Affinity DataKi: >0.0700nMAssay Description:Inhibition of human somatostatin receptor type 2More data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
East China University Of Science And Technology
Curated by ChEMBL
East China University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:Antagonist activity against human adenosine A2B receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
East China University Of Science And Technology
Curated by ChEMBL
East China University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 0.900nMAssay Description:Antagonist activity against human adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of human somatostatin receptor type 2More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of human somatostatin receptor type 2More data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
East China University Of Science And Technology
Curated by ChEMBL
East China University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 1.39nMAssay Description:Antagonist activity against human adenosine A2B receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
East China University Of Science And Technology
Curated by ChEMBL
East China University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 1.97nMAssay Description:Antagonist activity against human adenosine A2B receptorMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Health Research Institutes
Curated by ChEMBL
National Health Research Institutes
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Displacement of [3H]-naloxone from rat mu opioid receptor expressed in HEK cells after 60 minsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
East China University Of Science And Technology
Curated by ChEMBL
East China University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 2.13nMAssay Description:Antagonist activity against human adenosine A2B receptorMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa
Curated by ChEMBL
Tanabe Research Laboratories Usa
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
East China University Of Science And Technology
Curated by ChEMBL
East China University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 3.60nMAssay Description:Antagonist activity against human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Inhibition of human somatostatin receptor type 4More data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
East China University Of Science And Technology
Curated by ChEMBL
East China University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 4.20nMAssay Description:Antagonist activity against human adenosine A2B receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
East China University Of Science And Technology
Curated by ChEMBL
East China University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 5.5nMAssay Description:Antagonist activity against human adenosine A2B receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
East China University Of Science And Technology
Curated by ChEMBL
East China University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 6nMAssay Description:Antagonist activity against human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Inhibition of human somatostatin receptor type 2More data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
East China University Of Science And Technology
Curated by ChEMBL
East China University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 7nMAssay Description:Antagonist activity against human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Inhibition of human somatostatin receptor type 2 (n=6)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa
Curated by ChEMBL
Tanabe Research Laboratories Usa
Curated by ChEMBL
Affinity DataKi: 8.40nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
East China University Of Science And Technology
Curated by ChEMBL
East China University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 9.88nMAssay Description:Antagonist activity against human adenosine A2B receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
East China University Of Science And Technology
Curated by ChEMBL
East China University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Antagonist activity against human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Inhibition of human somatostatin receptor type 2More data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Inhibition of human somatostatin receptor type 2More data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
East China University Of Science And Technology
Curated by ChEMBL
East China University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Antagonist activity against human adenosine A2B receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
East China University Of Science And Technology
Curated by ChEMBL
East China University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Antagonist activity against human adenosine A2B receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
East China University Of Science And Technology
Curated by ChEMBL
East China University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Antagonist activity against human adenosine A2B receptorMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa
Curated by ChEMBL
Tanabe Research Laboratories Usa
Curated by ChEMBL
Affinity DataKi: 24nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Tanabe Research Laboratories Usa
Curated by ChEMBL
Tanabe Research Laboratories Usa
Curated by ChEMBL
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa
Curated by ChEMBL
Tanabe Research Laboratories Usa
Curated by ChEMBL
Affinity DataKi: 36nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa
Curated by ChEMBL
Tanabe Research Laboratories Usa
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
East China University Of Science And Technology
Curated by ChEMBL
East China University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 41nMAssay Description:Antagonist activity against human adenosine A2A receptorMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Tanabe Research Laboratories Usa
Curated by ChEMBL
Tanabe Research Laboratories Usa
Curated by ChEMBL
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Tanabe Research Laboratories Usa
Curated by ChEMBL
Tanabe Research Laboratories Usa
Curated by ChEMBL
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa
Curated by ChEMBL
Tanabe Research Laboratories Usa
Curated by ChEMBL
Affinity DataKi: 44nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Tanabe Research Laboratories Usa
Curated by ChEMBL
Tanabe Research Laboratories Usa
Curated by ChEMBL
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Tanabe Research Laboratories Usa
Curated by ChEMBL
Tanabe Research Laboratories Usa
Curated by ChEMBL
TargetAdenosine receptor A2b(Homo sapiens (Human))
East China University Of Science And Technology
Curated by ChEMBL
East China University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 49nMAssay Description:Antagonist activity against human adenosine A2B receptorMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa
Curated by ChEMBL
Tanabe Research Laboratories Usa
Curated by ChEMBL
Affinity DataKi: 52nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa
Curated by ChEMBL
Tanabe Research Laboratories Usa
Curated by ChEMBL
Affinity DataKi: 52nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
East China University Of Science And Technology
Curated by ChEMBL
East China University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 54nMAssay Description:Antagonist activity against human adenosine A3 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
East China University Of Science And Technology
Curated by ChEMBL
East China University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 54.8nMAssay Description:Antagonist activity against human adenosine A1 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
East China University Of Science And Technology
Curated by ChEMBL
East China University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 56nMAssay Description:Antagonist activity against human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Inhibition of human somatostatin receptor type 4More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa
Curated by ChEMBL
Tanabe Research Laboratories Usa
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
East China University Of Science And Technology
Curated by ChEMBL
East China University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 64nMAssay Description:Antagonist activity against rat adenosine A1 receptorMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa
Curated by ChEMBL
Tanabe Research Laboratories Usa
Curated by ChEMBL
Affinity DataKi: 64nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa
Curated by ChEMBL
Tanabe Research Laboratories Usa
Curated by ChEMBL
Affinity DataKi: 68nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
East China University Of Science And Technology
Curated by ChEMBL
East China University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 73nMAssay Description:Antagonist activity against human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 77nMAssay Description:Inhibition of human somatostatin receptor type 4 (n=5)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa
Curated by ChEMBL
Tanabe Research Laboratories Usa
Curated by ChEMBL
Affinity DataKi: 80nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair