Affinity DataEC50: 3.00E+6nMAssay Description:Agonist activity at GluR4 expressed in HEK293 cells by Fluo-4/Ca2+ assayMore data for this Ligand-Target Pair
Affinity DataEC50: 7.00E+5nMAssay Description:Agonist activity at GluR3 expressed in HEK293 cells by Fluo-4/Ca2+ assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.50E+5nMAssay Description:Agonist activity at GluR3 expressed in HEK293 cells by Fluo-4/Ca2+ assayMore data for this Ligand-Target Pair
Affinity DataEC50: >3.00E+6nMAssay Description:Agonist activity at GluR2Q expressed in HEK293 cells by Fluo-4/Ca2+ assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.80E+5nMAssay Description:Agonist activity at GluR1 expressed in HEK293 cells by Fluo-4/Ca2+ assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.80E+4nMAssay Description:Agonist activity at GluR4 expressed in HEK293 cells by Fluo-4/Ca2+ assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.20E+4nMAssay Description:Agonist activity at GluR1 expressed in HEK293 cells by Fluo-4/Ca2+ assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+6nMAssay Description:Agonist activity at GluR3 expressed in HEK293 cells by Fluo-4/Ca2+ assayMore data for this Ligand-Target Pair
Affinity DataEC50: 8.30E+5nMAssay Description:Agonist activity at GluR2Q expressed in HEK293 cells by Fluo-4/Ca2+ assayMore data for this Ligand-Target Pair
Affinity DataEC50: 7.10E+4nMAssay Description:Agonist activity at GluR1 expressed in HEK293 cells by Fluo-4/Ca2+ assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+6nMAssay Description:Agonist activity at GluR2Q expressed in HEK293 cells by Fluo-4/Ca2+ assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.80E+4nMAssay Description:Agonist activity at GluR3 expressed in HEK293 cells by Fluo-4/Ca2+ assayMore data for this Ligand-Target Pair
Affinity DataEC50: >3.00E+6nMAssay Description:Agonist activity at GluR2Q expressed in HEK293 cells by Fluo-4/Ca2+ assayMore data for this Ligand-Target Pair
Affinity DataEC50: >3.00E+6nMAssay Description:Agonist activity at GluR1 expressed in HEK293 cells by Fluo-4/Ca2+ assayMore data for this Ligand-Target Pair
Affinity DataEC50: 6.70E+4nMAssay Description:Agonist activity at GluR3 expressed in HEK293 cells by Fluo-4/Ca2+ assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.90E+5nMAssay Description:Agonist activity at GluR4 expressed in Xenopus oocyte cells S-GlutamateMore data for this Ligand-Target Pair
Affinity DataEC50: 4.00E+3nMAssay Description:Agonist activity at GluR4 expressed in HEK293 cells by Fluo-4/Ca2+ assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5.20E+4nMAssay Description:Agonist activity at GluR2Q expressed in HEK293 cells by Fluo-4/Ca2+ assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.00E+6nMAssay Description:Agonist activity at GluR1 expressed in HEK293 cells by Fluo-4/Ca2+ assayMore data for this Ligand-Target Pair
Affinity DataEC50: 7.50E+4nMAssay Description:Agonist activity at GluR4 expressed in HEK293 cells by Fluo-4/Ca2+ assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.40E+5nMAssay Description:Agonist activity at GluR2Q expressed in HEK293 cells by Fluo-4/Ca2+ assayMore data for this Ligand-Target Pair
Affinity DataEC50: >3.00E+6nMAssay Description:Agonist activity at GluR3 expressed in HEK293 cells by Fluo-4/Ca2+ assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5.50E+5nMAssay Description:Agonist activity at GluR1 expressed in HEK293 cells by Fluo-4/Ca2+ assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.60E+5nMAssay Description:Agonist activity at GluR4 expressed in HEK293 cells by Fluo-4/Ca2+ assayMore data for this Ligand-Target Pair
Affinity DataEC50: 7.90E+4nMAssay Description:Agonist activity at GluR4 expressed in HEK293 cells by Fluo-4/Ca2+ assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+6nMAssay Description:Activity at rat cloned mGluR1a expressed in CHO cells assessed as effect on cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 6.10E+5nMAssay Description:Activity at rat cloned mGluR1a expressed in CHO cells assessed as effect on cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+6nMAssay Description:Activity at rat cloned mGluR2 expressed in CHO cells assessed as effect on cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+6nMAssay Description:Activity at rat cloned mGluR2 expressed in CHO cells assessed as effect on cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 4.30E+4nMAssay Description:Activity at rat cloned mGluR1a expressed in CHO cells assessed as effect on cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 8.20E+4nMAssay Description:Activity at rat cloned mGluR1a expressed in CHO cells assessed as effect on cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+6nMAssay Description:Activity at rat cloned mGluR1a expressed in CHO cells assessed as effect on cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 8.40E+4nMAssay Description:Activity at rat cloned mGluR2 expressed in CHO cells assessed as effect on cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 1.10E+5nMAssay Description:Activity at rat cloned mGluR2 expressed in CHO cells assessed as effect on cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+6nMAssay Description:Activity at rat cloned mGluR4 expressed in CHO cells assessed as effect on cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+6nMAssay Description:Activity at rat cloned mGluR4 expressed in CHO cells assessed as effect on cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+6nMAssay Description:Activity at rat cloned mGluR4 expressed in CHO cells assessed as effect on cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+6nMAssay Description:Activity at rat cloned mGluR4 expressed in CHO cells assessed as effect on cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 7.90E+5nMAssay Description:Activity at rat cloned mGluR1a expressed in CHO cells assessed as effect on cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+6nMAssay Description:Activity at rat cloned mGluR2 expressed in CHO cells assessed as effect on cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+6nMAssay Description:Activity at rat cloned mGluR4 expressed in CHO cells assessed as effect on cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 1.10E+5nMAssay Description:Activity at rat cloned mGluR1a expressed in CHO cells assessed as effect on cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+5nMAssay Description:Activity at rat cloned mGluR2 expressed in CHO cells assessed as effect on cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+6nMAssay Description:Activity at rat cloned mGluR4 expressed in CHO cells assessed as effect on cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+6nMAssay Description:Activity at rat cloned iGluR1 expressed in human HEK293 cells by calcium imaging assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.50E+4nMAssay Description:Activity at rat cloned iGluR1 expressed in human HEK293 cells by calcium imaging assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+6nMAssay Description:Activity at rat cloned iGluR1 expressed in human HEK293 cells by calcium imaging assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.20E+5nMAssay Description:Activity at rat cloned iGluR1 expressed in human HEK293 cells by calcium imaging assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+6nMAssay Description:Activity at rat cloned iGluR2 expressed in human HEK293 cells by calcium imaging assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+6nMAssay Description:Activity at rat cloned iGluR2 expressed in human HEK293 cells by calcium imaging assayMore data for this Ligand-Target Pair