Compile Data Set for Download or QSAR
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 12122
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Cold Spring Harbor Laboratory

US Patent
LigandChemical structure of BindingDB Monomer ID 681331BDBM681331(US20240199561, Compound FC-2)
Affinity DataIC50: 19nMAssay Description:The ADP-GloTM Kinase Assay kit from Promega was used to screen the compounds before determination of their IC50 using the radiolabeled kinase assay. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Cold Spring Harbor Laboratory

US Patent
LigandChemical structure of BindingDB Monomer ID 681332BDBM681332(US20240199561, Compound FC-3)
Affinity DataIC50: 53nMAssay Description:The ADP-GloTM Kinase Assay kit from Promega was used to screen the compounds before determination of their IC50 using the radiolabeled kinase assay. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Cold Spring Harbor Laboratory

US Patent
LigandChemical structure of BindingDB Monomer ID 681345BDBM681345(US20240199561, Compound FC-204)
Affinity DataIC50: 57nMAssay Description:The ADP-GloTM Kinase Assay kit from Promega was used to screen the compounds before determination of their IC50 using the radiolabeled kinase assay. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Cold Spring Harbor Laboratory

US Patent
LigandChemical structure of BindingDB Monomer ID 681333BDBM681333(US20240199561, Compound FC-4)
Affinity DataIC50: 87nMAssay Description:The ADP-GloTM Kinase Assay kit from Promega was used to screen the compounds before determination of their IC50 using the radiolabeled kinase assay. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Cold Spring Harbor Laboratory

US Patent
LigandChemical structure of BindingDB Monomer ID 681334BDBM681334(US20240199561, Compound FC-5)
Affinity DataIC50: 95nMAssay Description:The ADP-GloTM Kinase Assay kit from Promega was used to screen the compounds before determination of their IC50 using the radiolabeled kinase assay. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Cold Spring Harbor Laboratory

US Patent
LigandChemical structure of BindingDB Monomer ID 681339BDBM681339(US20240199561, Compound FC-10)
Affinity DataIC50: 110nMAssay Description:The ADP-GloTM Kinase Assay kit from Promega was used to screen the compounds before determination of their IC50 using the radiolabeled kinase assay. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Cold Spring Harbor Laboratory

US Patent
LigandChemical structure of BindingDB Monomer ID 681334BDBM681334(US20240199561, Compound FC-5)
Affinity DataIC50: 144nMAssay Description:The ADP-GloTM Kinase Assay kit from Promega was used to screen the compounds before determination of their IC50 using the radiolabeled kinase assay. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Cold Spring Harbor Laboratory

US Patent
LigandChemical structure of BindingDB Monomer ID 681333BDBM681333(US20240199561, Compound FC-4)
Affinity DataIC50: 174nMAssay Description:The ADP-GloTM Kinase Assay kit from Promega was used to screen the compounds before determination of their IC50 using the radiolabeled kinase assay. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Cold Spring Harbor Laboratory

US Patent
LigandChemical structure of BindingDB Monomer ID 681335BDBM681335(US20240199561, Compound FC-6)
Affinity DataIC50: 180nMAssay Description:The ADP-GloTM Kinase Assay kit from Promega was used to screen the compounds before determination of their IC50 using the radiolabeled kinase assay. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Cold Spring Harbor Laboratory

US Patent
LigandChemical structure of BindingDB Monomer ID 681346BDBM681346(US20240199561, Compound FC-205)
Affinity DataIC50: 206nMAssay Description:The ADP-GloTM Kinase Assay kit from Promega was used to screen the compounds before determination of their IC50 using the radiolabeled kinase assay. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Cold Spring Harbor Laboratory

US Patent
LigandChemical structure of BindingDB Monomer ID 681336BDBM681336(US20240199561, Compound FC-7)
Affinity DataIC50: 229nMAssay Description:The ADP-GloTM Kinase Assay kit from Promega was used to screen the compounds before determination of their IC50 using the radiolabeled kinase assay. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Cold Spring Harbor Laboratory

US Patent
LigandChemical structure of BindingDB Monomer ID 681341BDBM681341(US20240199561, Compound FC-63)
Affinity DataIC50: 238nMAssay Description:The ADP-GloTM Kinase Assay kit from Promega was used to screen the compounds before determination of their IC50 using the radiolabeled kinase assay. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Cold Spring Harbor Laboratory

