Compile Data Set for Download or QSAR
Report error Found 38 Enz. Inhib. hit(s) with all data for entry = 12537
TargetTyrosine-protein kinase BTK(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 708087BDBM708087(US12172992, Example 3)
Affinity DataIC50: 0.0340nMAssay Description:Btk kinase activity was measured in vitro using an electrophoretic mobility shift assay (MSA). The ability of Btk to phosphorylate a fluorescent pept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 708096BDBM708096(US12172992, Example 12)
Affinity DataIC50: 0.0360nMAssay Description:Btk kinase activity was measured in vitro using an electrophoretic mobility shift assay (MSA). The ability of Btk to phosphorylate a fluorescent pept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 708090BDBM708090(US12172992, Example 6)
Affinity DataIC50: 0.0400nMAssay Description:Btk kinase activity was measured in vitro using an electrophoretic mobility shift assay (MSA). The ability of Btk to phosphorylate a fluorescent pept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 708098BDBM708098(US12172992, Example 14)
Affinity DataIC50: 0.0530nMAssay Description:Btk kinase activity was measured in vitro using an electrophoretic mobility shift assay (MSA). The ability of Btk to phosphorylate a fluorescent pept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 708092BDBM708092(US12172992, Example 8)
Affinity DataIC50: 0.0800nMAssay Description:Btk kinase activity was measured in vitro using an electrophoretic mobility shift assay (MSA). The ability of Btk to phosphorylate a fluorescent pept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 708095BDBM708095(US12172992, Example 11)
Affinity DataIC50: 0.0970nMAssay Description:Btk kinase activity was measured in vitro using an electrophoretic mobility shift assay (MSA). The ability of Btk to phosphorylate a fluorescent pept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 708091BDBM708091(US12172992, Example 7)
Affinity DataIC50: 0.0980nMAssay Description:Btk kinase activity was measured in vitro using an electrophoretic mobility shift assay (MSA). The ability of Btk to phosphorylate a fluorescent pept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 708085BDBM708085(US12172992, Example 1)
Affinity DataIC50: 0.0980nMAssay Description:Btk kinase activity was measured in vitro using an electrophoretic mobility shift assay (MSA). The ability of Btk to phosphorylate a fluorescent pept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 708099BDBM708099(US12172992, Example 15)
Affinity DataIC50: 0.0990nMAssay Description:Btk kinase activity was measured in vitro using an electrophoretic mobility shift assay (MSA). The ability of Btk to phosphorylate a fluorescent pept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 708093BDBM708093(US12172992, Example 9)
Affinity DataIC50: 0.0990nMAssay Description:Btk kinase activity was measured in vitro using an electrophoretic mobility shift assay (MSA). The ability of Btk to phosphorylate a fluorescent pept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 708103BDBM708103(US12172992, Example 19)
Affinity DataIC50: 0.100nMAssay Description:Btk kinase activity was measured in vitro using an electrophoretic mobility shift assay (MSA). The ability of Btk to phosphorylate a fluorescent pept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 708101BDBM708101(US12172992, Example 17)
Affinity DataIC50: 0.103nMAssay Description:Btk kinase activity was measured in vitro using an electrophoretic mobility shift assay (MSA). The ability of Btk to phosphorylate a fluorescent pept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 708094BDBM708094(US12172992, Example 10)
Affinity DataIC50: 0.106nMAssay Description:Btk kinase activity was measured in vitro using an electrophoretic mobility shift assay (MSA). The ability of Btk to phosphorylate a fluorescent pept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 708089BDBM708089(US12172992, Example 5)
Affinity DataIC50: 0.113nMAssay Description:Btk kinase activity was measured in vitro using an electrophoretic mobility shift assay (MSA). The ability of Btk to phosphorylate a fluorescent pept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 708086BDBM708086(US12172992, Example 2)
Affinity DataIC50: 0.128nMAssay Description:Btk kinase activity was measured in vitro using an electrophoretic mobility shift assay (MSA). The ability of Btk to phosphorylate a fluorescent pept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 708097BDBM708097(US12172992, Example 13)
Affinity DataIC50: 0.140nMAssay Description:Btk kinase activity was measured in vitro using an electrophoretic mobility shift assay (MSA). The ability of Btk to phosphorylate a fluorescent pept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 708088BDBM708088(US12172992, Example 4)
Affinity DataIC50: 0.141nMAssay Description:Btk kinase activity was measured in vitro using an electrophoretic mobility shift assay (MSA). The ability of Btk to phosphorylate a fluorescent pept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 708100BDBM708100(US12172992, Example 16)
Affinity DataIC50: 0.438nMAssay Description:Btk kinase activity was measured in vitro using an electrophoretic mobility shift assay (MSA). The ability of Btk to phosphorylate a fluorescent pept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 708102BDBM708102(US12172992, Example 18)
Affinity DataIC50: 0.496nMAssay Description:Btk kinase activity was measured in vitro using an electrophoretic mobility shift assay (MSA). The ability of Btk to phosphorylate a fluorescent pept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
US Patent

TargetProtein cereblon(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 708090BDBM708090(US12172992, Example 6)
Affinity DataIC50: 378nMAssay Description:Competition Assay: Test compounds in 100% dimethyl sulfoxide were plated onto white, low volume 384 well plates (PerkinElmer Proxiplate 384 plus #600...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
US Patent

TargetProtein cereblon(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 708091BDBM708091(US12172992, Example 7)
Affinity DataIC50: 609nMAssay Description:Competition Assay: Test compounds in 100% dimethyl sulfoxide were plated onto white, low volume 384 well plates (PerkinElmer Proxiplate 384 plus #600...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
US Patent

