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Compounds Sorted by Binding Targets per Compound

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304   310   315   323   339   369   370   371   372   373   374   375   376   377   378   380   381   383   384   
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429   443   447   515   
Compounds Sorted Alphabetically
Compound Name (alphabetical)
Binding Targets
Enz. Inhib. Data
ITC Data
Alternate Compound Names
  • ADORA1
  • Adenosine A1 receptor
  • Adenosine A2 receptor
  • Adenosine A2a receptor
  • Adenosine Receptors A2a (A2a)
  • Adenosine receptor
  • Adenosine receptor A1
  • Adenosine receptor A1 (A1)
  • Adenosine receptor A2a
  • Adenosine receptor A2a and A3
  • Adenosine receptor A2b
  • Adenosine receptor A3
  • Alkaline phosphatase, tissue-nonspecific isozyme
  • Bile salt export pump
  • Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B
  • Canalicular multispecific organic anion transporter 1
  • Canalicular multispecific organic anion transporter 2
  • Chitinase 1
  • Endochitinase B1
  • Heart phosphodiesterase
  • Homo sapiens phosphodiesterase 2A (PDE2A)
  • Intestinal alkaline phosphatase
  • Multidrug resistance-associated protein 4
  • Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
  • Phosphodiesterase 1
  • Phosphodiesterase 3
  • Phosphodiesterase 4
  • Phospholipase A-2-activating protein
  • cAMP-specific 3',5'-cyclic phosphodiesterase 4A
  • cAMP-specific 3',5'-cyclic phosphodiesterase 4C
173 Ki 24 IC50 1 Kd 1 EC50
  • 1,3-dimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-dione
  • 1,3-dimethyl-7H-purine-2,6-dione
  • Afonilum
  • Aminophyllin
  • Aminophylline
  • CHEMBL190
  • Cardophyllin
  • Euphylline
  • Theophylline
  • Theophylline (1,3-dimethylxanthine)
  • β-Carbonic anhydrase 2 (CA 2)
  • Alpha carbonic anhydrase
  • Astrosclerin-3
  • Beta-carbonic anhydrase
  • Carbonate dehydratase
  • Carbonic Anhydrase (hpCA)
  • Carbonic Anhydrase (mtCA 1)
  • Carbonic Anhydrase (mtCA 3)
  • Carbonic Anhydrase 2 (Can2)
  • Carbonic Anhydrase III
  • Carbonic Anhydrase IV
  • Carbonic Anhydrase VA
  • Carbonic Anhydrase VB
  • Carbonic Anhydrase XIII
  • Carbonic Anhydrase XIV
  • Carbonic Anhydrase XV
  • Carbonic anhydrase
  • Carbonic anhydrase 1
  • Carbonic anhydrase 12
  • Carbonic anhydrase 2
  • Carbonic anhydrase 4
  • Carbonic anhydrase 6 (CA-VI)
  • Carbonic anhydrase 7
  • Carbonic anhydrase 9
  • Carbonic anhydrase, alpha family
  • Carbonic anhydrases; II & IX
  • Delta carbonic anhydrase
  • Gamma-carbonic anhydrase
  • PROBABLE TRANSMEMBRANE CARBONIC ANHYDRASE (CARBONATE DEHYDRATASE) (CARBONIC DEHYDRATASE)
  • beta-Carbonic Anhydrase
174 Ki 2 IC50
  • 4-(2-aminoethyl)benzene-1-sulfonamide
  • CHEMBL7087
  • aromatic sulfonamide compound 7
  • aromatic/heteroaromatic sulfonamide 6
  • β-Carbonic anhydrase 2 (CA 2)
  • Alpha carbonic anhydrase
  • Astrosclerin-3
  • Beta-carbonic anhydrase
  • Carbonate dehydratase
  • Carbonic Anhydrase (hpCA)
