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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Leucine-rich repeat serine/threonine-protein kinase 2
(Homo sapiens (Human))
Elan Pharmaceuticals
Curated by
ChEMBL
Ligand
BDBM50428696
(CHEMBL2333120)
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Affinity Data
IC50: 9nM
Assay Description:
Inhibition of wild type GST-tagged LRRK2 (970 to 2527 amino acid residues) (unknown origin) assessed as inhibition of biotinylated-LRRKtide phosphory...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
In Depth
Details
Article
PubMed
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Target
Macrophage colony-stimulating factor 1 receptor
(Homo sapiens (Human))
Elan Pharmaceuticals
Curated by
ChEMBL
Ligand
BDBM50428696
(CHEMBL2333120)
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Copy InChI
Affinity Data
IC50: 22nM
Assay Description:
Inhibition of CSF1R (unknown origin) by TR-FRET assay in presence of ATP
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Platelet-derived growth factor receptor alpha
(Homo sapiens (Human))
Elan Pharmaceuticals
Curated by
ChEMBL
Ligand
BDBM50428696
(CHEMBL2333120)
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Copy InChI
Affinity Data
IC50: 262nM
Assay Description:
Inhibition of PDGFRalpha (unknown origin) by TR-FRET assay in presence of ATP
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI