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Found 96 with Last Name = 'camarda' and Initial = 'v'
TargetNociceptin receptor(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50181392((R)-N-(3-(3H-spiro[isobenzofuran-1,4'-piperidine]-...)
Affinity DataKi:  0.240nMAssay Description:Displacement of [3H]N/OFQ from human recombinant NOP receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50000788((morphine)4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-az...)
Affinity DataKi:  0.562nMAssay Description:Displacement of [3H]DPN from human recombinant mu-type opioid receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetNociceptin receptor(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50418594(CHEMBL1783826)
Affinity DataKi:  0.724nMAssay Description:Displacement of [3H]N/OFQ from human recombinant NOP receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50000788((morphine)4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-az...)
Affinity DataKi:  4.5nMAssay Description:Displacement of [3H]DPN from human recombinant kappa-type opioid receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50000788((morphine)4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-az...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]DPN from human recombinant delta-type opioid receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetNociceptin receptor(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50418589(CHEMBL1783821)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]N/OFQ from human recombinant NOP receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50418598(CHEMBL1783818)
Affinity DataKi:  59nMAssay Description:Displacement of [3H]N/OFQ from human recombinant NOP receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50418587(CHEMBL1783817)
Affinity DataKi:  59nMAssay Description:Displacement of [3H]N/OFQ from human recombinant NOP receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50418588(CHEMBL1783819)
Affinity DataKi:  60nMAssay Description:Displacement of [3H]N/OFQ from human recombinant NOP receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50418595(CHEMBL1783827)
Affinity DataKi:  83nMAssay Description:Displacement of [3H]N/OFQ from human recombinant NOP receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50418590(CHEMBL1783822)
Affinity DataKi:  107nMAssay Description:Displacement of [3H]N/OFQ from human recombinant NOP receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50418591(CHEMBL1783823)
Affinity DataKi:  158nMAssay Description:Displacement of [3H]N/OFQ from human recombinant NOP receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50418594(CHEMBL1783826)
Affinity DataKi:  191nMAssay Description:Displacement of [3H]DPN from human recombinant mu-type opioid receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50418594(CHEMBL1783826)
Affinity DataKi:  316nMAssay Description:Displacement of [3H]DPN from human recombinant kappa-type opioid receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50418594(CHEMBL1783826)
Affinity DataKi: <1.00E+3nMAssay Description:Displacement of [3H]DPN from human recombinant delta-type opioid receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50418597(CHEMBL1783820)
Affinity DataKi:  1.15E+3nMAssay Description:Displacement of [3H]N/OFQ from human recombinant NOP receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50418593(CHEMBL1783825)
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of [3H]N/OFQ from human recombinant NOP receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50418592(CHEMBL1783824)
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of [3H]N/OFQ from human recombinant NOP receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50418596(CHEMBL1783828)
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of [3H]N/OFQ from human recombinant NOP receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50423102(CHEMBL267479)
Affinity DataIC50:  537nMAssay Description:Antagonist activity at mouse NPSR expressed in HEK293 cells assessed as inhibition of 10 nM hNPS-induced calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50423102(CHEMBL267479)
Affinity DataIC50:  1.62E+3nMAssay Description:Antagonist activity at mouse NPSR expressed in HEK293 cells assessed as inhibition of 100 nM hNPS-induced calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50479767(CHEMBL451444)
Affinity DataEC50:  562nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells assessed as increase in intracellular calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50479768(CHEMBL503441)
Affinity DataEC50:  372nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells assessed as increase in intracellular calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50479769(CHEMBL510338)
Affinity DataEC50:  32nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells assessed as increase in intracellular calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50479770(CHEMBL500802)
Affinity DataEC50:  1.55E+3nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells assessed as increase in intracellular calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50479771(CHEMBL447434)
Affinity DataEC50:  166nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells assessed as increase in intracellular calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50479772(CHEMBL525031)
Affinity DataEC50:  85nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells assessed as increase in intracellular calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50479773(CHEMBL524688)
Affinity DataEC50:  22nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells assessed as increase in intracellular calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50479774(CHEMBL506383)
Affinity DataEC50:  129nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells assessed as increase in intracellular calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50479775(CHEMBL510673)
Affinity DataEC50:  204nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells assessed as increase in intracellular calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50479776(CHEMBL505996)
Affinity DataEC50:  240nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells assessed as increase in intracellular calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50479777(CHEMBL499957)
Affinity DataEC50:  1.26E+3nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells assessed as increase in intracellular calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50413782(CHEMBL1627325)
Affinity DataEC50:  1.90nMAssay Description:Antagonist activity at human recombinant delta opioid receptor expressed in CHO cells coexpressing alphaqi5 assessed as inhibition of DPDPE-induced i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50004178(Nociceptin | Nociceptin/orphanin FQ | ORPHANIN FQ)
Affinity DataEC50:  0.389nMAssay Description:Antagonist activity at human recombinant NOP receptor expressed in CHO cells coexpressing alphaqi5 assessed as inhibition of N/OFQ-induced intracellu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50001683(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataEC50:  3nMAssay Description:Antagonist activity at human recombinant delta opioid receptor expressed in CHO cells coexpressing alphaqi5 assessed as inhibition of DPDPE-induced i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50412700(CHEMBL526492)
Affinity DataEC50:  70.8nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50412701(CHEMBL525809)
Affinity DataEC50:  2.24nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50412702(CHEMBL526323)
Affinity DataEC50:  229nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50412703(CHEMBL505657)
Affinity DataEC50:  66.1nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50412704(CHEMBL507881)
Affinity DataEC50:  87.1nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50412705(CHEMBL526355)
Affinity DataEC50:  13.8nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50412706(CHEMBL525398)
Affinity DataEC50:  776nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50412707(CHEMBL230333)
Affinity DataEC50:  2.24nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50412707(CHEMBL230333)
Affinity DataEC50:  4.80nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50413778(CHEMBL500443)
Affinity DataEC50:  1.66E+3nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50413779(CHEMBL500458)
Affinity DataEC50:  661nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50413780(CHEMBL507664)
Affinity DataEC50:  2.69E+3nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50413781(CHEMBL509091)
Affinity DataEC50:  794nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
National Institute Of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50413782(CHEMBL1627325)
Affinity DataEC50:  0.0490nMAssay Description:Antagonist activity at human recombinant NK1 receptor expressed in CHO cells assessed as inhibition of NPS-induced intracellular calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
National Institute Of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50413782(CHEMBL1627325)
Affinity DataEC50:  0.0339nMAssay Description:Antagonist activity at human recombinant bradykinin 2 receptor expressed in CHO cells assessed as inhibition of bradykinin-induced intracellular calc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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