Affinity DataKi: 0.310nMAssay Description:Mixed-type inhibition of recombinant human MAO-B expressed in Pichia pastoris using benzylamine as substrate by fluorimetric horseradish peroxidase-A...More data for this Ligand-Target Pair
Affinity DataKi: 0.670nMAssay Description:Non-competitive inhibition of human microsomal MAO-B expressed in recombinant baculovirus infected insect BTI-TN-5B1-4 cells assessed as reduction in...More data for this Ligand-Target Pair
Affinity DataKi: 0.790nMAssay Description:Competitive inhibition of human microsomal MAO-B expressed in recombinant baculovirus infected insect BTI-TN-5B1-4 cells assessed as reduction in H2O...More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Noncompetitive inhibition of human recombinant microsomal MAOB expressed in baculovirus infected BTI-TN-5B1- 4 cells using p-tyramine as substrate as...More data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Inhibition of human recombinant microsomal MAOB expressed in baculovirus infected BTI-TN-5B1- 4 cells using p-tyramine as substrate assessed as decre...More data for this Ligand-Target Pair
Affinity DataKi: 7.5nMAssay Description:Non-competitive inhibition of recombinant human MAO-B expressed in Pichia pastoris using benzylamine as substrate by fluorimetric horseradish peroxid...More data for this Ligand-Target Pair
Affinity DataKi: 10.4nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cells after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Porto
Curated by ChEMBL
University Of Porto
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Inhibition of electric eel AChE assessed as inhibition constant using acetylthiocholine iodide as substrate pretreated for 5 mins followed by substra...More data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Tight-binding competitive inhibition of recombinant human MAO-B expressed in Pichia pastoris using benzylamine as substrate by fluorimetric horseradi...More data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Competitive inhibition of human microsomal MAO-B expressed in baculovirus infected BTI-TN-5B1-4 cells assessed as inhibition constant using kynuramin...More data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Tight-binding competitive inhibition of recombinant human MAO-B expressed in Pichia pastoris using benzylamine as substrate by fluorimetric horseradi...More data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Tight-binding competitive inhibition of recombinant human MAO-B expressed in Pichia pastoris using benzylamine as substrate by fluorimetric horseradi...More data for this Ligand-Target Pair
Affinity DataKi: 44nMAssay Description:Competitive inhibition of human microsomal MAO-B expressed in baculovirus infected BTI-TN-5B1-4 cells assessed as inhibition constant using kynuramin...More data for this Ligand-Target Pair
Affinity DataKi: 55nMAssay Description:Tight-binding competitive inhibition of recombinant human MAO-B expressed in Pichia pastoris using benzylamine as substrate by fluorimetric horseradi...More data for this Ligand-Target Pair
Affinity DataKi: 57nMAssay Description:Reversible competitive inhibition of human recombinant microsomal MAOA expressed in baculovirus infected BTI-TN-5B1- 4 cells using p-tyramine as subs...More data for this Ligand-Target Pair
Affinity DataKi: 75nMAssay Description:Competitive inhibition of human microsomal MAO-B expressed in baculovirus infected BTI-TN-5B1-4 cells assessed as inhibition constant using kynuramin...More data for this Ligand-Target Pair
Affinity DataKi: 190nMAssay Description:Mixed type inhibition of human AChE using acetylthiocholine iodide as substrate pretreated for 5 mins followed by substrate addition measured after 5...More data for this Ligand-Target Pair
Affinity DataKi: 258nMAssay Description:Displacement of [3H]HEMADO from human adenosine receptor A3 expressed in CHO cell membranes by radioligand competition assayMore data for this Ligand-Target Pair
Affinity DataKi: 337nMAssay Description:Reversible competitive inhibition of human recombinant microsomal MAOB expressed in baculovirus infected BTI-TN-5B1- 4 cells using p-tyramine as subs...More data for this Ligand-Target Pair
Affinity DataKi: 478nMAssay Description:Reversible competitive inhibition of human recombinant microsomal MAOB expressed in baculovirus infected BTI-TN-5B1- 4 cells using p-tyramine as subs...More data for this Ligand-Target Pair
Affinity DataKi: 1.35E+3nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cells after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.71E+3nMAssay Description:Displacement of [3H]NECA from human adenosine receptor A2A expressed in CHO cell membranes by radioligand competition assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.40E+3nMAssay Description:Displacement of [3H]CCPA from human adenosine receptor A1 expressed in CHO cell membranes by radioligand competition assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.89E+3nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cells after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.93E+3nMAssay Description:Tight-binding competitive inhibition of recombinant human MAO-B expressed in Pichia pastoris using benzylamine as substrate by fluorimetric horseradi...More data for this Ligand-Target Pair
Affinity DataKi: 3.24E+3nMAssay Description:The radioligands used were 1 nM (2R,3R,4S,5R)-2-(2-chloro-6-cyclopentylamino-purin-9-yl)-5-hydroxymethyl-tetrahydro-3,4-diol ([3H]CCPA) for hA1, 10 n...More data for this Ligand-Target Pair
Affinity DataKi: 3.85E+3nMAssay Description:Displacement of [3H]HEMADO from human adenosine receptor A3 expressed in CHO cell membranes by radioligand competition assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.93E+3nMAssay Description:Displacement of [3H]HEMADO from human adenosine receptor A3 expressed in CHO cell membranes by radioligand competition assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.62E+3nMAssay Description:Displacement of [3H]CCPA from human adenosine receptor A1 expressed in CHO cell membranes by radioligand competition assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.06E+3nMAssay Description:Displacement of [3H]HEMADO from human adenosine receptor A3 expressed in CHO cell membranes by radioligand competition assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.09E+3nMAssay Description:Displacement of [3H]HEMADO from human adenosine receptor A3 expressed in CHO cell membranes by radioligand competition assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.17E+3nMAssay Description:Displacement of [3H]HEMADO from human adenosine receptor A3 expressed in CHO cell membranes by radioligand competition assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.18E+3nMAssay Description:The radioligands used were 1 nM (2R,3R,4S,5R)-2-(2-chloro-6-cyclopentylamino-purin-9-yl)-5-hydroxymethyl-tetrahydro-3,4-diol ([3H]CCPA) for hA1, 10 n...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Porto
Curated by ChEMBL
University Of Porto
Curated by ChEMBL
Affinity DataKi: 5.20E+3nMAssay Description:Inhibition of electric eel AChE assessed as inhibition constant using acetylthiocholine iodide as substrate pretreated for 5 mins followed by substra...More data for this Ligand-Target Pair
Affinity DataKi: 5.32E+3nMAssay Description:Displacement of [3H]HEMADO from human adenosine receptor A3 expressed in CHO cell membranes by radioligand competition assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.82E+3nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cells after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 6.14E+3nMAssay Description:Displacement of [3H]HEMADO from human adenosine receptor A3 expressed in CHO cell membranes by radioligand competition assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.20E+3nMAssay Description:Displacement of [3H]CCPA from human adenosine receptor A1 expressed in CHO cell membranes by radioligand competition assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.28E+3nMAssay Description:Displacement of [3H]CCPA from human adenosine receptor A1 expressed in CHO cell membranes by radioligand competition assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.39E+3nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cells after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 6.77E+3nMAssay Description:Displacement of [3H]CCPA from human adenosine receptor A1 expressed in CHO cell membranes by radioligand competition assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.86E+3nMAssay Description:Displacement of [3H]HEMADO from human adenosine receptor A3 expressed in CHO cell membranes by radioligand competition assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.93E+3nMAssay Description:Displacement of [3H]CCPA from human adenosine receptor A1 expressed in CHO cell membranes by radioligand competition assayMore data for this Ligand-Target Pair
Affinity DataKi: 7.06E+3nMAssay Description:Displacement of [3H]HEMADO from human adenosine receptor A3 expressed in CHO cell membranes by radioligand competition assayMore data for this Ligand-Target Pair
Affinity DataKi: 8.02E+3nMAssay Description:Displacement of [3H]HEMADO from human adenosine receptor A3 expressed in CHO cell membranes by radioligand competition assayMore data for this Ligand-Target Pair
Affinity DataKi: 8.50E+3nMAssay Description:Displacement of [3H]HEMADO from human adenosine receptor A3 expressed in CHO cell membranes by radioligand competition assayMore data for this Ligand-Target Pair
Affinity DataKi: 8.51E+3nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cells after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 8.56E+3nMAssay Description:Displacement of [3H]CCPA from human adenosine receptor A1 expressed in CHO cell membranes by radioligand competition assayMore data for this Ligand-Target Pair
Affinity DataKi: 8.95E+3nMAssay Description:The radioligands used were 1 nM (2R,3R,4S,5R)-2-(2-chloro-6-cyclopentylamino-purin-9-yl)-5-hydroxymethyl-tetrahydro-3,4-diol ([3H]CCPA) for hA1, 10 n...More data for this Ligand-Target Pair
Affinity DataKi: 9.05E+3nMAssay Description:Displacement of [3H]HEMADO from human adenosine receptor A3 expressed in CHO cell membranes by radioligand competition assayMore data for this Ligand-Target Pair