TargetVIM-1 metallo-beta-lactamase(Klebsiella pneumoniae)
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of Escherichia coli VIM-1 using fluorocillin as substrate incubated for 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
TargetVIM-1 metallo-beta-lactamase(Klebsiella pneumoniae)
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of Escherichia coli VIM-1 using fluorocillin as substrate incubated for 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
TargetVIM-1 metallo-beta-lactamase(Klebsiella pneumoniae)
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of Escherichia coli VIM-1 using fluorocillin as substrate incubated for 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
TargetVIM-1 metallo-beta-lactamase(Klebsiella pneumoniae)
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of Escherichia coli VIM-1 using fluorocillin as substrate incubated for 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
TargetVIM-1 metallo-beta-lactamase(Klebsiella pneumoniae)
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of Escherichia coli VIM-1 using fluorocillin as substrate incubated for 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
TargetVIM-1 metallo-beta-lactamase(Klebsiella pneumoniae)
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of Escherichia coli VIM-1 using fluorocillin as substrate incubated for 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
TargetVIM-1 metallo-beta-lactamase(Klebsiella pneumoniae)
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Inhibition of Escherichia coli VIM-1 using fluorocillin as substrate incubated for 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
TargetVIM-1 metallo-beta-lactamase(Klebsiella pneumoniae)
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of Escherichia coli VIM-1 using fluorocillin as substrate incubated for 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
TargetVIM-1 metallo-beta-lactamase(Klebsiella pneumoniae)
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of Escherichia coli VIM-1 using fluorocillin as substrate incubated for 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
TargetVIM-1 metallo-beta-lactamase(Klebsiella pneumoniae)
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Inhibition of Escherichia coli VIM-1 using fluorocillin as substrate incubated for 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
TargetNeutrophil collagenase(Homo sapiens (Human))
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Inhibition of human MMP-8More data for this Ligand-Target Pair
TargetVIM-1 metallo-beta-lactamase(Klebsiella pneumoniae)
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of Escherichia coli VIM-1 using fluorocillin as substrate incubated for 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
TargetVIM-1 metallo-beta-lactamase(Klebsiella pneumoniae)
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of Escherichia coli VIM-1 using fluorocillin as substrate incubated for 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
TargetVIM-1 metallo-beta-lactamase(Klebsiella pneumoniae)
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:Inhibition of Escherichia coli VIM-1 using fluorocillin as substrate incubated for 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
TargetVIM-1 metallo-beta-lactamase(Klebsiella pneumoniae)
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of Escherichia coli VIM-1 using fluorocillin as substrate incubated for 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
TargetVIM-1 metallo-beta-lactamase(Klebsiella pneumoniae)
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of Escherichia coli VIM-1 using fluorocillin as substrate incubated for 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
TargetVIM-1 metallo-beta-lactamase(Klebsiella pneumoniae)
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of Escherichia coli VIM-1 using fluorocillin as substrate incubated for 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
TargetVIM-1 metallo-beta-lactamase(Klebsiella pneumoniae)
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of Escherichia coli VIM-1 using fluorocillin as substrate incubated for 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
TargetVIM-1 metallo-beta-lactamase(Klebsiella pneumoniae)
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of Escherichia coli VIM-1 using fluorocillin as substrate incubated for 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
TargetVIM-1 metallo-beta-lactamase(Klebsiella pneumoniae)
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of Escherichia coli VIM-1 using fluorocillin as substrate incubated for 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
Target72 kDa type IV collagenase(Homo sapiens (Human))
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of human MMP-2More data for this Ligand-Target Pair
TargetVIM-1 metallo-beta-lactamase(Klebsiella pneumoniae)
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of Escherichia coli VIM-1 using fluorocillin as substrate incubated for 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
TargetVIM-1 metallo-beta-lactamase(Klebsiella pneumoniae)
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of Escherichia coli VIM-1 using fluorocillin as substrate incubated for 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
TargetVIM-1 metallo-beta-lactamase(Klebsiella pneumoniae)
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of Escherichia coli VIM-1 using fluorocillin as substrate incubated for 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
TargetInterstitial collagenase(Homo sapiens (Human))
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of human MMP-1More data for this Ligand-Target Pair
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of human MMP-14More data for this Ligand-Target Pair
TargetStromelysin-1(Homo sapiens (Human))
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of human MMP-3More data for this Ligand-Target Pair
TargetElastase(Pseudomonas aeruginosa)
