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Found 297 with Last Name = 'cheng' and Initial = 'll'
TargetVasopressin V1b receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205313(CHEMBL265859 | d[Leu4]AVP)
Affinity DataKi:  0.0400nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50370109(CHEMBL1790723)
Affinity DataKi:  0.0900nMAssay Description:Binding affinity for human oxytocin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205305(CHEMBL375324 | d[Arg4]AVP)
Affinity DataKi:  0.130nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205309(CHEMBL412972 | d[Leu4,Lys8]VP)
Affinity DataKi:  0.160nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50370113(CHEMBL1790719)
Affinity DataKi:  0.170nMAssay Description:Binding affinity for human oxytocin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50370117(CHEMBL1790720)
Affinity DataKi:  0.180nMAssay Description:Binding affinity for human oxytocin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205296(CHEMBL385739 | d[Arg4,Dab8]VP)
Affinity DataKi:  0.190nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205291((S)-1-((4R,7S,10S,13S,16S)-7-(2-amino-2-oxoethyl)-...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205305(CHEMBL375324 | d[Arg4]AVP)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50370106(CHEMBL1790712)
Affinity DataKi:  0.210nMAssay Description:Binding affinity for human oxytocin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Medical College Of Ohio

Curated by ChEMBL
LigandPNGBDBM50145126((2S)-2-{[(2R)-1-{[(4S,7R,10S,13R,16S)-13-benzyl-7-...)
Affinity DataKi:  0.230nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50370110(CHEMBL1790721)
Affinity DataKi:  0.25nMAssay Description:Binding affinity for human oxytocin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205297(CHEMBL412973 | d[Leu4,Dab8]VP)
Affinity DataKi:  0.25nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205300(CHEMBL221436 | d[Val4]AVP)
Affinity DataKi:  0.25nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205304(CHEMBL435323 | dVDAVP)
Affinity DataKi:  0.260nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205301(CHEMBL375188 | d[Leu4,Orn8]VP)
Affinity DataKi:  0.260nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50370114(CHEMBL1790718)
Affinity DataKi:  0.290nMAssay Description:Binding affinity for human oxytocin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Medical College Of Ohio

Curated by ChEMBL
LigandPNGBDBM50145118(CHEMBL412353 | d[Val4]AVP)
Affinity DataKi:  0.290nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205308((S)-1-((4R,7S,10S,13S,16S)-7-(2-amino-2-oxoethyl)-...)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205300(CHEMBL221436 | d[Val4]AVP)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50370112(CHEMBL1790729)
Affinity DataKi:  0.320nMAssay Description:Binding affinity for human oxytocin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50370115(CHEMBL1790717)
Affinity DataKi:  0.340nMAssay Description:Binding affinity for human oxytocin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Medical College Of Ohio

Curated by ChEMBL
LigandPNGBDBM50145112((2S)-2-{[(2R)-1-{[(4S,7R,13R,16S)-13-benzyl-7-(car...)
Affinity DataKi:  0.370nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205303(CHEMBL373968 | d[Leu4,Dap8]VP)
Affinity DataKi:  0.380nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50370111(CHEMBL1790711)
Affinity DataKi:  0.400nMAssay Description:Binding affinity for human oxytocin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Medical College Of Ohio

Curated by ChEMBL
LigandPNGBDBM50370387(CHEMBL1790575)
Affinity DataKi:  0.420nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Medical College Of Ohio

Curated by ChEMBL
LigandPNGBDBM50145124((2S)-2-{[(2R)-1-{[(4S,7R,13R,16S)-13-benzyl-10-but...)
Affinity DataKi:  0.430nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205306(CHEMBL375323 | d[Orn4,Lys8]VP)
Affinity DataKi:  0.450nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205311(CHEMBL375096 | d[Orn4]AVP)
Affinity DataKi:  0.450nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Medical College Of Ohio

Curated by ChEMBL
LigandPNGBDBM50145107((2S)-2-{[(2R)-1-{[(4S,7R,13R,16S)-10-(3-aminopropy...)
Affinity DataKi:  0.490nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Medical College Of Ohio

Curated by ChEMBL
LigandPNGBDBM50145117((2S)-2-{[(2R)-1-{[(4S,7R,13R,16S)-13-benzyl-7-(car...)
Affinity DataKi:  0.520nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205298(CHEMBL375325 | d[Arg4,Lys8]VP)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205292(CHEMBL385068 | d[Arg4,Orn8]VP)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Medical College Of Ohio

Curated by ChEMBL
LigandPNGBDBM50145108((2S)-2-{[(2R)-1-{[(4S,7R,13R,16S)-13-benzyl-7-(car...)
Affinity DataKi:  0.780nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataKi:  0.800nMAssay Description:Binding affinity for human oxytocin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205291((S)-1-((4R,7S,10S,13S,16S)-7-(2-amino-2-oxoethyl)-...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205307(CHEMBL412742 | d[Cha4,Dab8]VP)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205310(CHEMBL219272 | d[Orn4,Orn8]VP)
Affinity DataKi:  0.910nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205291((S)-1-((4R,7S,10S,13S,16S)-7-(2-amino-2-oxoethyl)-...)
Affinity DataKi:  0.970nMAssay Description:Displacement of [3H]AVP from rat OT receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Medical College Of Ohio

Curated by ChEMBL
LigandPNGBDBM50145111((2S)-2-{[(2R)-1-{[(4S,7R,13R,16S)-13-benzyl-7-(car...)
Affinity DataKi:  1nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM35667(AVP | CHEMBL373742 | US10131692, 44 (AVP) | [3H]Ar...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]AVP from rat OT receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Medical College Of Ohio

Curated by ChEMBL
LigandPNGBDBM50145109((2S)-2-{[(2R)-1-{[(4S,7R,13R,16S)-13-benzyl-7-(car...)
Affinity DataKi:  1.20nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Medical College Of Ohio

Curated by ChEMBL
LigandPNGBDBM50145123(CHEMBL410573 | d[Cha4]AVP)
Affinity DataKi:  1.20nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Medical College Of Ohio

Curated by ChEMBL
LigandPNGBDBM50145118(CHEMBL412353 | d[Val4]AVP)
Affinity DataKi:  1.20nMAssay Description:Binding affinity against human vasopressin V2 receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT receptor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205312(CHEMBL265858 | d[Cha4]AVP)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Medical College Of Ohio

Curated by ChEMBL
LigandPNGBDBM50145129((2S)-2-{[(2R)-1-{[(4S,7R,13R,16S)-13-benzyl-7,10-b...)
Affinity DataKi:  1.5nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Medical College Of Ohio

Curated by ChEMBL
LigandPNGBDBM50145111((2S)-2-{[(2R)-1-{[(4S,7R,13R,16S)-13-benzyl-7-(car...)
Affinity DataKi:  1.5nMAssay Description:Binding affinity against human vasopressin V2 receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT receptor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Medical College Of Ohio

Curated by ChEMBL
LigandPNGBDBM50145129((2S)-2-{[(2R)-1-{[(4S,7R,13R,16S)-13-benzyl-7,10-b...)
Affinity DataKi:  1.5nMAssay Description:Binding affinity against human vasopressin V1a receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50370107(CHEMBL1790728)
Affinity DataKi:  1.80nMAssay Description:Binding affinity for human oxytocin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205296(CHEMBL385739 | d[Arg4,Dab8]VP)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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