BDBM103831 SPI-06

SMILES Cc1ccccc1\N=N\c1cc(c2ccccc2c1N)S(O)(=O)=O

InChI Key InChIKey=PIWJSAOBFMHEAW-FMQUCBEESA-N

Data  7 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 7 hits for monomerid = 103831   

TargetSentrin-specific protease 1(Homo sapiens (Human))
Beckman Research Institute of The City of Hope

LigandPNGBDBM103831(SPI-06)
Affinity DataIC50: >6.00E+7nMpH: 7.4Assay Description:Assays were performedby incubating SENPs with various concentrations of the inhibitor (0−60 μM) at RT for 10 min in assay buffer (50 mM Tr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 2(Homo sapiens (Human))
Beckman Research Institute of The City of Hope

LigandPNGBDBM103831(SPI-06)
Affinity DataIC50:  3.62E+3nMpH: 7.4Assay Description:Assays were performedby incubating SENPs with various concentrations of the inhibitor (0−60 μM) at RT for 10 min in assay buffer (50 mM Tr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 1(Homo sapiens (Human))
Beckman Research Institute of The City of Hope

LigandPNGBDBM103831(SPI-06)
Affinity DataIC50:  4.32E+4nMpH: 7.4Assay Description:Assays were performedby incubating SENPs with various concentrations of the inhibitor (0−60 μM) at RT for 10 min in assay buffer (50 mM Tr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 3(Homo sapiens)TBA
LigandPNGBDBM103831(SPI-06)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of SENP3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSentrin-specific protease 1(Homo sapiens (Human))
Beckman Research Institute of The City of Hope

LigandPNGBDBM103831(SPI-06)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibition of SENP1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSentrin-specific protease 2(Homo sapiens (Human))
Beckman Research Institute of The City of Hope

LigandPNGBDBM103831(SPI-06)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of SENP2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSentrin-specific protease 2(Homo sapiens (Human))
Beckman Research Institute of The City of Hope

LigandPNGBDBM103831(SPI-06)
Affinity DataIC50:  1.07E+4nMpH: 7.4Assay Description:Assays were performedby incubating SENPs with various concentrations of the inhibitor (0−60 μM) at RT for 10 min in assay buffer (50 mM Tr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed