BDBM103832 SPI-07::US11041859, Code SPI-07
SMILES Cc1cc(N)ccc1\N=N\c1cc(c2cccc(c2c1)S([O-])(=O)=O)S([O-])(=O)=O
InChI Key InChIKey=XXZDPVOWJBCNQC-FMQUCBEESA-L
Data 11 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 11 hits for monomerid = 103832
TargetSentrin-specific protease 1(Homo sapiens (Human))
Beckman Research Institute of The City of Hope
Beckman Research Institute of The City of Hope
Affinity DataIC50: >6.00E+7nMpH: 7.4Assay Description:Assays were performedby incubating SENPs with various concentrations of the inhibitor (0−60 μM) at RT for 10 min in assay buffer (50 mM Tr...More data for this Ligand-Target Pair
TargetSentrin-specific protease 2(Homo sapiens (Human))
Beckman Research Institute of The City of Hope
Beckman Research Institute of The City of Hope
Affinity DataIC50: >6.00E+4nMpH: 7.4Assay Description:Assays were performedby incubating SENPs with various concentrations of the inhibitor (0−60 μM) at RT for 10 min in assay buffer (50 mM Tr...More data for this Ligand-Target Pair
TargetSentrin-specific protease 1(Homo sapiens (Human))
Beckman Research Institute of The City of Hope
Beckman Research Institute of The City of Hope
Affinity DataIC50: 1.75E+4nMpH: 7.4Assay Description:Assays were performedby incubating SENPs with various concentrations of the inhibitor (0−60 μM) at RT for 10 min in assay buffer (50 mM Tr...More data for this Ligand-Target Pair
TargetSentrin-specific protease 2(Homo sapiens (Human))
Beckman Research Institute of The City of Hope
Beckman Research Institute of The City of Hope
Affinity DataIC50: 2.81E+4nMpH: 7.4Assay Description:Assays were performedby incubating SENPs with various concentrations of the inhibitor (0−60 μM) at RT for 10 min in assay buffer (50 mM Tr...More data for this Ligand-Target Pair
TargetSentrin-specific protease/Small ubiquitin-related modifier 1(Homo sapiens (Human))
City of Hope
US Patent
City of Hope
US Patent
Affinity DataIC50: >6.00E+4nMAssay Description:The inhibitors confer the non-competitive inhibitory mechanism, as shown by nuclear magnetic resonance (NMR) and quantitative enzyme kinetic analysis...More data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+3nMAssay Description:The inhibitors confer the non-competitive inhibitory mechanism, as shown by nuclear magnetic resonance (NMR) and quantitative enzyme kinetic analysis...More data for this Ligand-Target Pair
Affinity DataIC50: 1.75E+4nMAssay Description:The inhibitors confer the non-competitive inhibitory mechanism, as shown by nuclear magnetic resonance (NMR) and quantitative enzyme kinetic analysis...More data for this Ligand-Target Pair
TargetSentrin-specific protease/Small ubiquitin-related modifier 2(Homo sapiens (Human))
City of Hope
US Patent
City of Hope
US Patent
Affinity DataIC50: 2.81E+4nMAssay Description:The inhibitors confer the non-competitive inhibitory mechanism, as shown by nuclear magnetic resonance (NMR) and quantitative enzyme kinetic analysis...More data for this Ligand-Target Pair
TargetSentrin-specific protease 1(Homo sapiens (Human))
Beckman Research Institute of The City of Hope
Beckman Research Institute of The City of Hope
Affinity DataIC50: >6.00E+4nMAssay Description:The inhibitors confer the non-competitive inhibitory mechanism, as shown by nuclear magnetic resonance (NMR) and quantitative enzyme kinetic analysis...More data for this Ligand-Target Pair
TargetSentrin-specific protease 2(Homo sapiens (Human))
Beckman Research Institute of The City of Hope
Beckman Research Institute of The City of Hope
Affinity DataIC50: >6.00E+4nMAssay Description:The inhibitors confer the non-competitive inhibitory mechanism, as shown by nuclear magnetic resonance (NMR) and quantitative enzyme kinetic analysis...More data for this Ligand-Target Pair
TargetSentrin-specific protease 2/Small ubiquitin-related modifier 1(Homo sapiens (Human))
City of Hope
US Patent
City of Hope
US Patent
Affinity DataIC50: >6.00E+4nMAssay Description:The inhibitors confer the non-competitive inhibitory mechanism, as shown by nuclear magnetic resonance (NMR) and quantitative enzyme kinetic analysis...More data for this Ligand-Target Pair