Compile Data Set for Download or QSAR
Report error Found 837 Enz. Inhib. hit(s) with all data for entry = 9965
LigandChemical structure of BindingDB Monomer ID 500349BDBM500349(US11021481, Compound I-6 | 7-[[5-(4- methylpiperaz...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500370BDBM500370(US11021481, Compound I-28 | 4-(6-methoxy- 1H-indol...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500371BDBM500371(US11021481, Compound I-29 | 7-[[5-(4- methylpipera...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500373BDBM500373(US11021481, Compound I-31 | 7-[[5-(4- methylpipera...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500374BDBM500374(US11021481, Compound I-32 | 4-(6-fluoro- 1H-indol-...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500375BDBM500375(US11021481, Compound I-33 | 7-[[5-(4- methylpipera...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500376BDBM500376(US11021481, Compound I-34 | 4-(2-ethyl-1H- indol-3...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500379BDBM500379(US11021481, Compound I-37 | 7-[[5-(4-methylpiperaz...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500380BDBM500380(US11021481, Compound I-38 | 7-[[5-(4- methylpipera...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500381BDBM500381(US11021481, Compound I-39 | 4-imidazo[1,2- a]pyrid...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500382BDBM500382(US11021481, Compound I-40 | 7-[[5-(4-methylpiperaz...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500383BDBM500383(US11021481, Compound I-41 | 4-(1H-indol-4- yl)-7-[...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500384BDBM500384(US11021481, Compound I-42 | 7-[[5-(4- methylpipera...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500385BDBM500385(4-(1-methylpyrrolo] 2,3-b]pyridin- 4-yl)-7-[(5- pi...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500360BDBM500360(US11021481, Compound I-18 | 7-[[5-(4- methylpipera...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500361BDBM500361(US11021481, Compound I-19 | 7-[[5-(4- methylpipera...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500362BDBM500362(US11021481, Compound I-20 | 7-[[5-(4- methylpipera...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500363BDBM500363(US11021481, Compound I-21 | 7-[[5-(4- methylpipera...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500366BDBM500366(US11021481, Compound I-24 | 7-[[5-(4- methylpipera...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500403BDBM500403(US11021481, Compound I-62 | 7-[[5-[4- (methylamino...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500404BDBM500404(US11021481, Compound I-63 | 4-imidazo[1,2- a]pyrid...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500405BDBM500405(US11548890, Compound I-64 | US11021481, Compound I...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500406BDBM500406(US11021481, Compound I-65 | 7-[[5-(4- methylpipera...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500408BDBM500408(US11021481, Compound I-67 | 4-(5-fluoro-1- methyl-...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500409BDBM500409(US11021481, Compound I-68 | 4-(2,3- dihydro-1H- py...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500410BDBM500410(US11021481, Compound I-69 | 7-[[5-(4- methylpipera...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500411BDBM500411(US11021481, Compound I-70 | 7-[[5-(3,8- diazabicyc...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500412BDBM500412(US11021481, Compound I-71 | 7-[[5-[4- (methylamino...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500413BDBM500413(4-(7-methylimidazo [1,2-a]pyridin- 3-yl)-7-[(5- pi...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500414BDBM500414(US11021481, Compound I-73 | 4-(7- methylimidazo [1...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500415BDBM500415(US11021481, Compound I-74 | 3-[7-[[5-(4- methylpip...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500416BDBM500416(US11021481, Compound I-75 | 7-[[5-(4- hydroxy-1- p...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500417BDBM500417(US11021481, Compound I-76 | 4-imidazo[1,2- a]pyraz...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500387BDBM500387(US11021481, Compound I-45 | 7-[[5-(4-methylpiperaz...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500388BDBM500388(US11021481, Compound I-46 | 4-(1H-indol-3- yl)-7-[...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500389BDBM500389(US11021481, Compound I-47 | 4-[1-(2-methoxyethyl) ...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500391BDBM500391(US11021481, Compound I-49 | 4-(1-ethylpyrrolo]2,3-...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500393BDBM500393(US11021481, Compound I-51 | 4-(6- methylimidazo [1...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500394BDBM500394(US11021481, Compound I-52 | 4-(8-methylimidazo [1,...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500396BDBM500396(US11021481, Compound I-55 | 7-[[5-(4- methylpipera...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500397BDBM500397(US11021481, Compound I-56 | 4-imidazo[1,2- a]pyrid...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500398BDBM500398(US11021481, Compound I-57 | 7-[[5-[4- (methylamino...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500399BDBM500399(US11021481, Compound I-58 | 4-imidazo[1,2- a]pyrid...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500400BDBM500400(US11021481, Compound I-59 | 4-imidazo[1,2- b]pyrid...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500401BDBM500401(US11021481, Compound I-60 | 4-imidazo[1,2- a]pyrid...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 502240BDBM502240(US11028085, Compound I-93 | US11078201, Compound I...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500435BDBM500435(US11021481, Compound I-94 | 7-[[5-[(3S)-3- amino-1...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500436BDBM500436(US11021481, Compound I-95 | 7-[[5-[(3R)-3- amino-1...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 502243BDBM502243(US11028085, Compound I-96 | US11548890, Compound I...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 500438BDBM500438(US11021481, Compound I-97 | 7-[[5-[(3S)-3- (methyl...)
Affinity DataIC50: 100nMAssay Description:HPK1 biochemical enzyme assay: HPK1 enzyme inhibition was measured using a microfluidic mobility shift assay. Reactions were performed in a 384-well ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

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