BindingDB PrimarySearch_ki

Found 593 with Last Name = 'dzwonek' and Initial = 'k'

Acidic mammalian chitinase(Homo sapiens (Human))
Oncoarendi Therapeutics

Curated by ChEMBL

PNG

BDBM50554340(CHEMBL4788866)

Ki: 4.80nMAssay Description:Inhibition of full-length C-terminal his-tagged human AMCase expressed in CHO-K1 cells assessed as reduction in chitinolytic activity using 4-methylu...More data for this Ligand-Target Pair

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Acidic mammalian chitinase(Mus musculus)
Oncoarendi Therapeutics

Curated by ChEMBL

PNG

BDBM50554340(CHEMBL4788866)

Ki: 5.70nMAssay Description:Inhibition of full-length C-terminal his-tagged mouse AMCase expressed in expressed in CHO-K1 cells assessed as reduction in chitinolytic activity us...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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Acidic mammalian chitinase(Mus musculus)
Oncoarendi Therapeutics

Curated by ChEMBL

PNG

BDBM50243745(CHEMBL4076989)

Ki: 11nMAssay Description:Inhibition of mouse recombinant full length C-terminal His-tagged acidic mammalian chitinase expressed in CHO-K1 cells using 4-methylumbelliferyl-bet...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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Acidic mammalian chitinase(Homo sapiens (Human))
Oncoarendi Therapeutics

Curated by ChEMBL

PNG

BDBM50243745(CHEMBL4076989)

Ki: 14nMAssay Description:Inhibition of human recombinant full length C-terminal His-tagged acidic mammalian chitinase expressed in CHO-K1 cells using 4-methylumbelliferyl-bet...More data for this Ligand-Target Pair

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Chitotriosidase-1(Homo sapiens (Human))
Oncoarendi Therapeutics

Curated by ChEMBL

PNG

BDBM50554340(CHEMBL4788866)

Ki: 17nMAssay Description:Inhibition of full-length C-terminal his-tagged human recombinant CHIT1 catalytic domain (1 to 386 residues) expressed in HEK293F cells assessed as r...More data for this Ligand-Target Pair

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3D Structure (crystal)

Chitotriosidase-1(Mus musculus)
Oncoarendi Therapeutics

Curated by ChEMBL

PNG

BDBM50554340(CHEMBL4788866)

Ki: 26nMAssay Description:Inhibition of recombinant full-length C-terminal his-tagged mouse CHIT1 expressed in CHO-K1 cells assessed as reduction in chitinolytic activity usin...More data for this Ligand-Target Pair

Reactome pathway
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Chitotriosidase-1(Homo sapiens (Human))
Oncoarendi Therapeutics

Curated by ChEMBL

PNG

BDBM50243745(CHEMBL4076989)

Ki: 312nMAssay Description:Inhibition of human recombinant full length C-terminal His-tagged chitotriosidase expressed in CHO-K1 cells using 4-methylumbelliferyl-beta-D-N,N',N\...More data for this Ligand-Target Pair

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Chitotriosidase-1(Mus musculus)
Oncoarendi Therapeutics

Curated by ChEMBL

PNG

BDBM50243745(CHEMBL4076989)

Ki: 3.40E+3nMAssay Description:Inhibition of mouse recombinant full length C-terminal His-tagged chitotriosidase expressed in CHO-K1 cells using 4-methylumbelliferyl-beta-D-N,N',N\...More data for this Ligand-Target Pair

Reactome pathway
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Fibroblast growth factor receptor 2(Homo sapiens (Human))
Celon Pharma

Curated by ChEMBL

PNG

BDBM50587623(CHEMBL5173892)

IC50: 0.110nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human FGFR2 (399 to 821 residues) expressed in baculovirus expression system using IGF-1Rtide peptide...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Fibroblast growth factor receptor 1(Homo sapiens (Human))
Celon Pharma

Curated by ChEMBL

PNG

BDBM50065454(CHEBI:63453 | CHEMBL3348846)

