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Found 4 Enz. Inhib. hit(s) with Target = 'Transcriptional enhancer factor TEF-3' and Ligand = 'BDBM50547124'
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM50547124(CHEMBL242708 | NCI-0001009)
Affinity DataKi:  2.60E+3nMAssay Description:Reversible inhibition of CPM binding to nonacylated N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Codon...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM50547124(CHEMBL242708 | NCI-0001009)
Affinity DataIC50:  70nMAssay Description:Binding affinity to nonacylated N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-CodonPlus (DE3)-RIPL cell...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM50547124(CHEMBL242708 | NCI-0001009)
Affinity DataIC50:  200nMAssay Description:Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM50547124(CHEMBL242708 | NCI-0001009)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of CPM binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-CodonPlus (DE3)-RIPL cells p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed