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Found 5 Enz. Inhib. hit(s) with all data for entry = 8219
TargetFructose-bisphosphate aldolase(Mycobacterium tuberculosis (strain H37Rv))
The University Of Denver And Regis University

US Patent
LigandPNGBDBM382(1571-30-8 | 55088_ALDRICH | 8-hydroxy-2-quinolinec...)
Affinity DataIC50:  1.40E+4nMAssay Description:Enzymatic activity is measured by contacting the enzyme with a suitable substrate, such as fructose 1,6-bisphosphate, and measuring formation of a pr...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFructose-bisphosphate aldolase(Mycobacterium tuberculosis (strain H37Rv))
The University Of Denver And Regis University

US Patent
LigandPNGBDBM382(1571-30-8 | 55088_ALDRICH | 8-hydroxy-2-quinolinec...)
Affinity DataIC50:  1.70E+4nM Kd:  6.94E+3nMAssay Description:Enzymatic activity is measured by contacting the enzyme with a suitable substrate, such as fructose 1,6-bisphosphate, and measuring formation of a pr...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFructose-bisphosphate aldolase(Mycobacterium tuberculosis (strain H37Rv))
The University Of Denver And Regis University

US Patent
LigandPNGBDBM32144(8-quinolinamine | 8-quinolylamine | AS-232 | US100...)
Affinity DataIC50:  7.90E+4nMAssay Description:Enzymatic activity is measured by contacting the enzyme with a suitable substrate, such as fructose 1,6-bisphosphate, and measuring formation of a pr...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFructose-bisphosphate aldolase(Mycobacterium tuberculosis (strain H37Rv))
The University Of Denver And Regis University

US Patent
LigandPNGBDBM32203(8-quinolinol | CHEMBL310555 | US10005735, Table 1....)
Affinity DataIC50:  3.00E+5nMAssay Description:Enzymatic activity is measured by contacting the enzyme with a suitable substrate, such as fructose 1,6-bisphosphate, and measuring formation of a pr...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFructose-bisphosphate aldolase(Mycobacterium tuberculosis (strain H37Rv))
The University Of Denver And Regis University

US Patent
LigandPNGBDBM237137(US9394254, 34)
Affinity DataIC50:  5.70E+5nMAssay Description:Enzymatic activity is measured by contacting the enzyme with a suitable substrate, such as fructose 1,6-bisphosphate, and measuring formation of a pr...More data for this Ligand-Target Pair
In DepthDetails US Patent