IC50: 0.200nMAssay Description:Inhibition of recombinant human FGFR1 in the presence of ATP at Km concentrationMore data for this Ligand-Target Pair

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Fibroblast growth factor receptor 2(Homo sapiens (Human))
Celon Pharma

Curated by ChEMBL

PNG

BDBM50587622(CHEMBL5171314)

IC50: 0.270nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human FGFR2 (399 to 821 residues) expressed in baculovirus expression system using IGF-1Rtide peptide...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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Fibroblast growth factor receptor 2(Homo sapiens (Human))
Celon Pharma

Curated by ChEMBL

PNG

BDBM50587621(CHEMBL5179660)

IC50: 0.290nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human FGFR2 (399 to 821 residues) expressed in baculovirus expression system using IGF-1Rtide peptide...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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Fibroblast growth factor receptor 1(Homo sapiens (Human))
Celon Pharma

Curated by ChEMBL

PNG

BDBM301310(3-(2,6-difluoro-3,5-dimethoxyphenyl)-1-ethyl-8-(mo...)

IC50: 0.400nMAssay Description:Inhibition of FGFR1 (unknown origin)More data for this Ligand-Target Pair

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3D Structure (crystal)

Fibroblast growth factor receptor 1(Homo sapiens (Human))
Celon Pharma

Curated by ChEMBL

PNG

BDBM50587619(CHEMBL5205436)

IC50: 0.430nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human FGFR1 (398 to 822 residues) expressed in baculovirus expression system using IGF-1Rtide peptide...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Fibroblast growth factor receptor 2(Homo sapiens (Human))
Celon Pharma

Curated by ChEMBL

PNG

BDBM50587619(CHEMBL5205436)

IC50: 0.430nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human FGFR2 (399 to 821 residues) expressed in baculovirus expression system using IGF-1Rtide peptide...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Fibroblast growth factor receptor 2(Homo sapiens (Human))
Celon Pharma

Curated by ChEMBL

PNG

BDBM50587620(CHEMBL5189958)

IC50: 0.437nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human FGFR2 (399 to 821 residues) expressed in baculovirus expression system using IGF-1Rtide peptide...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Fibroblast growth factor receptor 2(Homo sapiens (Human))
Celon Pharma

Curated by ChEMBL

PNG

BDBM50587625(CHEMBL5199374)

IC50: 0.5nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human FGFR2 (399 to 821 residues) expressed in baculovirus expression system using IGF-1Rtide peptide...More data for this Ligand-Target Pair

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Fibroblast growth factor receptor 2(Homo sapiens (Human))
Celon Pharma

Curated by ChEMBL

PNG

BDBM301310(3-(2,6-difluoro-3,5-dimethoxyphenyl)-1-ethyl-8-(mo...)

IC50: 0.5nMAssay Description:Inhibition of FGFR2 (unknown origin)More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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3D Structure (crystal)

Fibroblast growth factor receptor 2(Homo sapiens (Human))
Celon Pharma

Curated by ChEMBL

PNG

BDBM50587646(CHEMBL5177815)

IC50: 0.630nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human FGFR2 (399 to 821 residues) expressed in baculovirus expression system using IGF-1Rtide peptide...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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Acidic mammalian chitinase(Homo sapiens (Human))
Oncoarendi Therapeutics

Curated by ChEMBL

PNG

BDBM50541950(CHEMBL4643001)

IC50: 0.700nMAssay Description:Inhibition of full length recombinant C-terminal His-tagged human acidic mammalian chitinase expressed in CHOK1 cells assessed as reduction in chitin...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Fibroblast growth factor receptor 1(Homo sapiens (Human))
Celon Pharma

Curated by ChEMBL

PNG

BDBM50587625(CHEMBL5199374)

IC50: 0.75nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human FGFR1 (398 to 822 residues) expressed in baculovirus expression system using IGF-1Rtide peptide...More data for this Ligand-Target Pair

