinity DataIC50: 100nMAssay Description:The biochemical assay to measure G9a enzyme activity relies on time-resolved fluorescence energy transfer (TR-FRET) between europium cryptate (donor)...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase EHMT2(Human)
FundaciÓN Para La InvestigaciÓN MÉDica Aplicada

US Patent
LigandChemical structure of BindingDB Monomer ID 413409BDBM413409(US10407423, Compound 3-03)
Affinity DataIC50: 100nMAssay Description:The biochemical assay to measure G9a enzyme activity relies on time-resolved fluorescence energy transfer (TR-FRET) between europium cryptate (donor)...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase EHMT2(Human)
FundaciÓN Para La InvestigaciÓN MÉDica Aplicada

US Patent
LigandChemical structure of BindingDB Monomer ID 413402BDBM413402(US10407423, Compound 2-09)
Affinity DataIC50: 100nMAssay Description:The biochemical assay to measure G9a enzyme activity relies on time-resolved fluorescence energy transfer (TR-FRET) between europium cryptate (donor)...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
US Patent

TargetDNA (cytosine-5)-methyltransferase 1(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 413391BDBM413391(US10407423, Compound 1-02)
Affinity DataIC50: 300nMAssay Description:The biochemical assay to measure DNMT1 enzyme activity relies on time-resolved fluorescence energy transfer (TR-FRET) between lumi4-Tb (donor) and d2...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase EHMT2(Human)
FundaciÓN Para La InvestigaciÓN MÉDica Aplicada

US Patent
LigandChemical structure of BindingDB Monomer ID 413392BDBM413392(US10407423, Compound 1-03)
Affinity DataIC50: 300nMAssay Description:The biochemical assay to measure G9a enzyme activity relies on time-resolved fluorescence energy transfer (TR-FRET) between europium cryptate (donor)...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
US Patent

TargetDNA (cytosine-5)-methyltransferase 1(Human)
FundaciÓN Para La InvestigaciÓN MÉDica Aplicada

US Patent
LigandChemical structure of BindingDB Monomer ID 413399BDBM413399(US10407423, Compound 2-06)
Affinity DataIC50: 300nMAssay Description:The biochemical assay to measure DNMT1 enzyme activity relies on time-resolved fluorescence energy transfer (TR-FRET) between lumi4-Tb (donor) and d2...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase EHMT2(Human)
FundaciÓN Para La InvestigaciÓN MÉDica Aplicada

US Patent
LigandChemical structure of BindingDB Monomer ID 413408BDBM413408(US10407423, Compound 3-02)
Affinity DataIC50: 300nMAssay Description:The biochemical assay to measure G9a enzyme activity relies on time-resolved fluorescence energy transfer (TR-FRET) between europium cryptate (donor)...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase EHMT2(Human)
FundaciÓN Para La InvestigaciÓN MÉDica Aplicada

US Patent
LigandChemical structure of BindingDB Monomer ID 413391BDBM413391(US10407423, Compound 1-02)
Affinity DataIC50: 300nMAssay Description:The biochemical assay to measure G9a enzyme activity relies on time-resolved fluorescence energy transfer (TR-FRET) between europium cryptate (donor)...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase EHMT2(Human)
FundaciÓN Para La InvestigaciÓN MÉDica Aplicada

US Patent
LigandChemical structure of BindingDB Monomer ID 413393BDBM413393(US10407423, Compound 1-05)
Affinity DataIC50: 300nMAssay Description:The biochemical assay to measure G9a enzyme activity relies on time-resolved fluorescence energy transfer (TR-FRET) between europium cryptate (donor)...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase EHMT2(Human)
FundaciÓN Para La InvestigaciÓN MÉDica Aplicada

US Patent
LigandChemical structure of BindingDB Monomer ID 413410BDBM413410(US10407423, Compound 3-04)
Affinity DataIC50: 300nMAssay Description:The biochemical assay to measure G9a enzyme activity relies on time-resolved fluorescence energy transfer (TR-FRET) between europium cryptate (donor)...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
US Patent

TargetDNA (cytosine-5)-methyltransferase 1(Human)
FundaciÓN Para La InvestigaciÓN MÉDica Aplicada

US Patent
LigandChemical structure of BindingDB Monomer ID 413398BDBM413398(US10407423, Compound 2-05)
Affinity DataIC50: 750nMAssay Description:The biochemical assay to measure DNMT1 enzyme activity relies on time-resolved fluorescence energy transfer (TR-FRET) between lumi4-Tb (donor) and d2...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
US Patent

TargetDNA (cytosine-5)-methyltransferase 1(Human)
FundaciÓN Para La InvestigaciÓN MÉDica Aplicada

US Patent
LigandChemical structure of BindingDB Monomer ID 413392BDBM413392(US10407423, Compound 1-03)
Affinity DataIC50: 750nMAssay Description:The biochemical assay to measure DNMT1 enzyme activity relies on time-resolved fluorescence energy transfer (TR-FRET) between lumi4-Tb (donor) and d2...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
US Patent