  • Carbonic Anhydrase (mtCA 1)
  • Carbonic Anhydrase (mtCA 3)
  • Carbonic Anhydrase 2 (Can2)
  • Carbonic Anhydrase III
  • Carbonic Anhydrase IV
  • Carbonic Anhydrase VA
  • Carbonic Anhydrase VB
  • Carbonic Anhydrase XIV
  • Carbonic Anhydrase XV
  • Carbonic anhydrase
  • Carbonic anhydrase 1
  • Carbonic anhydrase 12
  • Carbonic anhydrase 13 (CA XIII)
  • Carbonic anhydrase 15
  • Carbonic anhydrase 2
  • Carbonic anhydrase 4
  • Carbonic anhydrase 6 (CA-VI)
  • Carbonic anhydrase 7
  • Carbonic anhydrase 9
  • Carbonic anhydrase, alpha family
  • Chitinase (chiA1)
  • Delta carbonic anhydrase
  • Serum paraoxonase/arylesterase 1
  • beta-Carbonic Anhydrase
154 Ki 16 IC50
  • 1,3,4-Thiadiazole-2-sulfonamide, 6
  • 1,3,4-thiadiazole-2-sulfonamide 15
  • 5-Amino-1,3,4-thiadiazole-2-sulphonamide (1)
  • 5-amino-1,3,4-thiadiazole-2-sulfonamide
  • CHEMBL265674
  • aromatic/heteroaromatic sulfonamide 13
  • β-Carbonic anhydrase 2 (CA 2)
  • Alpha carbonic anhydrase
  • Astrosclerin-3
  • Beta-carbonic anhydrase
  • Carbonic Anhydrase (hpCA)
  • Carbonic Anhydrase (mtCA 1)
  • Carbonic Anhydrase (mtCA 3)
  • Carbonic Anhydrase 2 (Can2)
  • Carbonic Anhydrase III
  • Carbonic Anhydrase IV
  • Carbonic Anhydrase V
  • Carbonic Anhydrase VA
  • Carbonic Anhydrase VB
  • Carbonic Anhydrase XIII
  • Carbonic Anhydrase XIV
  • Carbonic Anhydrase XV
  • Carbonic anhydrase
  • Carbonic anhydrase 1
  • Carbonic anhydrase 12
  • Carbonic anhydrase 13 (CA XIII)
  • Carbonic anhydrase 2
  • Carbonic anhydrase 4
  • Carbonic anhydrase 6 (CA-VI)
  • Carbonic anhydrase 7
  • Carbonic anhydrase 9
  • Delta carbonic anhydrase
  • Gamma-carbonic anhydrase
  • PROBABLE TRANSMEMBRANE CARBONIC ANHYDRASE (CARBONATE DEHYDRATASE) (CARBONIC DEHYDRATASE)
  • beta-Carbonic Anhydrase
  • corticotropin releasing factor-binding protein
290 Ki 11 IC50 2 EC50
  • CHEMBL288100
  • METHAZOLAMIDE
  • MZA3
  • Methazolamide
  • Methazolamide (MZA)
  • Methazolamide, MZA
  • N-[(2Z)-3-methyl-5-sulfamoyl-2,3-dihydro-1,3,4-thiadiazol-2-ylidene]acetamide
  • Sulfonamide, 2
  • cid_4100
  • sulfonamide 2
  • β-Carbonic anhydrase 2 (CA 2)
  • Alpha carbonic anhydrase
  • Astrosclerin-3
  • Beta-carbonic anhydrase
  • Carbonate dehydratase
  • Carbonic Anhydrase (hpCA)
  • Carbonic Anhydrase (mtCA 1)
  • Carbonic Anhydrase (mtCA 3)
  • Carbonic Anhydrase 2 (Can2)
  • Carbonic Anhydrase III
  • Carbonic Anhydrase IV
  • Carbonic Anhydrase VA
  • Carbonic Anhydrase VB
  • Carbonic Anhydrase XIII
  • Carbonic Anhydrase XIV
  • Carbonic Anhydrase XV
  • Carbonic anhydrase
  • Carbonic anhydrase 1
  • Carbonic anhydrase 12
  • Carbonic anhydrase 2
  • Carbonic anhydrase 4
  • Carbonic anhydrase 6 (CA-VI)
  • Carbonic anhydrase 7
  • Carbonic anhydrase 9
  • Carbonic anhydrase, alpha family
  • Carbonic anhydrases; II & IX
  • Delta carbonic anhydrase
  • Gamma-carbonic anhydrase
  • PROBABLE TRANSMEMBRANE CARBONIC ANHYDRASE (CARBONATE DEHYDRATASE) (CARBONIC DEHYDRATASE)
  • beta-Carbonic Anhydrase
