Affinity DataKi: 0.302nMAssay Description:Inhibition of [3H]NC-NH2 binding to mouse forebrain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.398nMAssay Description:Inhibition of [3H]NC-NH2 binding to mouse forebrain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.603nMAssay Description:Inhibition of [3H]NC-NH2 binding to mouse forebrain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.794nMAssay Description:Inhibition of [3H]NC-NH2 binding to mouse forebrain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.794nMAssay Description:Affinity to nociceptin receptors on mouse forebrain membranes by [3H]NC-NH2 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.794nMAssay Description:Affinity to nociceptin receptors on mouse forebrain membranes by [3H]NC-NH2 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.891nMAssay Description:Inhibition of [3H]NC-NH2 binding to mouse forebrain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.912nMAssay Description:Inhibition of [3H]NC-NH2 binding to mouse forebrain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Affinity to nociceptin receptors on mouse forebrain membranes by [3H]NC-NH2 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of [3H]NC-NH2 binding to mouse forebrain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Inhibition of [3H]NC-NH2 binding to mouse forebrain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Inhibition of [3H]NC-NH2 binding to mouse forebrain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Affinity to nociceptin receptors on mouse forebrain membranes by [3H]NC-NH2 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Inhibition of [3H]NC-NH2 binding to mouse forebrain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Affinity to nociceptin receptors on mouse forebrain membranes by [3H]NC-NH2 displacement.More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
Leicester Royal Infirmary
Curated by PDSP Ki Database
Leicester Royal Infirmary
Curated by PDSP Ki Database
Affinity DataKi: 10nMAssay Description:Affinity to nociceptin receptors on mouse forebrain membranes by [3H]NC-NH2 displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
Leicester Royal Infirmary
Curated by PDSP Ki Database
Leicester Royal Infirmary
Curated by PDSP Ki Database
TargetMu-type opioid receptor(Homo sapiens (Human))
Leicester Royal Infirmary
Curated by PDSP Ki Database
Leicester Royal Infirmary
Curated by PDSP Ki Database
Affinity DataKi: 16nMAssay Description:Affinity to nociceptin receptors on mouse forebrain membranes by [3H]NC-NH2 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Inhibition of [3H]NC-NH2 binding to mouse forebrain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Affinity to nociceptin receptors on mouse forebrain membranes by [3H]NC-NH2 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Affinity to nociceptin receptors on mouse forebrain membranes by [3H]NC-NH2 displacement.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Leicester Royal Infirmary
Curated by PDSP Ki Database
Leicester Royal Infirmary
Curated by PDSP Ki Database
Affinity DataKi: 89nMAssay Description:Inhibition of [3H]NC-NH2 binding to mouse forebrain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Affinity to nociceptin receptors on mouse forebrain membranes by [3H]NC-NH2 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Affinity to nociceptin receptors on mouse forebrain membranes by [3H]NC-NH2 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 126nMAssay Description:Affinity to nociceptin receptors on mouse forebrain membranes by [3H]NC-NH2 displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
Leicester Royal Infirmary
Curated by PDSP Ki Database
Leicester Royal Infirmary
Curated by PDSP Ki Database
Affinity DataKi: 200nMAssay Description:Affinity to nociceptin receptors on mouse forebrain membranes by [3H]NC-NH2 displacement.More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
Leicester Royal Infirmary
Curated by PDSP Ki Database
Leicester Royal Infirmary
Curated by PDSP Ki Database
TargetKappa-type opioid receptor(Homo sapiens (Human))
Leicester Royal Infirmary
Curated by PDSP Ki Database
Leicester Royal Infirmary
Curated by PDSP Ki Database
TargetDelta-type opioid receptor(Homo sapiens (Human))
Leicester Royal Infirmary
Curated by PDSP Ki Database
Leicester Royal Infirmary
Curated by PDSP Ki Database
Affinity DataKi: 316nMAssay Description:Affinity to nociceptin receptors on mouse forebrain membranes by [3H]NC-NH2 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 398nMAssay Description:Affinity to nociceptin receptors on mouse forebrain membranes by [3H]NC-NH2 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 501nMAssay Description:Inhibition of [3H]NC-NH2 binding to mouse forebrain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 631nMAssay Description:Affinity to nociceptin receptors on mouse forebrain membranes by [3H]NC-NH2 displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
Leicester Royal Infirmary
Curated by PDSP Ki Database
Leicester Royal Infirmary
Curated by PDSP Ki Database
Affinity DataKi: 1.78E+3nMAssay Description:Inhibition of [3H]NC-NH2 binding to mouse forebrain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.51E+3nMAssay Description:Affinity to nociceptin receptors on mouse forebrain membranes by [3H]NC-NH2 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 2.51E+3nMAssay Description:Affinity to nociceptin receptors on mouse forebrain membranes by [3H]NC-NH2 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 2.51E+3nMAssay Description:Affinity to nociceptin receptors on mouse forebrain membranes by [3H]NC-NH2 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 3.16E+3nMAssay Description:Affinity to nociceptin receptors on mouse forebrain membranes by [3H]NC-NH2 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 3.16E+3nMAssay Description:Affinity to nociceptin receptors on mouse forebrain membranes by [3H]NC-NH2 displacement.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Leicester Royal Infirmary
Curated by PDSP Ki Database
Leicester Royal Infirmary
Curated by PDSP Ki Database
Affinity DataKi: <1.00E+4nMAssay Description:Binding affinity towards Orphanin FQ receptor on mouse forebrain membranes was determined using [3H]-NC-NH2 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+4nMAssay Description:Affinity to nociceptin receptors on mouse forebrain membranes by [3H]NC-NH2 displacement.More data for this Ligand-Target Pair