Affinity DataIC50: 17nMAssay Description:Compound was tested for the inhibition of [3H]-ketanserin binding to 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Compound was tested for the inhibition of [3H]-ketanserin binding to 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 25.4nMAssay Description:Compound was tested for it's binding affinity towards 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 2(Homo sapiens (Human))
Prassis Istituto Di Ricerche Sigma-Tau
Curated by ChEMBL
Prassis Istituto Di Ricerche Sigma-Tau
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Compound was evaluated for its ability to inhibit the specific [3H]-ouabain binding to dog kidney Na+/K+ ATPaseMore data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:Compound was tested for the inhibition of [3H]-ketanserin binding to 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 2(Homo sapiens (Human))
Prassis Istituto Di Ricerche Sigma-Tau
Curated by ChEMBL
Prassis Istituto Di Ricerche Sigma-Tau
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Compound was evaluated for its ability to inhibit the specific [3H]-ouabain binding to dog kidney Na+/K+ ATPaseMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 2(Homo sapiens (Human))
Prassis Istituto Di Ricerche Sigma-Tau
Curated by ChEMBL
Prassis Istituto Di Ricerche Sigma-Tau
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Compound was evaluated for its ability to inhibit the specific [3H]-ouabain binding to dog kidney Na+/K+ ATPaseMore data for this Ligand-Target Pair
Affinity DataIC50: 94nMAssay Description:Compound was tested for the inhibition of [3H]-ketanserin binding to 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 2(Homo sapiens (Human))
Prassis Istituto Di Ricerche Sigma-Tau
Curated by ChEMBL
Prassis Istituto Di Ricerche Sigma-Tau
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Compound was evaluated for its ability to inhibit the specific [3H]-ouabain binding to dog kidney Na+/K+ ATPaseMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 2(Homo sapiens (Human))
Prassis Istituto Di Ricerche Sigma-Tau
Curated by ChEMBL
Prassis Istituto Di Ricerche Sigma-Tau
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Compound was evaluated for its ability to inhibit the specific [3H]-ouabain binding to dog kidney Na+/K+ ATPaseMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 2(Homo sapiens (Human))
Prassis Istituto Di Ricerche Sigma-Tau
Curated by ChEMBL
Prassis Istituto Di Ricerche Sigma-Tau
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Compound was evaluated for its ability to inhibit the specific [3H]-ouabain binding to dog kidney Na+/K+ ATPaseMore data for this Ligand-Target Pair
Affinity DataIC50: 169nMAssay Description:Compound was tested for the inhibition of [3H]-ketanserin binding to 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 2(Homo sapiens (Human))
Prassis Istituto Di Ricerche Sigma-Tau
Curated by ChEMBL
Prassis Istituto Di Ricerche Sigma-Tau
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Compound was evaluated for its ability to inhibit the specific [3H]-ouabain binding to dog kidney Na+/K+ ATPaseMore data for this Ligand-Target Pair
Affinity DataIC50: 234nMAssay Description:Compound was tested for it's binding affinity towards 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 2(Homo sapiens (Human))
Prassis Istituto Di Ricerche Sigma-Tau
Curated by ChEMBL
Prassis Istituto Di Ricerche Sigma-Tau
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Compound was evaluated for its ability to inhibit the specific [3H]-ouabain binding to dog kidney Na+/K+ ATPaseMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 2(Homo sapiens (Human))
Prassis Istituto Di Ricerche Sigma-Tau
Curated by ChEMBL
Prassis Istituto Di Ricerche Sigma-Tau
Curated by ChEMBL
Affinity DataIC50: 350nMAssay Description:Compound was evaluated for its ability to inhibit the specific [3H]-ouabain binding to dog kidney Na+/K+ ATPaseMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligandMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligandMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligandMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibitory activity against rat heart mitochondrial carnitine palmitoyltransferase 1b using [14C]-palmitoyl-CoA as radioligandMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligandMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibitory activity against rat heart mitochondrial carnitine palmitoyltransferase 1b using [14C]-palmitoyl-CoA as radioligandMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibitory activity against rat heart mitochondrial carnitine palmitoyltransferase 1b using [14C]-palmitoyl-CoA as radioligandMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibitory activity against rat heart mitochondrial carnitine palmitoyltransferase 1b using [14C]-palmitoyl-CoA as radioligandMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 2(Homo sapiens (Human))
Prassis Istituto Di Ricerche Sigma-Tau
Curated by ChEMBL
Prassis Istituto Di Ricerche Sigma-Tau
Curated by ChEMBL
Affinity DataIC50: 5.89E+3nMAssay Description:Compound was evaluated for its ability to inhibit the specific [3H]-ouabain binding to dog kidney Na+/K+ ATPaseMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligandMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligandMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against rat heart mitochondrial carnitine palmitoyltransferase 1b using [14C]-palmitoyl-CoA as radioligandMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against rat heart mitochondrial carnitine palmitoyltransferase 1b using [14C]-palmitoyl-CoA as radioligandMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 1.95E+4nMAssay Description:Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligandMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 2.23E+4nMAssay Description:Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligandMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 4.70E+4nMAssay Description:Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligandMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 8.32E+4nMAssay Description:Inhibitory activity against rat heart mitochondrial carnitine palmitoyltransferase 1b using [14C]-palmitoyl-CoA as radioligandMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 1.22E+5nMAssay Description:Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligandMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 2.11E+5nMAssay Description:Inhibitory activity against rat heart mitochondrial carnitine palmitoyltransferase 1b using [14C]-palmitoyl-CoA as radioligandMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 2.30E+5nMAssay Description:Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligandMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligandMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligandMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligandMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligandMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligandMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligandMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligandMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligandMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligandMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligandMore data for this Ligand-Target Pair