295 Ki 8 IC50 1 Kd
  • (2S,4S)-4-(ethylamino)-2-methyl-1,1-dioxo-2H,3H,4H-1,7-thieno[2,3-b]thiopyran-6-sulfonamide
  • Dorzolamide (DRZ)
  • Dorzolamide (DZA)
  • β-Carbonic anhydrase 2 (CA 2)
  • Alpha carbonic anhydrase
  • Amine oxidase [flavin-containing]
  • Amine oxidase [flavin-containing] B
  • Astrosclerin-3
  • Beta-carbonic anhydrase
  • Carbonic Anhydrase (hpCA)
  • Carbonic Anhydrase (mtCA 1)
  • Carbonic Anhydrase (mtCA 3)
  • Carbonic Anhydrase 2 (Can2)
  • Carbonic Anhydrase III
  • Carbonic Anhydrase VA
  • Carbonic Anhydrase VB
  • Carbonic Anhydrase XIV
  • Carbonic Anhydrase XV
  • Carbonic anhydrase
  • Carbonic anhydrase 1
  • Carbonic anhydrase 12
  • Carbonic anhydrase 13 (CA XIII)
  • Carbonic anhydrase 15
  • Carbonic anhydrase 2
  • Carbonic anhydrase 3 (CA III)
  • Carbonic anhydrase 4
  • Carbonic anhydrase 6 (CA-VI)
  • Carbonic anhydrase 7
  • Carbonic anhydrase 9
  • Delta carbonic anhydrase
  • Monoamine Oxidase Type B (MAO-B)
  • PROBABLE TRANSMEMBRANE CARBONIC ANHYDRASE (CARBONATE DEHYDRATASE) (CARBONIC DEHYDRATASE)
  • beta-Carbonic Anhydrase
143 Ki 2 IC50 3 Kd 1 Koff 1 Kon
  • 1,2-benzoxazol-3-ylmethanesulfonamide
  • CHEMBL750
  • SPR_2
  • US10172837, Zonisamide
  • Zonisamide
  • Zonisamide (ZNA)
  • Zonisamide (ZNS)
  • Zonisamide, 1
  • Zonisamide, ZNS
  • 6-phosphogluconate dehydrogenase (6PGD)
  • AICAR transformylase
  • Alpha trans-inducing protein (VP16)
  • Bile salt export pump
  • Bile salt export pump (BSEP)
  • Canalicular multispecific organic anion transporter 1
  • Canalicular multispecific organic anion transporter 2
  • Dihydrofolate Reductase (DHFR)
  • Dihydrofolate reductase
  • Dihydrofolate reductase (DHFR)
  • Folate receptor alpha
  • Folate receptor beta
  • Folate transporter 1
  • Folylpoly-gamma-glutamate synthetase
  • GAR transformylase
  • Glucose 6-phosphate dehydrogenase (G6PD)
  • Glycinamide ribonucleotide formyltransferase (GARFTase)
  • Multidrug resistance associated protein
  • Nuclear receptor coactivator 1
  • Organic anion-transporting polypeptide 1D1 (Oatp1d1)
  • Proton-coupled folate transporter
  • Pteridine reductase 1
  • Solute carrier family 22 member 20
  • Solute carrier family 22 member 6
  • Thymidylate Synthase (TS)
  • Thymidylate synthase
  • Thymidylate synthase (EC 2.1.1.45) (TS) (TSase)
  • Thymidylate synthase (TS)
  • nuclear receptor coactivator 3 isoform a
  • protein-arginine deiminase type-4
48 Ki 210 IC50 10 Kd 3 EC50 3 Koff 3 Kon
  • 2-[(4-{[(2,4-diaminopteridin-6-yl)methyl](methyl)amino}phenyl)formamido]pentanedioic acid
  • CHEMBL34259
  • METHOTREXATE
  • MTX
  • Methotrexate
  • cid_126941
  • ALK tyrosine kinase receptor
  • Axin-1/Glycogen synthase kinase-3 beta
  • CaM kinase IV
  • Homeodomain-interacting protein kinase 1
  • Homeodomain-interacting protein kinase 2 (HIPK2)
  • Homeodomain-interacting protein kinase 3
  • MAP kinase-activated protein kinase 3
  • MAP kinase-activated protein kinase 5
  • Mitogen-activated protein kinase 1
