Affinity DataKi: 2.30nMAssay Description:Inhibitory concentration against human Coagulation factor Xa (fXa)More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity against human coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity against human coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity against human coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Binding affinity against human coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Inhibitory concentration against human Coagulation factor Xa(fXa)More data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Inhibitory concentration against human Coagulation factor Xa (fXa)More data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Binding affinity against human coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Inhibitory concentration against human Coagulation factor Xa (fXa)More data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Binding affinity against human coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Binding affinity against human coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:Inhibitory concentration against human Coagulation factor Xa (fXa)More data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Binding affinity against human coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Binding affinity against human coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Binding affinity against human coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 145nMAssay Description:Binding affinity against human coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 159nMAssay Description:Inhibitory concentration against bovine trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Inhibitory concentration against human Coagulation factor Xa (fXa)More data for this Ligand-Target Pair
Affinity DataKi: 220nMAssay Description:Inhibitory concentration against human Coagulation factor Xa (fXa)More data for this Ligand-Target Pair
Affinity DataKi: 275nMAssay Description:Binding affinity of the compound against human Coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 282nMAssay Description:Binding affinity against human coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Binding affinity against human coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Binding affinity against human coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Binding affinity against human coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 320nMAssay Description:Binding affinity against human trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 340nMAssay Description:Binding affinity against human trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 460nMAssay Description:Binding affinity against human trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Binding affinity against human coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Binding affinity against human coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 540nMAssay Description:Binding affinity against human trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 560nMAssay Description:Binding affinity against human trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 630nMAssay Description:Inhibitory concentration against bovine trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 650nMAssay Description:Binding affinity against human trypsinMore data for this Ligand-Target Pair
TargetCytochrome P450 2D6(Homo sapiens (Human))
Albany College Of Pharmacy And Health Sciences
Curated by ChEMBL
Albany College Of Pharmacy And Health Sciences
Curated by ChEMBL
Affinity DataKi: 720nMAssay Description:Time dependent inhibition of CYP2D6 in human liver microsomes assessed as equilibrium inhibition binding constant in presence of NADPH by LC-MS/MS an...More data for this Ligand-Target Pair
Affinity DataKi: 800nMAssay Description:Binding affinity against human coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 850nMAssay Description:Binding affinity against human coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 870nMAssay Description:Non-competitive inhibition of recombinant human AChE expressed in HEK293 cells using varying levels of acetylthiocholine iodide as substrate pretreat...More data for this Ligand-Target Pair
Affinity DataKi: 910nMAssay Description:Binding affinity against human coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 980nMAssay Description:Inhibitory concentration against bovine trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+3nMAssay Description:Binding affinity against human trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 1.18E+3nMAssay Description:Affinity for human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 1.26E+3nMAssay Description:Binding affinity against human trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 1.26E+3nMAssay Description:Affinity for human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 1.35E+3nMAssay Description:Affinity for human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 1.60E+3nMAssay Description:Inhibitory concentration against bovine trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 1.60E+3nMAssay Description:Inhibitory concentration against thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 1.70E+3nMAssay Description:Inhibitory concentration against bovine trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 1.74E+3nMAssay Description:Affinity for human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nMAssay Description:Affinity for human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+3nMAssay Description:Inhibitory concentration against thrombin.More data for this Ligand-Target Pair