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Found 1150 with Last Name = 'cheng' and Initial = 'f'
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50370582(CHEMBL1791306)
Affinity DataKi: >0.0700nMAssay Description:Inhibition of human somatostatin receptor type 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
East China University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50268107(CHEMBL485862 | CHEMBL500634 | N-(2-(2-phenyl-6-(4-...)
Affinity DataKi:  0.5nMAssay Description:Antagonist activity against human adenosine A2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
East China University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM21173(1,3-dipropyl-8-cyclopentylxanthine | 8-cyclopentyl...)
Affinity DataKi:  0.900nMAssay Description:Antagonist activity against human adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50370578(CHEMBL1791304)
Affinity DataKi:  1nMAssay Description:Inhibition of human somatostatin receptor type 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50370577(CHEMBL1791312)
Affinity DataKi:  1nMAssay Description:Inhibition of human somatostatin receptor type 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
East China University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50086173(CHEMBL17002 | N-(4-Acetyl-phenyl)-2-[4-(2,6-dioxo-...)
Affinity DataKi:  1.39nMAssay Description:Antagonist activity against human adenosine A2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
East China University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50086170((4-Cyano-phenyl)-carbamic acid 4-(2,6-dioxo-1,3-di...)
Affinity DataKi:  1.97nMAssay Description:Antagonist activity against human adenosine A2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50000788((morphine)4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-az...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-naloxone from rat mu opioid receptor expressed in HEK cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
East China University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50086165(2-(4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H...)
Affinity DataKi:  2.13nMAssay Description:Antagonist activity against human adenosine A2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221531(6-methoxy-7-(3-(4-methylpiperazin-1-yl)propoxy)-4-...)
Affinity DataKi:  3nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
East China University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50190709(8-(4-(4-benzylpiperazin-1-ylsulfonyl)phenyl)-1-pro...)
Affinity DataKi:  3.60nMAssay Description:Antagonist activity against human adenosine A2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50370582(CHEMBL1791306)
Affinity DataKi:  3.70nMAssay Description:Inhibition of human somatostatin receptor type 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
East China University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50190706(8-[4-(benzylamidosulfonyl)phenyl]-1-propylxanthine...)
Affinity DataKi:  4.20nMAssay Description:Antagonist activity against human adenosine A2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
East China University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50229885(CHEMBL260331 | CHEMBL506685 | N-(benzo[d][1,3]diox...)
Affinity DataKi:  5.5nMAssay Description:Antagonist activity against human adenosine A2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
East China University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50233088(1-ethyl-8-(1-(3-(trifluoromethyl)benzyl)-1H-pyrazo...)
Affinity DataKi:  6nMAssay Description:Antagonist activity against human adenosine A2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50370580(CHEMBL1791307)
Affinity DataKi:  6.30nMAssay Description:Inhibition of human somatostatin receptor type 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
East China University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50233086(8-(1-((5-(4-chlorophenyl)-1,2,4-oxadiazol-3-yl)met...)
Affinity DataKi:  7nMAssay Description:Antagonist activity against human adenosine A2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50370578(CHEMBL1791304)
Affinity DataKi:  7nMAssay Description:Inhibition of human somatostatin receptor type 2 (n=6)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221516(6-methoxy-7-(3-morpholinopropoxy)-4-((1R,2S)-2-phe...)
Affinity DataKi:  8.40nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
East China University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50086176(CHEMBL275149 | N,N-Dibenzyl-2-[4-(2,6-dioxo-1,3-di...)
Affinity DataKi:  9.88nMAssay Description:Antagonist activity against human adenosine A2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
East China University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50322845(3-methyl-1-propyl-8-(1-(3-(trifluoromethyl)benzyl)...)
Affinity DataKi:  14nMAssay Description:Antagonist activity against human adenosine A2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50370581(CHEMBL1791310)
Affinity DataKi:  20nMAssay Description:Inhibition of human somatostatin receptor type 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50370583(CHEMBL1791311)
Affinity DataKi:  20nMAssay Description:Inhibition of human somatostatin receptor type 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
East China University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50322843(1-(cyclopropylmethyl)-3-ethyl-8-(1-(3-(trifluorome...)
Affinity DataKi:  22nMAssay Description:Antagonist activity against human adenosine A2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
East China University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50188569(8-(1-(2-chloro-5-(trifluoromethyl)benzyl)-1H-pyraz...)
Affinity DataKi:  22nMAssay Description:Antagonist activity against human adenosine A2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
East China University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50322846(3-ethyl-1-propyl-8-(1-((pyridin-3-yl)methyl)-1H-py...)
Affinity DataKi:  22nMAssay Description:Antagonist activity against human adenosine A2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221518(6,7-dimethoxy-4-((1R,2S)-2-phenylcyclopropylamino)...)
Affinity DataKi:  24nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221531(6-methoxy-7-(3-(4-methylpiperazin-1-yl)propoxy)-4-...)
Affinity DataKi:  27nMAssay Description:Inhibition of SRCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221535(4-((1R,2S)-2-(2-fluorophenyl)cyclopropylamino)-6,7...)
Affinity DataKi:  36nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221522(6-(4-(aminomethyl)phenyl)-4-((1R,2S)-2-phenylcyclo...)
Affinity DataKi:  40nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
East China University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50254264(3-(2-Fluorobenzyl)-7-(2-oxazolyl)-3H-[1,2,3]triazo...)
Affinity DataKi:  41nMAssay Description:Antagonist activity against human adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221531(6-methoxy-7-(3-(4-methylpiperazin-1-yl)propoxy)-4-...)
Affinity DataKi:  41nMAssay Description:Inhibition of SYKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221531(6-methoxy-7-(3-(4-methylpiperazin-1-yl)propoxy)-4-...)
Affinity DataKi:  44nMAssay Description:Inhibition of ABLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221530(6,7-diethyl-2-ethynyl-1-(((1S,2R)-2-p-tolylcyclopr...)
Affinity DataKi:  44nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221516(6-methoxy-7-(3-morpholinopropoxy)-4-((1R,2S)-2-phe...)
Affinity DataKi:  45nMAssay Description:Inhibition of SRCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221524(6-methoxy-4-((1R,2S)-2-phenylcyclopropylamino)-7-(...)
Affinity DataKi:  49nMAssay Description:Inhibition of SRCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
East China University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50322844(3-ethyl-1-propyl-8-(1H-pyrazol-4-yl)-1H-purine-2,6...)
Affinity DataKi:  49nMAssay Description:Antagonist activity against human adenosine A2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221527(7-methoxy-6-(3-morpholinopropoxy)-4-((1R,2S)-2-phe...)
Affinity DataKi:  52nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221533(4-((1R,2S)-2-(3-bromophenyl)cyclopropylamino)-6,7-...)
Affinity DataKi:  52nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
East China University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50188569(8-(1-(2-chloro-5-(trifluoromethyl)benzyl)-1H-pyraz...)
Affinity DataKi:  54nMAssay Description:Antagonist activity against human adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
East China University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50190706(8-[4-(benzylamidosulfonyl)phenyl]-1-propylxanthine...)
Affinity DataKi:  54.8nMAssay Description:Antagonist activity against human adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
East China University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM21173(1,3-dipropyl-8-cyclopentylxanthine | 8-cyclopentyl...)
Affinity DataKi:  56nMAssay Description:Antagonist activity against human adenosine A2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50370578(CHEMBL1791304)
Affinity DataKi:  60nMAssay Description:Inhibition of human somatostatin receptor type 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221517(6-methoxy-7-(2-methoxyethoxy)-4-((1R,2S)-2-phenylc...)
Affinity DataKi:  60nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
East China University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50190708(2-(4-(1,3-dimethyl-2,6-dioxo-2,3,6,7-tetrahydro-1H...)
Affinity DataKi:  64nMAssay Description:Antagonist activity against rat adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221521(7-methoxy-6-(2-morpholinoethoxy)-4-((1R,2S)-2-phen...)
Affinity DataKi:  64nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221528(7-methoxy-4-((1R,2S)-2-phenylcyclopropylamino)-6-(...)
Affinity DataKi:  68nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
East China University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50254006(3-(4-Cyanobenzyl)-7-(2-furyl)-3H-[1,2,3]triazolo[4...)
Affinity DataKi:  73nMAssay Description:Antagonist activity against human adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50370578(CHEMBL1791304)
Affinity DataKi:  77nMAssay Description:Inhibition of human somatostatin receptor type 4 (n=5)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221532(6,7-dimethoxy-4-((1R,2S)-2-(4-phenoxyphenyl)cyclop...)
Affinity DataKi:  80nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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