  • Mitogen-activated protein kinase 10
  • Mitogen-activated protein kinase 3
  • Mitogen-activated protein kinase 8
  • Myotonin-protein kinase
  • PAK 1/CDC42
  • Proto-oncogene tyrosine-protein kinase Src
  • RAC-alpha serine/threonine-protein kinase
  • Serine/threonine-protein kinase 24
  • Serine/threonine-protein kinase AKT
  • Serine/threonine-protein kinase AKT2
  • Serine/threonine-protein kinase MARK1
  • Serine/threonine-protein kinase MST4
  • Serine/threonine-protein kinase Nek1
  • Serine/threonine-protein kinase Nek2
  • Serine/threonine-protein kinase VRK1
  • Serine/threonine-protein kinase c-TAK1
  • Serine/threonine-protein kinase pim-2
  • Tyrosine-protein kinase BRK
  • Tyrosine-protein kinase JAK3
  • p21-Activated kinase 2 (PAK2)
  • p21-Activated kinase 3 (PAK3)
30 IC50
  • CHEMBL3133821
  • 5-HT3A Serotonin Receptor
  • 5-hydroxytryptamine receptor 1A
  • 5-hydroxytryptamine receptor 2A
  • ADRA2C
  • Adrenergic receptor alpha-2
  • Alpha-1 Adrenergic Receptor/ adrenergic receptor/ adrenergic receptor
  • Alpha-1A adrenergic receptor
  • Alpha-1D adrenergic receptor
  • Alpha-2A adrenergic receptor
  • Alpha-2B adrenergic receptor
  • Alpha-2C adrenergic receptor
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Bile salt export pump
  • Bile salt export pump (BSEP)
  • Canalicular multispecific organic anion transporter 1
  • Canalicular multispecific organic anion transporter 2
  • Cerebral cortex alpha adrenergic receptor
  • D(1A) dopamine receptor
  • D(2) dopamine receptor
  • Imidazoline I1
  • Imidazoline I2-receptor
  • Imidazoline receptor 1 (I1R)
  • Multidrug resistance-associated protein 4
  • Nischarin
  • Serotonin (5-HT) receptor
  • Serotonin receptor 2a and 2c (5HT2A and 5HT2C)
  • Sodium-dependent noradrenaline transporter
  • adrenergic Alpha1
  • adrenergic Alpha2
70 Ki 13 IC50
  • 2-(2,3-dihydro-1,4-benzodioxin-2-yl)-4,5-dihydro-1H-imidazole
  • 4,5-dihydro-2-(2,3-dihydro-1,4-benzodioxin-2-yl)-1H-imidazole
  • CHEMBL10316
  • Idazoxan
  • US8633208, Idazoxan
  • ALK tyrosine kinase receptor
  • BDNF/NT-3 growth factors receptor
  • Cytoplasmic tyrosine-protein kinase BMX
  • Fibroblast growth factor receptor 3
  • Fibroblast growth factor receptor 4
  • Hepatocyte growth factor receptor
  • High affinity nerve growth factor receptor
  • Insulin receptor
  • Insulin-like growth factor I receptor
  • Macrophage colony-stimulating factor 1 receptor (CSF1R)
  • Macrophage-stimulating protein receptor
  • Mast/stem cell growth factor receptor Kit
  • NT-3 growth factor receptor
  • Platelet-derived growth factor receptor beta
  • Proto-oncogene tyrosine-protein kinase ROS
  • Proto-oncogene tyrosine-protein kinase Src
  • Proto-oncogene tyrosine-protein kinase receptor Ret
  • Serine/threonine-protein kinase B-raf
  • Tyrosine-protein kinase ABL1
  • Tyrosine-protein kinase Fgr
  • Tyrosine-protein kinase JAK2
  • Tyrosine-protein kinase Lck
  • Tyrosine-protein kinase Lyn
  • Tyrosine-protein kinase Mer
  • Tyrosine-protein kinase SYK