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Fibroblast growth factor receptor 1(Homo sapiens (Human))
Celon Pharma

Curated by ChEMBL

PNG

BDBM50587646(CHEMBL5177815)

IC50: 0.790nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human FGFR1 (398 to 822 residues) expressed in baculovirus expression system using IGF-1Rtide peptide...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Fibroblast growth factor receptor 2(Homo sapiens (Human))
Celon Pharma

Curated by ChEMBL

PNG

BDBM50587631(CHEMBL5191338)

IC50: 0.810nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human FGFR2 (399 to 821 residues) expressed in baculovirus expression system using IGF-1Rtide peptide...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Fibroblast growth factor receptor 2(Homo sapiens (Human))
Celon Pharma

Curated by ChEMBL

PNG

BDBM50587630(CHEMBL5174735)

IC50: 0.840nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human FGFR2 (399 to 821 residues) expressed in baculovirus expression system using IGF-1Rtide peptide...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Fibroblast growth factor receptor 2(Homo sapiens (Human))
Celon Pharma

Curated by ChEMBL

PNG

BDBM50587628(CHEMBL5186357)

IC50: 0.890nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human FGFR2 (399 to 821 residues) expressed in baculovirus expression system using IGF-1Rtide peptide...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Fibroblast growth factor receptor 2(Homo sapiens (Human))
Celon Pharma

Curated by ChEMBL

PNG

BDBM50587626(CHEMBL5207255)

IC50: 0.915nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human FGFR2 (399 to 821 residues) expressed in baculovirus expression system using IGF-1Rtide peptide...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Fibroblast growth factor receptor 2(Homo sapiens (Human))
Celon Pharma

Curated by ChEMBL

PNG

BDBM342461(US9776988, Example 21)

IC50: 0.950nMAssay Description:The compounds were dissolved in 100% DMSO, and obtained solutions were serially diluted in reaction buffer (50 mM Tris pH 7.5, 10 mM MgCl2, 0.25 mM E...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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Fibroblast growth factor receptor 3(Homo sapiens (Human))
Celon Pharma

Curated by ChEMBL

PNG

BDBM301310(3-(2,6-difluoro-3,5-dimethoxyphenyl)-1-ethyl-8-(mo...)

IC50: 1nMAssay Description:Inhibition of FGFR3 (unknown origin)More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Fibroblast growth factor receptor 2(Homo sapiens (Human))
Celon Pharma

Curated by ChEMBL

PNG

BDBM50587647(CHEMBL5186648)

IC50: 1nMAssay Description:Inhibition of FGFR2 (unknown origin)More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Acidic mammalian chitinase(Mus musculus)
Oncoarendi Therapeutics

Curated by ChEMBL

PNG

BDBM50554344(CHEMBL4756869)

IC50: 1nMAssay Description:Inhibition of full-length C-terminal his-tagged mouse AMCase expressed in expressed in CHO-K1 cells assessed as reduction in chitinolytic activity us...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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Fibroblast growth factor receptor 2(Homo sapiens (Human))
Celon Pharma

Curated by ChEMBL

PNG

BDBM342487(US9776988, Example 3)

IC50: 1.07nMAssay Description:The compounds were dissolved in 100% DMSO, and obtained solutions were serially diluted in reaction buffer (50 mM Tris pH 7.5, 10 mM MgCl2, 0.25 mM E...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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Fibroblast growth factor receptor 2(Homo sapiens (Human))
Celon Pharma

Curated by ChEMBL

PNG

BDBM342487(US9776988, Example 3)

IC50: 1.10nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human FGFR2 (399 to 821 residues) expressed in baculovirus expression system using IGF-1Rtide peptide...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Fibroblast growth factor receptor 1(Homo sapiens (Human))
Celon Pharma

Curated by ChEMBL

PNG

BDBM50525939(Balversa | Erdafitinib | Jnj-42756493)

IC50: 1.20nMAssay Description:Inhibition of FGFR1 (unknown origin)More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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3D Structure (crystal)

Fibroblast growth factor receptor 3(Homo sapiens (Human))
Celon Pharma

Curated by ChEMBL

PNG

BDBM50587619(CHEMBL5205436)

IC50: 1.20nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged FGFR3 (436 to 806 residues) expressed in baculovirus expression system using IGF-1Rtide peptide...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Fibroblast growth factor receptor 2(Homo sapiens (Human))
Celon Pharma

Curated by ChEMBL

PNG

BDBM342463(US9776988, Example 27)

IC50: 1.26nMAssay Description:The compounds were dissolved in 100% DMSO, and obtained solutions were serially diluted in reaction buffer (50 mM Tris pH 7.5, 10 mM MgCl2, 0.25 mM E...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Details US Patent

Acidic mammalian chitinase(Mus musculus)
Oncoarendi Therapeutics

Curated by ChEMBL

PNG

BDBM50554342(CHEMBL4776610)

IC50: 1.30nMAssay Description:Inhibition of full-length C-terminal his-tagged mouse AMCase expressed in expressed in CHO-K1 cells assessed as reduction in chitinolytic activity us...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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GoogleScholar

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Fibroblast growth factor receptor 2(Homo sapiens (Human))
Celon Pharma

Curated by ChEMBL

PNG

BDBM50587637(CHEMBL5192921)

IC50: 1.40nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human FGFR2 (399 to 821 residues) expressed in baculovirus expression system using IGF-1Rtide peptide...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Acidic mammalian chitinase(Homo sapiens (Human))
Oncoarendi Therapeutics

Curated by ChEMBL

PNG

BDBM50541949(CHEMBL4635305)

IC50: 1.40nMAssay Description:Inhibition of full length recombinant C-terminal His-tagged human acidic mammalian chitinase expressed in CHOK1 cells assessed as reduction in chitin...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Details Article PubMed

Fibroblast growth factor receptor 2(Homo sapiens (Human))
Celon Pharma

Curated by ChEMBL

PNG

BDBM50587627(CHEMBL5201819)

IC50: 1.5nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human FGFR2 (399 to 821 residues) expressed in baculovirus expression system using IGF-1Rtide peptide...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Acidic mammalian chitinase(Homo sapiens (Human))
Oncoarendi Therapeutics

Curated by ChEMBL

PNG

BDBM50554344(CHEMBL4756869)

IC50: 1.60nMAssay Description:Inhibition of full-length C-terminal his-tagged human AMCase expressed in CHO-K1 cells assessed as reduction in chitinolytic activity using 4-methylu...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Details Article PubMed

Fibroblast growth factor receptor 2(Homo sapiens (Human))
Celon Pharma

Curated by ChEMBL

PNG

BDBM342456(US9776988, Example 14)

IC50: 1.63nMAssay Description:The compounds were dissolved in 100% DMSO, and obtained solutions were serially diluted in reaction buffer (50 mM Tris pH 7.5, 10 mM MgCl2, 0.25 mM E...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details US Patent

Fibroblast growth factor receptor 3(Homo sapiens (Human))
Celon Pharma

Curated by ChEMBL

PNG

BDBM50065454(CHEBI:63453 | CHEMBL3348846)

IC50: 1.80nMAssay Description:Inhibition of recombinant human FGFR3 in the presence of ATP at Km concentrationMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Fibroblast growth factor receptor 2(Homo sapiens (Human))
Celon Pharma

Curated by ChEMBL

PNG

BDBM50587632(CHEMBL5191301)

IC50: 1.90nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human FGFR2 (399 to 821 residues) expressed in baculovirus expression system using IGF-1Rtide peptide...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Acidic mammalian chitinase(Homo sapiens (Human))
Oncoarendi Therapeutics

Curated by ChEMBL

PNG

BDBM50541930(CHEMBL4637417)

IC50: 2nMAssay Description:Inhibition of full length recombinant C-terminal His-tagged human acidic mammalian chitinase expressed in CHOK1 cells assessed as reduction in chitin...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Details Article PubMed

Acidic mammalian chitinase(Homo sapiens (Human))
Oncoarendi Therapeutics

Curated by ChEMBL

PNG

BDBM50541931(CHEMBL4634943)

IC50: 2nMAssay Description:Inhibition of full length recombinant C-terminal His-tagged human acidic mammalian chitinase expressed in CHOK1 cells assessed as reduction in chitin...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Details Article PubMed

Fibroblast growth factor receptor 2(Homo sapiens (Human))
Celon Pharma

Curated by ChEMBL

PNG

BDBM339992(US9776988, Example 18)

IC50: 2.05nMAssay Description:The compounds were dissolved in 100% DMSO, and obtained solutions were serially diluted in reaction buffer (50 mM Tris pH 7.5, 10 mM MgCl2, 0.25 mM E...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details US Patent

Acidic mammalian chitinase(Mus musculus)
Oncoarendi Therapeutics

Curated by ChEMBL

PNG

BDBM50554343(CHEMBL4794014)

IC50: 2.10nMAssay Description:Inhibition of full-length C-terminal his-tagged mouse AMCase expressed in expressed in CHO-K1 cells assessed as reduction in chitinolytic activity us...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Fibroblast growth factor receptor 2(Homo sapiens (Human))
Celon Pharma

Curated by ChEMBL

PNG

BDBM50587633(CHEMBL5183603)

IC50: 2.10nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human FGFR2 (399 to 821 residues) expressed in baculovirus expression system using IGF-1Rtide peptide...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Fibroblast growth factor receptor 2(Homo sapiens (Human))
Celon Pharma

Curated by ChEMBL

PNG

BDBM340025(US9776988, Example 8)

IC50: 2.13nMAssay Description:The compounds were dissolved in 100% DMSO, and obtained solutions were serially diluted in reaction buffer (50 mM Tris pH 7.5, 10 mM MgCl2, 0.25 mM E...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details US Patent

Fibroblast growth factor receptor 2(Homo sapiens (Human))
Celon Pharma

Curated by ChEMBL

PNG

BDBM342472(US9776988, Example 4)

IC50: 2.18nMAssay Description:The compounds were dissolved in 100% DMSO, and obtained solutions were serially diluted in reaction buffer (50 mM Tris pH 7.5, 10 mM MgCl2, 0.25 mM E...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details US Patent

Displayed 1 to 50 (of 593 total ) | Next | Last >>

Filter my 593 hits

Targets 14▿
- Acidic mammalian chitinase 173
- Chitotriosidase-1 172
- Potassium voltage-gated channel subfamily H member 2 61
- Fibroblast growth factor receptor 1 46
- Fibroblast growth factor receptor 3 41
- Fibroblast growth factor receptor 2 40
- Vascular endothelial growth factor receptor 2 33
- Arginase-1 16
- Fibroblast growth factor receptor 4 5
- Sodium-dependent dopamine transporter 2
- Receptor-type tyrosine-protein kinase FLT3 1
- Tyrosine-protein kinase JAK2 1
- Platelet-derived growth factor receptor beta 1
- Aurora kinase A 1
- ...
Publications 7▿
- Eur J Med Chem 210: (2021) 137
- J Med Chem 62: 7126-7145 (2019) 136
- J Med Chem 61: 695-710 (2018) 113
- J Med Chem 63: 15527-15540 (2020) 87
- ACS Med Chem Lett 11: 1228-1235 (2020) 72
- US Patent US9776988 (2017) 32
- ACS Med Chem Lett 11: 433-438 (2020) 16
Institutions 2▿
- Oncoarendi Therapeutics 424
- Celon Pharma 169
Affinity: 0.11 to 1.0E+5 nM▿
- Ki 8
- IC50 585
- Affinity ≤ nM
Xtal structures: 9
Docked structures: 0
Catalog Cmpds: 11