TargetProtein cereblon(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 708089BDBM708089(US12172992, Example 5)
Affinity DataIC50: 648nMAssay Description:Competition Assay: Test compounds in 100% dimethyl sulfoxide were plated onto white, low volume 384 well plates (PerkinElmer Proxiplate 384 plus #600...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
US Patent

TargetProtein cereblon(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 708093BDBM708093(US12172992, Example 9)
Affinity DataIC50: 658nMAssay Description:Competition Assay: Test compounds in 100% dimethyl sulfoxide were plated onto white, low volume 384 well plates (PerkinElmer Proxiplate 384 plus #600...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
US Patent

TargetProtein cereblon(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 708086BDBM708086(US12172992, Example 2)
Affinity DataIC50: 749nMAssay Description:Competition Assay: Test compounds in 100% dimethyl sulfoxide were plated onto white, low volume 384 well plates (PerkinElmer Proxiplate 384 plus #600...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
US Patent

TargetProtein cereblon(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 708102BDBM708102(US12172992, Example 18)
Affinity DataIC50: 1.25E+3nMAssay Description:Competition Assay: Test compounds in 100% dimethyl sulfoxide were plated onto white, low volume 384 well plates (PerkinElmer Proxiplate 384 plus #600...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
US Patent

TargetProtein cereblon(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 708085BDBM708085(US12172992, Example 1)
Affinity DataIC50: 1.26E+3nMAssay Description:Competition Assay: Test compounds in 100% dimethyl sulfoxide were plated onto white, low volume 384 well plates (PerkinElmer Proxiplate 384 plus #600...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
US Patent

TargetProtein cereblon(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 708096BDBM708096(US12172992, Example 12)
Affinity DataIC50: 2.01E+3nMAssay Description:Competition Assay: Test compounds in 100% dimethyl sulfoxide were plated onto white, low volume 384 well plates (PerkinElmer Proxiplate 384 plus #600...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
US Patent

TargetProtein cereblon(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 708095BDBM708095(US12172992, Example 11)
Affinity DataIC50: 2.15E+3nMAssay Description:Competition Assay: Test compounds in 100% dimethyl sulfoxide were plated onto white, low volume 384 well plates (PerkinElmer Proxiplate 384 plus #600...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
US Patent

TargetProtein cereblon(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 708098BDBM708098(US12172992, Example 14)
Affinity DataIC50: 2.33E+3nMAssay Description:Competition Assay: Test compounds in 100% dimethyl sulfoxide were plated onto white, low volume 384 well plates (PerkinElmer Proxiplate 384 plus #600...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
US Patent

TargetProtein cereblon(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 708092BDBM708092(US12172992, Example 8)
Affinity DataIC50: 3.38E+3nMAssay Description:Competition Assay: Test compounds in 100% dimethyl sulfoxide were plated onto white, low volume 384 well plates (PerkinElmer Proxiplate 384 plus #600...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
US Patent

TargetProtein cereblon(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 708101BDBM708101(US12172992, Example 17)
Affinity DataIC50: 3.87E+3nMAssay Description:Competition Assay: Test compounds in 100% dimethyl sulfoxide were plated onto white, low volume 384 well plates (PerkinElmer Proxiplate 384 plus #600...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
US Patent

TargetProtein cereblon(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 708094BDBM708094(US12172992, Example 10)
Affinity DataIC50: 6.31E+3nMAssay Description:Competition Assay: Test compounds in 100% dimethyl sulfoxide were plated onto white, low volume 384 well plates (PerkinElmer Proxiplate 384 plus #600...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
US Patent

TargetProtein cereblon(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 708087BDBM708087(US12172992, Example 3)
Affinity DataIC50: 9.57E+3nMAssay Description:Competition Assay: Test compounds in 100% dimethyl sulfoxide were plated onto white, low volume 384 well plates (PerkinElmer Proxiplate 384 plus #600...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
US Patent

TargetProtein cereblon(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 708100BDBM708100(US12172992, Example 16)
Affinity DataIC50: 1.00E+4nMAssay Description:Competition Assay: Test compounds in 100% dimethyl sulfoxide were plated onto white, low volume 384 well plates (PerkinElmer Proxiplate 384 plus #600...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
US Patent

TargetProtein cereblon(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 708099BDBM708099(US12172992, Example 15)
Affinity DataIC50: 1.00E+4nMAssay Description:Competition Assay: Test compounds in 100% dimethyl sulfoxide were plated onto white, low volume 384 well plates (PerkinElmer Proxiplate 384 plus #600...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
US Patent

TargetProtein cereblon(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 708097BDBM708097(US12172992, Example 13)
Affinity DataIC50: 1.00E+4nMAssay Description:Competition Assay: Test compounds in 100% dimethyl sulfoxide were plated onto white, low volume 384 well plates (PerkinElmer Proxiplate 384 plus #600...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
US Patent

TargetProtein cereblon(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 708088BDBM708088(US12172992, Example 4)
Affinity DataIC50: 1.00E+4nMAssay Description:Competition Assay: Test compounds in 100% dimethyl sulfoxide were plated onto white, low volume 384 well plates (PerkinElmer Proxiplate 384 plus #600...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
US Patent

TargetProtein cereblon(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 708103BDBM708103(US12172992, Example 19)
Affinity DataIC50: 1.00E+4nMAssay Description:Competition Assay: Test compounds in 100% dimethyl sulfoxide were plated onto white, low volume 384 well plates (PerkinElmer Proxiplate 384 plus #600...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
US Patent