  • Tyrosine-protein kinase ZAP-70
  • Tyrosine-protein kinase receptor FLT3
  • Tyrosine-protein kinase receptor Tie-1
  • Vascular endothelial growth factor receptor 1
  • Vascular endothelial growth factor receptor 2
32 IC50
  • CHEMBL3582427
  • 5-hydroxytryptamine receptor 1A
  • 5-hydroxytryptamine receptor 3A
  • 5-hydroxytryptamine receptor 5A
  • 5-hydroxytryptamine receptor 6
  • 5-hydroxytryptamine receptor 7
  • Adrenergic receptor
  • Alpha-1A adrenergic receptor
  • Alpha-2A adrenergic receptor
  • Beta-2 adrenergic receptor
  • Beta-2 adrenergic receptor and beta-3 adrenergic receptor
  • Bile salt export pump
  • Canalicular multispecific organic anion transporter 1
  • Canalicular multispecific organic anion transporter 2
  • Cystic fibrosis transmembrane conductance regulator
  • D(1A) dopamine receptor
  • D(1B) dopamine receptor
  • D(2) dopamine receptor
  • D(3) dopamine receptor
  • D(4) dopamine receptor
  • DRD1
  • Delta-type opioid receptor
  • Dopamine receptor
  • Histamine H2 receptor
  • Histamine receptor (H3 and H4)
  • Multidrug resistance-associated protein 4
  • Muscarinic acetylcholine receptor M1
  • Muscarinic acetylcholine receptor M1 and M3
  • Muscarinic acetylcholine receptor M2 and M5
  • Serotonin (5-HT) receptor
  • Sigma non-opioid intracellular receptor 1
62 Ki 9 IC50 1 Kd 17 EC50
  • (-)-Pramipexole
  • (6S)-N(6)-propyl-4,5,6,7-tetrahydro-1,3-benzothiazole-2,6-diamine
  • 2,6-Benzothiazolediamine, 4,5,6,7-tetrahydro-N(sup 6)-propyl-, (S)-
  • CHEMBL301265
  • PRAMIPEXOLE
  • cid_119570
  • 5-hydroxytryptamine receptor 1A
  • 5-hydroxytryptamine receptor 1B
  • 5-hydroxytryptamine receptor 2A
  • 5-hydroxytryptamine receptor 2B
  • 5-hydroxytryptamine receptor 2C
  • 5-hydroxytryptamine receptor 6
  • 5-hydroxytryptamine receptor 7
  • Alpha-2A adrenergic receptor
  • Alpha-2B adrenergic receptor
  • Alpha-2C adrenergic receptor
  • Beta-1 adrenergic receptor
  • Beta-2 adrenergic receptor
  • C-C chemokine receptor type 1
  • C-C chemokine receptor type 2
  • C-C chemokine receptor type 3
  • C-C chemokine receptor type 5
  • C-C chemokine receptor type 6 (CCR6)
  • D(1A) dopamine receptor
  • D(2) dopamine receptor
  • D(3) dopamine receptor
  • D(4) dopamine receptor
  • Delta-type opioid receptor
  • Kappa-type opioid receptor
  • Mu-type opioid receptor
  • Muscarinic acetylcholine receptor M1
  • Muscarinic acetylcholine receptor M2
  • Muscarinic acetylcholine receptor M3
  • Muscarinic acetylcholine receptor M4
  • Muscarinic acetylcholine receptor M5
  • Serotonin 3a (5-HT3a)/3b (5-HT3b)/3c (5-HT3c)/3d (5-HT3d)/3e (5-HT3e) receptor
34 IC50
  • (R)-N-(2-(3-(4-(4-fluorobenzyl)-2-methylpiperazin-1-yl)-3-oxoprop-1-enyl)-5-chlorophenyl)acetamide
  • CHEMBL198949
  • ALK tyrosine kinase receptor
  • Cyclin-dependent kinase 1
  • Cyclin-dependent kinase 4
  • Cyclin-dependent kinase 6
  • Discoidin domain-containing receptor 2
  • Ephrin type-A receptor 2
  • Epidermal growth factor receptor