US Patent
LigandChemical structure of BindingDB Monomer ID 681338BDBM681338(US20240199561, Compound FC-8)
Affinity DataIC50: 238nMAssay Description:The ADP-GloTM Kinase Assay kit from Promega was used to screen the compounds before determination of their IC50 using the radiolabeled kinase assay. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Cold Spring Harbor Laboratory

US Patent
LigandChemical structure of BindingDB Monomer ID 681338BDBM681338(US20240199561, Compound FC-8)
Affinity DataIC50: 317nMAssay Description:The ADP-GloTM Kinase Assay kit from Promega was used to screen the compounds before determination of their IC50 using the radiolabeled kinase assay. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Cold Spring Harbor Laboratory

US Patent
LigandChemical structure of BindingDB Monomer ID 681340BDBM681340(US20240199561, Compound FC-14)
Affinity DataIC50: 400nMAssay Description:The ADP-GloTM Kinase Assay kit from Promega was used to screen the compounds before determination of their IC50 using the radiolabeled kinase assay. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Cold Spring Harbor Laboratory

US Patent
LigandChemical structure of BindingDB Monomer ID 681343BDBM681343(US20240199561, Compound FC-195)
Affinity DataIC50: 420nMAssay Description:The ADP-GloTM Kinase Assay kit from Promega was used to screen the compounds before determination of their IC50 using the radiolabeled kinase assay. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Cold Spring Harbor Laboratory

US Patent
LigandChemical structure of BindingDB Monomer ID 681344BDBM681344(US20240199561, Compound FC-196)
Affinity DataIC50: 500nMAssay Description:The ADP-GloTM Kinase Assay kit from Promega was used to screen the compounds before determination of their IC50 using the radiolabeled kinase assay. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Cold Spring Harbor Laboratory

US Patent
LigandChemical structure of BindingDB Monomer ID 681342BDBM681342(US20240199561, Compound FC-115)
Affinity DataIC50: 524nMAssay Description:The ADP-GloTM Kinase Assay kit from Promega was used to screen the compounds before determination of their IC50 using the radiolabeled kinase assay. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Cold Spring Harbor Laboratory

US Patent
LigandChemical structure of BindingDB Monomer ID 681335BDBM681335(US20240199561, Compound FC-6)
Affinity DataIC50: 552nMAssay Description:The ADP-GloTM Kinase Assay kit from Promega was used to screen the compounds before determination of their IC50 using the radiolabeled kinase assay. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Cold Spring Harbor Laboratory

US Patent
LigandChemical structure of BindingDB Monomer ID 681337BDBM681337(US20240199561, Compound FC-7A)
Affinity DataIC50: 560nMAssay Description:The ADP-GloTM Kinase Assay kit from Promega was used to screen the compounds before determination of their IC50 using the radiolabeled kinase assay. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Cold Spring Harbor Laboratory

US Patent
LigandChemical structure of BindingDB Monomer ID 681347BDBM681347(US20240199561, Compound FC-208)
Affinity DataIC50: 560nMAssay Description:The ADP-GloTM Kinase Assay kit from Promega was used to screen the compounds before determination of their IC50 using the radiolabeled kinase assay. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Cold Spring Harbor Laboratory

US Patent
LigandChemical structure of BindingDB Monomer ID 681331BDBM681331(US20240199561, Compound FC-2)
Affinity DataIC50: 1.00E+4nMAssay Description:The ADP-GloTM Kinase Assay kit from Promega was used to screen the compounds before determination of their IC50 using the radiolabeled kinase assay. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Cold Spring Harbor Laboratory

US Patent
LigandChemical structure of BindingDB Monomer ID 681341BDBM681341(US20240199561, Compound FC-63)
Affinity DataIC50: 1.00E+4nMAssay Description:The ADP-GloTM Kinase Assay kit from Promega was used to screen the compounds before determination of their IC50 using the radiolabeled kinase assay. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Cold Spring Harbor Laboratory

US Patent
LigandChemical structure of BindingDB Monomer ID 681332BDBM681332(US20240199561, Compound FC-3)
Affinity DataIC50: 1.00E+4nMAssay Description:The ADP-GloTM Kinase Assay kit from Promega was used to screen the compounds before determination of their IC50 using the radiolabeled kinase assay. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Cold Spring Harbor Laboratory

US Patent
LigandChemical structure of BindingDB Monomer ID 681336BDBM681336(US20240199561, Compound FC-7)
Affinity DataIC50: 1.00E+4nMAssay Description:The ADP-GloTM Kinase Assay kit from Promega was used to screen the compounds before determination of their IC50 using the radiolabeled kinase assay. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent