BDBM24710 6-chloro-2-methoxyacridin-9-amine::9-Amino-6-Chloro-2-Methoxyacridine
SMILES COc1ccc2nc3cc(Cl)ccc3c(N)c2c1
InChI Key InChIKey=IHHSSHCBRVYGJX-UHFFFAOYSA-N
Data 4 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 24710
Affinity DataKi: 49nM ΔG°: -9.86kcal/molepH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Estimates of the competitive inhibition constants (Ki) were ob...More data for this Ligand-Target Pair
Affinity DataKi: 5.80E+3nM ΔG°: -7.07kcal/molepH: 7.4 T: 2°CAssay Description:Inhibition constants were calculated by assessment of the reduction in the formation of o-nitrophenol, as monitored by a spectrophotometric assay at ...More data for this Ligand-Target Pair
Affinity DataKi: 7.00E+3nMAssay Description:The competitive inhibitory activity against trypanothione reductase was evaluated from Lineweaver Burk plotsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nM ΔG°: >-5.40kcal/molepH: 7.4 T: 2°CAssay Description:Inhibition constants were calculated by assessment of the reduction in the formation of o-nitrophenol, as monitored by a spectrophotometric assay at ...More data for this Ligand-Target Pair