  • Fibroblast growth factor receptor 1
  • Fibroblast growth factor receptor 2
  • Fibroblast growth factor receptor 3
  • Fibroblast growth factor receptor 4
  • Hepatocyte growth factor receptor
  • Insulin receptor
  • Insulin-like growth factor I receptor
  • Leukocyte tyrosine kinase receptor
  • Mast/stem cell growth factor receptor Kit
  • Mitogen-activated protein kinase 1
  • Platelet-derived growth factor receptor alpha
  • Platelet-derived growth factor receptor beta
  • Proto-oncogene tyrosine-protein kinase ROS
  • Proto-oncogene tyrosine-protein kinase Src
  • Proto-oncogene tyrosine-protein kinase receptor Ret
  • Receptor protein-tyrosine kinase erbB-4
  • Receptor tyrosine-protein kinase erbB-2
  • Tyrosine-protein kinase ABL1
  • Tyrosine-protein kinase Mer
  • Tyrosine-protein kinase receptor TYRO3
  • Tyrosine-protein kinase receptor UFO
  • Vascular endothelial growth factor receptor 1
  • Vascular endothelial growth factor receptor 2
37 IC50
  • CHEMBL4062877
  • ALK tyrosine kinase receptor
  • Aurora kinase A/Targeting protein for Xklp2
  • Axin-1/Glycogen synthase kinase-3 beta
  • Cyclin-dependent kinase 2
  • Ephrin receptor
  • Ephrin type-B receptor 4
  • Fibroblast growth factor receptor 3
  • Hepatocyte growth factor receptor
  • Insulin receptor
  • Insulin-like growth factor I receptor
  • MAP kinase-interacting serine/threonine-protein kinase 2
  • Mast/stem cell growth factor receptor Kit
  • Mitogen-activated protein kinase 1
  • Mitogen-activated protein kinase 14
  • Non-receptor tyrosine-protein kinase TYK2
  • Protein kinase N1
  • Protein kinase N2
  • Proto-oncogene tyrosine-protein kinase receptor Ret
  • Receptor tyrosine-protein kinase erbB-2
  • Rho-associated protein kinase 2
  • Tyrosine-protein kinase BTK
  • Tyrosine-protein kinase JAK1
  • Tyrosine-protein kinase JAK2
  • Tyrosine-protein kinase JAK3
  • Tyrosine-protein kinase Lck
  • Tyrosine-protein kinase ZAP-70
  • Tyrosine-protein kinase receptor UFO
  • Vascular endothelial growth factor receptor 2
  • [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial
  • cAMP-dependent protein kinase (PKA)
38 IC50
  • (3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,10,11,12-hexahydro-1H-benzo[c][1]oxacyclotetradecine-1,7(8H)-dione
  • CHEMBL1651521
  • CHEMBL1651522
  • Aurora kinase A/Targeting protein for Xklp2
  • Axin-1/Glycogen synthase kinase-3 beta
  • Casein kinase I isoform delta
  • Cyclin-dependent kinase 2
  • Epidermal growth factor receptor
  • Fibroblast growth factor receptor 1
  • Hepatocyte growth factor receptor
  • High affinity nerve growth factor receptor
  • Inhibitor of nuclear factor kappa-B kinase subunit beta
  • Inhibitor of nuclear factor kappa-B kinase subunit epsilon
  • Insulin receptor
  • MAP kinase-activated protein kinase 2
  • Mitogen-activated protein kinase 1
  • Protein kinase C (PKC)
  • Proto-oncogene tyrosine-protein kinase Src
  • RAC-alpha serine/threonine-protein kinase
  • Serine/threonine-protein kinase CHK2
  • Serine/threonine-protein kinase Chk1/2
  • Serine/threonine-protein kinase PAK 4
  • Serine/threonine-protein kinase Sgk1
  • Serine/threonine-protein kinase TAO3
  • Serine/threonine-protein kinase pim-2
  • Syk protein
  • Tyrosine-protein kinase ABL1
  • Tyrosine-protein kinase BTK
  • Tyrosine-protein kinase Lck
  • Tyrosine-protein kinase Mer
  • Tyrosine-protein kinase receptor UFO
  • Vascular endothelial growth factor receptor 2
  • [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial
30 IC50
  • CHEMBL1933552
  • 1-phosphatidylinositol 3-phosphate 5-kinase
  • Aurora kinase A/B
  • Aurora kinase A/Targeting protein for Xklp2
  • BMP-2-inducible protein kinase
  • Casein kinase I isoform epsilon
  • Citron Rho-interacting kinase
  • Dual-specificity tyrosine-phosphorylation regulated kinase 1A
  • Interleukin-1 receptor-associated kinase 3
  • Mitogen-activated protein kinase 15
  • Mitogen-activated protein kinase kinase kinase 11
  • Mitogen-activated protein kinase kinase kinase 7
  • Mitogen-activated protein kinase kinase kinase 9
  • Mitogen-activated protein kinase kinase kinase kinase 2
  • Myosin light chain kinase family member 4
  • Non-receptor tyrosine-protein kinase TYK2
  • Phosphatidylinositol 4-kinase, PI4K
  • Serine/threonine-protein kinase 17A
  • Serine/threonine-protein kinase 17B (STK17B)
  • Serine/threonine-protein kinase 35
  • Serine/threonine-protein kinase 36
  • Serine/threonine-protein kinase DCLK3
  • Serine/threonine-protein kinase GAK
  • Serine/threonine-protein kinase RIO1
  • Serine/threonine-protein kinase RIPK2
  • Serine/threonine-protein kinase SIK3
  • Serine/threonine-protein kinase pim-1
  • Serine/threonine-protein kinase pim-2
  • Serine/threonine-protein kinase pim-3
  • Tyrosine-protein kinase JAK1
  • Tyrosine-protein kinase receptor FLT3
17 IC50 19 Kd
  • CHEMBL4564337
  • 5-HT5
  • 5-HT5B
  • 5-hydroxytryptamine receptor 1A
  • 5-hydroxytryptamine receptor 1B
  • 5-hydroxytryptamine receptor 1D
  • 5-hydroxytryptamine receptor 2A
  • 5-hydroxytryptamine receptor 2B
  • 5-hydroxytryptamine receptor 2C
  • 5-hydroxytryptamine receptor 5A
  • 5-hydroxytryptamine receptor 6
  • 5-hydroxytryptamine receptor 7
  • 5-hydroxytryptamine receptor 7 (5HT7)
  • ADRA1A
  • ADRA1B
  • D(2) dopamine receptor
  • DRD1
  • G protein-coupled receptor
  • HTR1A
  • HTR1D
  • HTR1E
  • HTR1F
  • HTR2C
  • HTR5A
  • HTR6
  • HTR7
  • Human herpesvirus 5 chemokine receptor
  • Serotonin (5-HT) receptor
  • Serotonin 1B/1D receptor
  • Serotonin receptor 2a and 2c (5HT2A and 5HT2C)
  • ubiquitin-conjugating enzyme E2 N
119 Ki 12 IC50 5 EC50
  • METHIOTHEPIN
  • MLS000859918
  • Methiothepin mesylate salt
  • SMR000326779
  • cid_3039995
  • mesylic acid;1-methyl-4-[3-(methylthio)-5,6-dihydrobenzo[b][1]benzothiepin-5-yl]piperazine
  • methanesulfonic acid;1-methyl-4-(3-methylsulfanyl-5,6-dihydrobenzo[b][1]benzothiepin-5-yl)piperazine
  • methanesulfonic acid;1-methyl-4-[3-(methylthio)-5,6-dihydrobenzo[b][1]benzothiepin-5-yl]piperazine