TargetDNA (cytosine-5)-methyltransferase 1(Human)
FundaciÓN Para La InvestigaciÓN MÉDica Aplicada

US Patent
LigandChemical structure of BindingDB Monomer ID 413397BDBM413397(US10407423, Compound 2-04)
Affinity DataIC50: 750nMAssay Description:The biochemical assay to measure DNMT1 enzyme activity relies on time-resolved fluorescence energy transfer (TR-FRET) between lumi4-Tb (donor) and d2...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
US Patent

TargetDNA (cytosine-5)-methyltransferase 1(Human)
FundaciÓN Para La InvestigaciÓN MÉDica Aplicada

US Patent
LigandChemical structure of BindingDB Monomer ID 413405BDBM413405(US10407423, Compound 2-12)
Affinity DataIC50: 750nMAssay Description:The biochemical assay to measure DNMT1 enzyme activity relies on time-resolved fluorescence energy transfer (TR-FRET) between lumi4-Tb (donor) and d2...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
US Patent

TargetDNA (cytosine-5)-methyltransferase 1(Human)
FundaciÓN Para La InvestigaciÓN MÉDica Aplicada

US Patent
LigandChemical structure of BindingDB Monomer ID 413402BDBM413402(US10407423, Compound 2-09)
Affinity DataIC50: 750nMAssay Description:The biochemical assay to measure DNMT1 enzyme activity relies on time-resolved fluorescence energy transfer (TR-FRET) between lumi4-Tb (donor) and d2...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
US Patent

TargetDNA (cytosine-5)-methyltransferase 1(Human)
FundaciÓN Para La InvestigaciÓN MÉDica Aplicada

US Patent
LigandChemical structure of BindingDB Monomer ID 413403BDBM413403(US10407423, Compound 2-10)
Affinity DataIC50: 750nMAssay Description:The biochemical assay to measure DNMT1 enzyme activity relies on time-resolved fluorescence energy transfer (TR-FRET) between lumi4-Tb (donor) and d2...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
US Patent

TargetDNA (cytosine-5)-methyltransferase 1(Human)
FundaciÓN Para La InvestigaciÓN MÉDica Aplicada

US Patent
LigandChemical structure of BindingDB Monomer ID 413395BDBM413395(US10407423, Compound 2-02)
Affinity DataIC50: 750nMAssay Description:The biochemical assay to measure DNMT1 enzyme activity relies on time-resolved fluorescence energy transfer (TR-FRET) between lumi4-Tb (donor) and d2...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
US Patent

TargetDNA (cytosine-5)-methyltransferase 1(Human)
FundaciÓN Para La InvestigaciÓN MÉDica Aplicada

US Patent
LigandChemical structure of BindingDB Monomer ID 413400BDBM413400(US10407423, Compound 2-07)
Affinity DataIC50: 750nMAssay Description:The biochemical assay to measure DNMT1 enzyme activity relies on time-resolved fluorescence energy transfer (TR-FRET) between lumi4-Tb (donor) and d2...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
US Patent

TargetDNA (cytosine-5)-methyltransferase 1(Human)
FundaciÓN Para La InvestigaciÓN MÉDica Aplicada

US Patent
LigandChemical structure of BindingDB Monomer ID 413408BDBM413408(US10407423, Compound 3-02)
Affinity DataIC50: 750nMAssay Description:The biochemical assay to measure DNMT1 enzyme activity relies on time-resolved fluorescence energy transfer (TR-FRET) between lumi4-Tb (donor) and d2...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
US Patent

TargetDNA (cytosine-5)-methyltransferase 1(Human)
FundaciÓN Para La InvestigaciÓN MÉDica Aplicada

US Patent
LigandChemical structure of BindingDB Monomer ID 413393BDBM413393(US10407423, Compound 1-05)
Affinity DataIC50: 750nMAssay Description:The biochemical assay to measure DNMT1 enzyme activity relies on time-resolved fluorescence energy transfer (TR-FRET) between lumi4-Tb (donor) and d2...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
US Patent

TargetDNA (cytosine-5)-methyltransferase 1(Human)
FundaciÓN Para La InvestigaciÓN MÉDica Aplicada

US Patent
LigandChemical structure of BindingDB Monomer ID 413401BDBM413401(US10407423, Compound 2-08)
Affinity DataIC50: 750nMAssay Description:The biochemical assay to measure DNMT1 enzyme activity relies on time-resolved fluorescence energy transfer (TR-FRET) between lumi4-Tb (donor) and d2...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
US Patent

TargetDNA (cytosine-5)-methyltransferase 1(Human)
FundaciÓN Para La InvestigaciÓN MÉDica Aplicada

US Patent
LigandChemical structure of BindingDB Monomer ID 413406BDBM413406(US10407423, Compound 2-13)
Affinity DataIC50: 5.50E+3nMAssay Description:The biochemical assay to measure DNMT1 enzyme activity relies on time-resolved fluorescence energy transfer (TR-FRET) between lumi4-Tb (donor) and d2...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase EHMT2(Human)
FundaciÓN Para La InvestigaciÓN MÉDica Aplicada

