BDBM228839 b-PTHRct-22::biotin-DEEASCPERPPALLQEEWETVM
SMILES CSCC[C@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](C)NC(=O)[C@@H]1CCCN1C(=O)[C@@H]1CCCN1C(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H]1CCCN1C(=O)[C@H](CS)NC(=O)[C@H](CO)NC(=O)[C@H](C)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CC(O)=O)NC(=O)CCCC[C@@H]1SC[C@@H]2NC(=O)N[C@H]12)[C@@H](C)O)C(C)C)C(O)=O
InChI Key
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 228839
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1 [133-300](Homo sapiens (Human))
The University of Queensland
The University of Queensland
Affinity DataKi: 7.00E+3nM ΔG°: -6.98kcal/molepH: 7.4 T: 2°CAssay Description:Competition assays were performed in FP buffer (DTT was avoided for Cys-PTHRct-9) containing fixed concentrations of both the fluorescently labeled p...More data for this Ligand-Target Pair
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1 [133-300](Homo sapiens (Human))
The University of Queensland
The University of Queensland
Affinity DataKd: 1.15E+4nMpH: 7.4 T: 2°CAssay Description:SPR measurements were performed with a Biacore X100 instrument (GE Healthcare Life Sciences, Piscataway, NJ) at 15.0 °C. The biotinylated PTHRct-...More data for this Ligand-Target Pair
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1 [1-140](Homo sapiens (Human))
The University of Queensland
The University of Queensland
Affinity DataKd: 1.60E+4nMpH: 7.4 T: 2°CAssay Description:SPR measurements were performed with a Biacore X100 instrument (GE Healthcare Life Sciences, Piscataway, NJ) at 15.0 °C. The biotinylated PTHRct-...More data for this Ligand-Target Pair