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Found 244 Enz. Inhib. hit(s) with Target = 'Calcium release-activated calcium channel protein 1'
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM81818(CAS_1794 | CHEMBL1909810 | HMA | NSC_1794)
Affinity DataKi:  54nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM22913(CHEMBL1237146 | CHEMBL498770 | Iodophenpropit | {[...)
Affinity DataKi:  400nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM22913(CHEMBL1237146 | CHEMBL498770 | Iodophenpropit | {[...)
Affinity DataKi:  560nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM81819(Benzamil | CAS_1937-37-7 | CHEMBL212579 | NSC_1081...)
Affinity DataKi:  2.70E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM16173(3,5-diamino-6-chloro-N-(diaminomethylene)pyrazinam...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM50035057((eltoprazine)1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM50094703(5-(3-Bromo-phenyl)-7-(6-morpholin-4-yl-pyridin-3-y...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM22914(CHEMBL260374 | N-cyclohexyl-4-(1H-imidazol-5-yl)pi...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM22914(CHEMBL260374 | N-cyclohexyl-4-(1H-imidazol-5-yl)pi...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM652093(US11905244, Compound 112)
Affinity DataIC50:  0.200nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM652068(US11905244, Compound 87)
Affinity DataIC50:  0.950nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM652092(US11905244, Compound 111)
Affinity DataIC50:  1.60nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM652087(US11905244, Compound 106)
Affinity DataIC50:  5.01nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM652094(US11905244, Compound 113)
Affinity DataIC50:  5.83nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM652096(US11905244, Compound 115)
Affinity DataIC50:  5.84nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM652067(US11905244, Compound 86)
Affinity DataIC50:  6.34nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM652083(US11905244, Compound 102)
Affinity DataIC50:  9.20nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM652047(US11905244, Compound 66)
Affinity DataIC50:  10.5nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM652077(US11905244, Compound 96)
Affinity DataIC50:  10.9nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM652082(US11905244, Compound 101)
Affinity DataIC50:  11.2nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM652043(US11905244, Compound 62)
Affinity DataIC50:  11.3nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM652060(US11905244, Compound 79)
Affinity DataIC50:  11.7nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM652034(US11905244, Compound 53)
Affinity DataIC50:  13nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM652081(US11905244, Compound 100)
Affinity DataIC50:  14.8nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM652084(US11905244, Compound 103)
Affinity DataIC50:  15.8nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM652080(US11905244, Compound 99)
Affinity DataIC50:  18.2nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM141416(US10668051, Compound Example 67 | US8921364, 67)
Affinity DataIC50:  20.4nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM141426(US10668051, Compound Example 84 | US8921364, 84)
Affinity DataIC50:  20.8nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM652079(US11905244, Compound 98)
Affinity DataIC50:  21.2nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM652063(US11905244, Compound 82)
Affinity DataIC50:  22.4nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM141438(US10668051, Compound Example 104 | US8921364, 104)
Affinity DataIC50:  23nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM652045(US11905244, Compound 64)
Affinity DataIC50:  24.9nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM50204536(CHEMBL3984105)
Affinity DataIC50:  26nMAssay Description:Inhibition of Orai1 (unknown origin) by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM652046(US11905244, Compound 65)
Affinity DataIC50:  30.6nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM141428(US10668051, Compound Example 87 | US8921364, 87)
Affinity DataIC50:  32.6nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM141421(US10668051, Compound Example 78 | US8921364, 78)
Affinity DataIC50:  34.1nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM141424(US10668051, Compound Example 82 | US8921364, 82)
Affinity DataIC50:  35.7nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM141396(US10668051, Compound Example 7 | US8921364, 7)
Affinity DataIC50:  36.4nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM141444(US10668051, Compound Example 114 | US8921364, 114)
Affinity DataIC50:  37.6nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM152937(US8993612, 20)
Affinity DataIC50:  39.2nMT: 2°CAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat # T9033) induced endoplasmic calcium release in Jurkat cells. (see Yasu...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM141442(US10668051, Compound Example 111 | US8921364, 111)
Affinity DataIC50:  47.2nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM141419(US10668051, Compound Example 74 | US8921364, 74)
Affinity DataIC50:  48nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM141418(US10668051, Compound Example 72 | US8921364, 72)
Affinity DataIC50:  48.2nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM141425(US10668051, Compound Example 83 | US8921364, 83)
Affinity DataIC50:  48.2nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM141441(US10668051, Compound Example 108 | US8921364, 108)
Affinity DataIC50:  50.6nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM152932(US8993612, 6)
Affinity DataIC50:  51.3nMT: 2°CAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat # T9033) induced endoplasmic calcium release in Jurkat cells. (see Yasu...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM141448(US10668051, Compound Example 126 | US8921364, 126)
Affinity DataIC50:  52.6nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM152936(US8993612, 18)
Affinity DataIC50:  53.4nMT: 2°CAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat # T9033) induced endoplasmic calcium release in Jurkat cells. (see Yasu...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM141439(US10668051, Compound Example 106 | US8921364, 106)
Affinity DataIC50:  60nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences

Curated by PDSP Ki Database
LigandPNGBDBM141402(US10668051, Compound Example 28 | US8921364, 28)
Affinity DataIC50:  60.3nMAssay Description:Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...More data for this Ligand-Target Pair
In DepthDetails US Patent
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