Compile Data Set for Download or QSAR
Report error Found 124 Enz. Inhib. hit(s) with all data for entry = 6071
TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107176BDBM107176(US8592426, 25)
Affinity DataIC50: 0.100nMAssay Description:Calcium mobilization assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107181BDBM107181(US8592426, 30)
Affinity DataIC50: 0.100nMAssay Description:Calcium mobilization assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107189BDBM107189(US8592426, 38)
Affinity DataIC50: 0.200nMAssay Description:Calcium mobilization assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107206BDBM107206(US8592426, 56)
Affinity DataIC50: 0.200nMAssay Description:Calcium mobilization assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107212BDBM107212(US8592426, 63)
Affinity DataIC50: 0.200nMAssay Description:Calcium mobilization assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107193BDBM107193(US8592426, 42)
Affinity DataIC50: 0.200nMAssay Description:Calcium mobilization assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107177BDBM107177(US8592426, 26)
Affinity DataIC50: 0.200nMAssay Description:Calcium mobilization assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107190BDBM107190(US8592426, 116 | US8592426, 117 | US8592426, 39/40...)
Affinity DataIC50: 0.200nMAssay Description:Calcium mobilization assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107197BDBM107197(US8592426, 47)
Affinity DataIC50: 0.200nMAssay Description:Calcium mobilization assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107214BDBM107214(US8592426, 65)
Affinity DataIC50: 0.200nMAssay Description:Calcium mobilization assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107179BDBM107179(US8592426, 28)
Affinity DataIC50: 0.300nMAssay Description:Calcium mobilization assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107194BDBM107194(US8592426, 43)
Affinity DataIC50: 0.300nMAssay Description:Calcium mobilization assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107209BDBM107209(US8592426, 59)
Affinity DataIC50: 0.300nMAssay Description:Calcium mobilization assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107208BDBM107208(US8592426, 58)
Affinity DataIC50: 0.400nMAssay Description:Calcium mobilization assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107207BDBM107207(US8592426, 57)
Affinity DataIC50: 0.400nMAssay Description:Calcium mobilization assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107178BDBM107178(US8592426, 27)
Affinity DataIC50: 0.400nMAssay Description:Calcium mobilization assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107200BDBM107200(US8592426, 50)
Affinity DataIC50: 0.400nMAssay Description:Calcium mobilization assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107203BDBM107203(US8592426, 53)
Affinity DataIC50: 0.400nMAssay Description:Calcium mobilization assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107163BDBM107163(US8592426, 12)
Affinity DataIC50: 0.5nMAssay Description:Calcium mobilization assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107167BDBM107167(US8592426, 16)
Affinity DataIC50: 0.5nMAssay Description:Calcium mobilization assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107213BDBM107213(US8592426, 64)
Affinity DataIC50: 0.5nMAssay Description:Calcium mobilization assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107164BDBM107164(US8592426, 13)
Affinity DataIC50: 0.5nMAssay Description:Calcium mobilization assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107186BDBM107186(US8592426, 35)
Affinity DataIC50: 0.5nMAssay Description:Calcium mobilization assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107169BDBM107169(US8592426, 18)
Affinity DataIC50: 0.5nMAssay Description:Calcium mobilization assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107184BDBM107184(US8592426, 33)
Affinity DataIC50: 0.5nMAssay Description:Calcium mobilization assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107190BDBM107190(US8592426, 116 | US8592426, 117 | US8592426, 39/40...)
Affinity DataIC50: 0.600nMAssay Description:Calcium mobilization assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107156BDBM107156(US8592426, 5)
Affinity DataIC50: 0.600nMAssay Description:Calcium mobilization assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107185BDBM107185(US8592426, 34)
Affinity DataIC50: 0.600nMAssay Description:Calcium mobilization assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107168BDBM107168(US8592426, 17)
Affinity DataIC50: 0.600nMAssay Description:Calcium mobilization assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107173BDBM107173(US8592426, 22)
Affinity DataIC50: 0.800nMAssay Description:Calcium mobilization assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107155BDBM107155(US8592426, 4)
Affinity DataIC50: 2nMAssay Description:Calcium mobilization assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107172BDBM107172(US8592426, 21)
Affinity DataIC50: 2.30nMAssay Description:Calcium mobilization assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107177BDBM107177(US8592426, 26)
Affinity DataKi:  2.60nMAssay Description:Binding assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107201BDBM107201(US8592426, 51)
Affinity DataIC50: 2.70nMAssay Description:Calcium mobilization assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107189BDBM107189(US8592426, 38)
Affinity DataKi:  3nMAssay Description:Binding assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107176BDBM107176(US8592426, 25)
Affinity DataKi:  3.10nMAssay Description:Binding assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107180BDBM107180(US8592426, 29)
Affinity DataIC50: 3.40nMAssay Description:Calcium mobilization assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107209BDBM107209(US8592426, 59)
Affinity DataKi:  3.5nMAssay Description:Binding assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107203BDBM107203(US8592426, 53)
Affinity DataKi:  3.60nMAssay Description:Binding assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107178BDBM107178(US8592426, 27)
Affinity DataKi:  3.60nMAssay Description:Binding assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107171BDBM107171(US8592426, 20)
Affinity DataIC50: 3.60nMAssay Description:Calcium mobilization assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107187BDBM107187(US8592426, 36)
Affinity DataIC50: 3.60nMAssay Description:Calcium mobilization assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107181BDBM107181(US8592426, 30)
Affinity DataKi:  3.90nMAssay Description:Binding assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107193BDBM107193(US8592426, 42)
Affinity DataKi:  4nMAssay Description:Binding assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107190BDBM107190(US8592426, 116 | US8592426, 117 | US8592426, 39/40...)
Affinity DataKi:  4nMAssay Description:Binding assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107162BDBM107162(US8592426, 11)
Affinity DataIC50: 4nMAssay Description:Calcium mobilization assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107198BDBM107198(US8592426, 48)
Affinity DataIC50: 4nMAssay Description:Calcium mobilization assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107179BDBM107179(US8592426, 28)
Affinity DataKi:  4.10nMAssay Description:Binding assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107202BDBM107202(US8592426, 52)
Affinity DataIC50: 4.30nMAssay Description:Calcium mobilization assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

TargetKininogen-1(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 107214BDBM107214(US8592426, 65)
Affinity DataKi:  4.40nMAssay Description:Binding assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2014
Entry Details
US Patent

Displayed 1 to 50 (of 124 total ) | Next | Last >>
Jump to: