Affinity DataIC50: 30nMAssay Description:Inhibition of Enterobacter cloacae IMI1 beta lactamase expressed in Escherichia coli DH5alpha by SDS-PAGEMore data for this Ligand-Target Pair
TargetCarbapenem-hydrolyzing beta-lactamase KPC(Klebsiella pneumoniae)
University Of Aveiro
Curated by ChEMBL
University Of Aveiro
Curated by ChEMBL
Affinity DataIC50: 374nMAssay Description:Inhibition of Klebsiella pneumoniae KPC-1 beta lactamase expressed in Escherichia coli DH5alpha by SDS-PAGEMore data for this Ligand-Target Pair
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of Serratia fonticola UTAD54 SFC1 beta lactamase expressed in Escherichia coli BL21(DE3) by SDS-PAGEMore data for this Ligand-Target Pair
Affinity DataIC50: 2.27E+4nMAssay Description:Inhibition of Serratia fonticola UTAD54 SFC1 beta lactamase expressed in Escherichia coli BL21(DE3) by SDS-PAGEMore data for this Ligand-Target Pair
Affinity DataIC50: 7.28E+4nMAssay Description:Inhibition of Serratia fonticola UTAD54 SFC1 beta lactamase expressed in Escherichia coli BL21(DE3) by SDS-PAGEMore data for this Ligand-Target Pair
Affinity DataEC50: 5.10nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO cells assessed as inhibition forskolin-induced cAMP releaseMore data for this Ligand-Target Pair
Affinity DataEC50: 1.02E+3nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO cells assessed as inhibition forskolin-induced cAMP releaseMore data for this Ligand-Target Pair
Affinity DataEC50: 637nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO cells assessed as inhibition forskolin-induced cAMP releaseMore data for this Ligand-Target Pair
Affinity DataEC50: 523nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO cells assessed as inhibition forskolin-induced cAMP releaseMore data for this Ligand-Target Pair
Affinity DataEC50: 320nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO cells assessed as inhibition forskolin-induced cAMP releaseMore data for this Ligand-Target Pair
Affinity DataEC50: 1.40E+4nMAssay Description:Agonist activity at human recombinant CB1 receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 24.5nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO cells assessed as inhibition forskolin-induced cAMP releaseMore data for this Ligand-Target Pair
Affinity DataEC50: 14.2nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO cells assessed as inhibition forskolin-induced cAMP releaseMore data for this Ligand-Target Pair
Affinity DataEC50: 9.10nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO cells assessed as inhibition forskolin-induced cAMP releaseMore data for this Ligand-Target Pair
Affinity DataEC50: 7.90nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO cells assessed as inhibition forskolin-induced cAMP releaseMore data for this Ligand-Target Pair
Affinity DataEC50: 18.5nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO cells assessed as inhibition forskolin-induced cAMP releaseMore data for this Ligand-Target Pair
Affinity DataEC50: 55.4nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO cells assessed as inhibition forskolin-induced cAMP releaseMore data for this Ligand-Target Pair
Affinity DataEC50: 7nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO cells assessed as inhibition forskolin-induced cAMP releaseMore data for this Ligand-Target Pair
Affinity DataEC50: 380nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO cells assessed as inhibition forskolin-induced cAMP releaseMore data for this Ligand-Target Pair
Affinity DataEC50: 878nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO cells assessed as inhibition forskolin-induced cAMP releaseMore data for this Ligand-Target Pair
Affinity DataEC50: 3.00E+3nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO cells assessed as inhibition forskolin-induced cAMP releaseMore data for this Ligand-Target Pair
Affinity DataEC50: 560nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO cells assessed as inhibition forskolin-induced cAMP releaseMore data for this Ligand-Target Pair
Affinity DataEC50: 295nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO cells assessed as inhibition forskolin-induced cAMP releaseMore data for this Ligand-Target Pair
Affinity DataEC50: 7.50E+3nMAssay Description:Agonist activity at human recombinant CB1 receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.80E+4nMAssay Description:Agonist activity at human recombinant CB1 receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 13.4nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO cells assessed as inhibition forskolin-induced cAMP releaseMore data for this Ligand-Target Pair
Affinity DataEC50: 26.7nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO cells assessed as inhibition forskolin-induced cAMP releaseMore data for this Ligand-Target Pair
Affinity DataEC50: 21.5nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO cells assessed as inhibition forskolin-induced cAMP releaseMore data for this Ligand-Target Pair
Affinity DataEC50: 403nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO cells assessed as inhibition forskolin-induced cAMP releaseMore data for this Ligand-Target Pair
Affinity DataEC50: 439nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO cells assessed as inhibition forskolin-induced cAMP releaseMore data for this Ligand-Target Pair
Affinity DataEC50: 21.8nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO cells assessed as inhibition forskolin-induced cAMP releaseMore data for this Ligand-Target Pair