BDBM461421 US10774069, Compound 1::US11072585, Example 120::US11459309, Compound 2::US11793797, Compound 1
SMILES NCc1cc(Oc2cccc(c2)C(=O)N2C[C@@H](O)[C@H](F)C2)nc(c1)C(F)(F)F
InChI Key InChIKey=ODGXXYXJORZPHE-ZIAGYGMSSA-N
Data 11 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 11 hits for monomerid = 461421
Affinity DataIC50: <300nMAssay Description:LOXL2 amine oxidase activity was evaluated by measuring Amplex Red fluorescence using 10-20× concentrated conditioned media (non BSA-containing) from...More data for this Ligand-Target Pair
Affinity DataIC50: <300nMAssay Description:LOXL2 amine oxidase activity is evaluated by measuring Amplex Red fluorescence using 10-20× concentrated conditioned media from CHO cells stably expr...More data for this Ligand-Target Pair
Affinity DataIC50: <300nMAssay Description:LOXL2 amine oxidase activity is evaluated by measuring Amplex Red fluorescence using 10-20× concentrated conditioned media from CHO cells stably expr...More data for this Ligand-Target Pair
Affinity DataIC50: <300nMAssay Description:LOXL2 amine oxidase activity was evaluated by measuring Amplex Red fluorescence using 10-20× concentrated conditioned media (non BSA-containing) from...More data for this Ligand-Target Pair
Affinity DataIC50: <300nMAssay Description:LOXL2 amine oxidase activity was evaluated by measuring Amplex Red fluorescence using 10-20× concentrated conditioned media (non BSA-containing) from...More data for this Ligand-Target Pair
Affinity DataIC50: 4.70E+4nMAssay Description:Table 9: Human LOX amine oxidase activity was evaluated by measuring Amplex Red fluorescence using 10-20× concentrated conditioned media (BSA-contain...More data for this Ligand-Target Pair
Affinity DataIC50: <300nMAssay Description:Table 8: LOXL2 amine oxidase activity was evaluated by measuring Amplex Red fluorescence using 10-20× concentrated conditioned media (non BSA-contain...More data for this Ligand-Target Pair
Affinity DataIC50: 75.1nMAssay Description:Table 9: Human LOX amine oxidase activity was evaluated by measuring Amplex Red fluorescence using 10-20× concentrated conditioned media (BSA-contain...More data for this Ligand-Target Pair
Affinity DataIC50: 209nMAssay Description:Table 9: The amine oxidase activity was evaluated by measuring Amplex Red fluorescence using commercially available purified, recombinant human LOXL2...More data for this Ligand-Target Pair
Affinity DataIC50: 1.21E+3nMAssay Description:Table 9: The amine oxidase activity was evaluated by measuring Amplex Red fluorescence using commercially available purified, recombinant human LOXL3...More data for this Ligand-Target Pair
Affinity DataIC50: <300nMAssay Description:Table 8: LOXL2 amine oxidase activity was evaluated by measuring Amplex Red fluorescence using 10-20× concentrated conditioned media (non BSA-contain...More data for this Ligand-Target Pair