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa PA14 LasB elastase preincubated for 15 mins followed by substrate addition and measured after 60 mins using 2-am...More data for this Ligand-Target Pair
TargetElastase(Pseudomonas aeruginosa)
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Affinity DataIC50: 6.60E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa PA14 LasB elastase preincubated for 15 mins followed by substrate addition and measured after 60 mins using 2-am...More data for this Ligand-Target Pair
TargetMatrilysin(Homo sapiens (Human))
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of human MMP-7More data for this Ligand-Target Pair
TargetVIM-1 metallo-beta-lactamase(Klebsiella pneumoniae)
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Escherichia coli VIM-1 using fluorocillin as substrate incubated for 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
TargetElastase(Pseudomonas aeruginosa)
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa PA14 LasB elastase preincubated for 15 mins followed by substrate addition and measured after 60 mins using 2-am...More data for this Ligand-Target Pair
TargetElastase(Pseudomonas aeruginosa)
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa PA14 LasB elastase preincubated for 15 mins followed by substrate addition and measured after 60 mins using 2-am...More data for this Ligand-Target Pair
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of human MMP-14More data for this Ligand-Target Pair
TargetElastase(Pseudomonas aeruginosa)
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa PA14 LasB elastase preincubated for 15 mins followed by substrate addition and measured after 60 mins using 2-am...More data for this Ligand-Target Pair
TargetElastase(Pseudomonas aeruginosa)
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa PA14 LasB elastase preincubated for 15 mins followed by substrate addition and measured after 60 mins using 2-am...More data for this Ligand-Target Pair
TargetElastase(Pseudomonas aeruginosa)
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa PA14 LasB elastase preincubated for 15 mins followed by substrate addition and measured after 60 mins using 2-am...More data for this Ligand-Target Pair
TargetElastase(Pseudomonas aeruginosa)
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa PA14 LasB elastase preincubated for 15 mins followed by substrate addition and measured after 60 mins using 2-am...More data for this Ligand-Target Pair
TargetElastase(Pseudomonas aeruginosa)
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa PA14 LasB elastase preincubated for 15 mins followed by substrate addition and measured after 60 mins using 2-am...More data for this Ligand-Target Pair
TargetElastase(Pseudomonas aeruginosa)
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa PA14 LasB elastase preincubated for 15 mins followed by substrate addition and measured after 60 mins using 2-am...More data for this Ligand-Target Pair
TargetElastase(Pseudomonas aeruginosa)
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa PA14 LasB elastase preincubated for 15 mins followed by substrate addition and measured after 60 mins using 2-am...More data for this Ligand-Target Pair
TargetElastase(Pseudomonas aeruginosa)
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa PA14 LasB elastase preincubated for 15 mins followed by substrate addition and measured after 60 mins using 2-am...More data for this Ligand-Target Pair
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of human MMP-14More data for this Ligand-Target Pair
TargetElastase(Pseudomonas aeruginosa)
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Affinity DataIC50: 3.60E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa PA14 LasB elastase preincubated for 15 mins followed by substrate addition and measured after 60 mins using 2-am...More data for this Ligand-Target Pair
TargetElastase(Pseudomonas aeruginosa)
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Affinity DataIC50: 3.80E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa PA14 LasB elastase preincubated for 15 mins followed by substrate addition and measured after 60 mins using 2-am...More data for this Ligand-Target Pair
TargetElastase(Pseudomonas aeruginosa)
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Affinity DataIC50: 3.90E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa PA14 LasB elastase preincubated for 15 mins followed by substrate addition and measured after 60 mins using 2-am...More data for this Ligand-Target Pair
TargetElastase(Pseudomonas aeruginosa)
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Affinity DataIC50: 4.80E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa PA14 LasB elastase preincubated for 15 mins followed by substrate addition and measured after 60 mins using 2-am...More data for this Ligand-Target Pair
TargetElastase(Pseudomonas aeruginosa)
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Affinity DataIC50: 4.80E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa PA14 LasB elastase preincubated for 15 mins followed by substrate addition and measured after 60 mins using 2-am...More data for this Ligand-Target Pair
TargetElastase(Pseudomonas aeruginosa)
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Affinity DataIC50: 5.20E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa PA14 LasB elastase preincubated for 15 mins followed by substrate addition and measured after 60 mins using 2-am...More data for this Ligand-Target Pair
TargetElastase(Pseudomonas aeruginosa)
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Helmholtz Institute For Pharmaceutical Research Saarland (Hips)
Curated by ChEMBL
Affinity DataIC50: 5.40E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa PA14 LasB elastase preincubated for 15 mins followed by substrate addition and measured after 60 mins using 2-am...More data for this Ligand-Target Pair
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