US Patent
LigandChemical structure of BindingDB Monomer ID 413407BDBM413407(US10407423, Compound 3-01)
Affinity DataIC50: 5.50E+3nMAssay Description:The biochemical assay to measure G9a enzyme activity relies on time-resolved fluorescence energy transfer (TR-FRET) between europium cryptate (donor)...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
US Patent

TargetDNA (cytosine-5)-methyltransferase 1(Human)
FundaciÓN Para La InvestigaciÓN MÉDica Aplicada

US Patent
LigandChemical structure of BindingDB Monomer ID 413407BDBM413407(US10407423, Compound 3-01)
Affinity DataIC50: 5.50E+3nMAssay Description:The biochemical assay to measure DNMT1 enzyme activity relies on time-resolved fluorescence energy transfer (TR-FRET) between lumi4-Tb (donor) and d2...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
US Patent

TargetDNA (cytosine-5)-methyltransferase 1(Human)
FundaciÓN Para La InvestigaciÓN MÉDica Aplicada

US Patent
LigandChemical structure of BindingDB Monomer ID 413404BDBM413404(US10407423, Compound 2-11)
Affinity DataIC50: 5.50E+3nMAssay Description:The biochemical assay to measure DNMT1 enzyme activity relies on time-resolved fluorescence energy transfer (TR-FRET) between lumi4-Tb (donor) and d2...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
US Patent

TargetDNA (cytosine-5)-methyltransferase 1(Human)
FundaciÓN Para La InvestigaciÓN MÉDica Aplicada

US Patent
LigandChemical structure of BindingDB Monomer ID 413396BDBM413396(US10407423, Compound 2-03)
Affinity DataIC50: 5.50E+3nMAssay Description:The biochemical assay to measure DNMT1 enzyme activity relies on time-resolved fluorescence energy transfer (TR-FRET) between lumi4-Tb (donor) and d2...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
US Patent

TargetDNA (cytosine-5)-methyltransferase 1(Human)
FundaciÓN Para La InvestigaciÓN MÉDica Aplicada

US Patent
LigandChemical structure of BindingDB Monomer ID 413411BDBM413411(US10407423, Compound 4-03)
Affinity DataIC50: 5.50E+3nMAssay Description:The biochemical assay to measure DNMT1 enzyme activity relies on time-resolved fluorescence energy transfer (TR-FRET) between lumi4-Tb (donor) and d2...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
US Patent

TargetDNA (cytosine-5)-methyltransferase 1(Human)
FundaciÓN Para La InvestigaciÓN MÉDica Aplicada

US Patent
LigandChemical structure of BindingDB Monomer ID 413394BDBM413394(US10407423, Compound 2-01)
Affinity DataIC50: 5.50E+3nMAssay Description:The biochemical assay to measure DNMT1 enzyme activity relies on time-resolved fluorescence energy transfer (TR-FRET) between lumi4-Tb (donor) and d2...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
US Patent

TargetDNA (cytosine-5)-methyltransferase 1(Human)
FundaciÓN Para La InvestigaciÓN MÉDica Aplicada

US Patent
LigandChemical structure of BindingDB Monomer ID 413412BDBM413412(US10407423, Compound 4-04)
Affinity DataIC50: 5.50E+3nMAssay Description:The biochemical assay to measure DNMT1 enzyme activity relies on time-resolved fluorescence energy transfer (TR-FRET) between lumi4-Tb (donor) and d2...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase EHMT2(Human)
FundaciÓN Para La InvestigaciÓN MÉDica Aplicada

US Patent
LigandChemical structure of BindingDB Monomer ID 413395BDBM413395(US10407423, Compound 2-02)
Affinity DataIC50: 5.50E+3nMAssay Description:The biochemical assay to measure G9a enzyme activity relies on time-resolved fluorescence energy transfer (TR-FRET) between europium cryptate (donor)...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
US Patent

TargetDNA (cytosine-5)-methyltransferase 1(Human)
FundaciÓN Para La InvestigaciÓN MÉDica Aplicada

US Patent
LigandChemical structure of BindingDB Monomer ID 413413BDBM413413(US10407423, Compound 4-05)
Affinity DataIC50: 5.50E+3nMAssay Description:The biochemical assay to measure DNMT1 enzyme activity relies on time-resolved fluorescence energy transfer (TR-FRET) between lumi4-Tb (donor) and d2...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
US Patent

TargetDNA (cytosine-5)-methyltransferase 1(Human)
FundaciÓN Para La InvestigaciÓN MÉDica Aplicada

US Patent
LigandChemical structure of BindingDB Monomer ID 413409BDBM413409(US10407423, Compound 3-03)
Affinity DataIC50: 5.50E+3nMAssay Description:The biochemical assay to measure DNMT1 enzyme activity relies on time-resolved fluorescence energy transfer (TR-FRET) between lumi4-Tb (donor) and d2...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
US Patent