Compile Data Set for Download or QSAR
maximum 50k data
Found 14 Enz. Inhib. hit(s) with all data for entry = 10663
TargetBromodomain-containing protein 4 [49-170](Homo sapiens (Human))
Epigenetix

US Patent
LigandPNGBDBM449849(5-[2-cyclobutyl-3-[2-(trifluoromethoxy)ethyl]benzi...)
Affinity DataIC50:  91nMAssay Description:To measure activity of bromodomain inhibitors, a His-epitope tagged BRD4 BD149-170 is purchased from BPS Bioscience. BRD4 binding and inhibition is a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 4 [49-170](Homo sapiens (Human))
Epigenetix

US Patent
LigandPNGBDBM449854(5-[3-[(1R)-2-methoxy-1-methyl-ethyl]-2-methyl-benz...)
Affinity DataIC50:  98nMAssay Description:To measure activity of bromodomain inhibitors, a His-epitope tagged BRD4 BD149-170 is purchased from BPS Bioscience. BRD4 binding and inhibition is a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 4 [49-170](Homo sapiens (Human))
Epigenetix

US Patent
LigandPNGBDBM449853(5-[3-[(1R)-2-methoxy-1-methyl-ethyl]-2-tetrahydrop...)
Affinity DataIC50:  99nMAssay Description:To measure activity of bromodomain inhibitors, a His-epitope tagged BRD4 BD149-170 is purchased from BPS Bioscience. BRD4 binding and inhibition is a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 4 [49-170](Homo sapiens (Human))
Epigenetix

US Patent
LigandPNGBDBM449857(5-[2-cyclopropyl-3-[(1R)-2-methoxy-1-methylethyl]b...)
Affinity DataIC50:  100nMAssay Description:To measure activity of bromodomain inhibitors, a His-epitope tagged BRD4 BD149-170 is purchased from BPS Bioscience. BRD4 binding and inhibition is a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 4 [49-170](Homo sapiens (Human))
Epigenetix

US Patent
LigandPNGBDBM449847(5-[2-(1-acetyl-4-piperidyl)-3-[2-(trifluoromethoxy...)
Affinity DataIC50:  130nMAssay Description:To measure activity of bromodomain inhibitors, a His-epitope tagged BRD4 BD149-170 is purchased from BPS Bioscience. BRD4 binding and inhibition is a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 4 [49-170](Homo sapiens (Human))
Epigenetix

US Patent
LigandPNGBDBM449844(1,3-dimethyl-5-[2-tetrahydropyran-4-yl-3-[2-(trifl...)
Affinity DataIC50:  140nMAssay Description:To measure activity of bromodomain inhibitors, a His-epitope tagged BRD4 BD149-170 is purchased from BPS Bioscience. BRD4 binding and inhibition is a...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4 [49-170](Homo sapiens (Human))
Epigenetix

US Patent
LigandPNGBDBM449845(5-[2-cyclopropyl-3-[2-(trifluoromethoxy)ethyl]benz...)
Affinity DataIC50:  190nMAssay Description:To measure activity of bromodomain inhibitors, a His-epitope tagged BRD4 BD149-170 is purchased from BPS Bioscience. BRD4 binding and inhibition is a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 4 [49-170](Homo sapiens (Human))
Epigenetix

US Patent
LigandPNGBDBM449848(1,3-dimethyl-5-[2-methyl-3-[2-(trifluoromethoxy)et...)
Affinity DataIC50:  190nMAssay Description:To measure activity of bromodomain inhibitors, a His-epitope tagged BRD4 BD149-170 is purchased from BPS Bioscience. BRD4 binding and inhibition is a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 4 [49-170](Homo sapiens (Human))
Epigenetix

US Patent
LigandPNGBDBM449851(5-[3-(2-methoxyethyl)-2-methyl-benzimidazol-5-yl]-...)
Affinity DataIC50:  210nMAssay Description:To measure activity of bromodomain inhibitors, a His-epitope tagged BRD4 BD149-170 is purchased from BPS Bioscience. BRD4 binding and inhibition is a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 4 [49-170](Homo sapiens (Human))
Epigenetix

US Patent
LigandPNGBDBM449852(5-[3-(2-methoxyethyl)-2-tetrahydropyran-4-yl-benzi...)
Affinity DataIC50:  220nMAssay Description:To measure activity of bromodomain inhibitors, a His-epitope tagged BRD4 BD149-170 is purchased from BPS Bioscience. BRD4 binding and inhibition is a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 4 [49-170](Homo sapiens (Human))
Epigenetix

US Patent
LigandPNGBDBM449850(5-[2-cyclopropyl-3-(2-methoxyethyl)benzimidazol-5-...)
Affinity DataIC50:  280nMAssay Description:To measure activity of bromodomain inhibitors, a His-epitope tagged BRD4 BD149-170 is purchased from BPS Bioscience. BRD4 binding and inhibition is a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 4 [49-170](Homo sapiens (Human))
Epigenetix

US Patent
LigandPNGBDBM449846(1,3-dimethyl-5-[3-[2-(trifluoromethoxy)ethyl]benzi...)
Affinity DataIC50:  310nMAssay Description:To measure activity of bromodomain inhibitors, a His-epitope tagged BRD4 BD149-170 is purchased from BPS Bioscience. BRD4 binding and inhibition is a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 4 [49-170](Homo sapiens (Human))
Epigenetix

US Patent
LigandPNGBDBM449855(5-[3-[(1R)-2-methoxy-1-methyl-ethyl]benzimidazol-5...)
Affinity DataIC50:  330nMAssay Description:To measure activity of bromodomain inhibitors, a His-epitope tagged BRD4 BD149-170 is purchased from BPS Bioscience. BRD4 binding and inhibition is a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 4 [49-170](Homo sapiens (Human))
Epigenetix

US Patent
LigandPNGBDBM557859(5-[2-cyclopropyl-3-[2-(trifluoromethoxy)ethyl]benz...)
Affinity DataIC50:  810nMAssay Description:To measure activity of bromodomain inhibitors, a His-epitope tagged BRD4 BD149-170 is purchased from BPS Bioscience. BRD4 binding and inhibition is a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent