BDBM50547124 CHEMBL242708::NCI-0001009

SMILES OCc1cc(=O)c(O)c(o1)C(Nc1ccccc1)c1ccccc1

InChI Key InChIKey=SDUJCHJWBKZEPC-UHFFFAOYSA-N

Data  1 KI  6 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 7 hits for monomerid = 50547124   

TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM50547124(CHEMBL242708 | NCI-0001009)
Affinity DataKi:  2.60E+3nMAssay Description:Reversible inhibition of CPM binding to nonacylated N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Codon...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM50547124(CHEMBL242708 | NCI-0001009)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of CPM binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-CodonPlus (DE3)-RIPL cells p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM50547124(CHEMBL242708 | NCI-0001009)
Affinity DataIC50:  200nMAssay Description:Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscriptional enhancer factor TEF-5(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM50547124(CHEMBL242708 | NCI-0001009)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of CPM binding to N-terminal His6-tagged human TEAD3 (216 to 434 residues) expressed in Escherichia coli BL21-CodonPlus (DE3)-RIPL cells p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscriptional enhancer factor TEF-1(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM50547124(CHEMBL242708 | NCI-0001009)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of CPM binding to nonacylated N-terminal His6/GST-tagged human TEAD1 (209 to 426 residues) expressed in Escherichia coli BL21-CodonPlus (D...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscriptional enhancer factor TEF-4(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM50547124(CHEMBL242708 | NCI-0001009)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of CPM binding to nonacylated N-terminal His6-tagged human TEAD2 (217 to 447 residues) expressed in Escherichia coli BL21-CodonPlus (DE3)-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM50547124(CHEMBL242708 | NCI-0001009)
Affinity DataIC50:  70nMAssay Description:Binding affinity to nonacylated N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-CodonPlus (DE3)-RIPL cell...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed