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Found 55 with Last Name = 'marsden' and Initial = 'bd'
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Oxford University

Curated by ChEMBL
LigandPNGBDBM2683(2-[1-(3-dimethylaminopropyl)-indol-3-yl]-3-(indol-...)
Affinity DataIC50:  27nMAssay Description:Inhibitory activity against PIM1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Oxford University

Curated by ChEMBL
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-4H-chrome...)
Affinity DataIC50:  43nMAssay Description:Inhibitory activity against PIM1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Oxford University

Curated by ChEMBL
LigandPNGBDBM11835(1-(3-{6-[(cyclopropylmethyl)amino]imidazo[1,2-a]py...)
Affinity DataIC50:  61nMAssay Description:Inhibitory activity against PIM1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495431(CHEMBL3108800)
Affinity DataIC50:  158nMAssay Description:Displacement of H4Ac4 peptide from CECR2 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495426(CHEMBL3108801)
Affinity DataIC50:  158nMAssay Description:Displacement of H4Ac4 peptide from BRD4 bromodomain-1 (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetBromodomain-containing protein 9(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495426(CHEMBL3108801)
Affinity DataIC50:  200nMAssay Description:Displacement of H2K9(Ac)K13(Ac)K15(Ac) peptide from BRD9 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetCREB-binding protein(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495426(CHEMBL3108801)
Affinity DataIC50:  200nMAssay Description:Displacement of H3K56(Ac) peptide from CREBBP bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495431(CHEMBL3108800)
Affinity DataIC50:  251nMAssay Description:Displacement of H4Ac4 peptide from BRD4 bromodomain-1 (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495429(CHEMBL3108781)
Affinity DataIC50:  251nMAssay Description:Displacement of H4Ac4 peptide from CECR2 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495431(CHEMBL3108800)
Affinity DataIC50:  316nMAssay Description:Displacement of H2K9(Ac)K13(Ac)K15(Ac) peptide from BRD9 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495428(CHEMBL3110357)
Affinity DataIC50:  501nMAssay Description:Displacement of H4Ac4 peptide from CECR2 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495428(CHEMBL3110357)
Affinity DataIC50:  501nMAssay Description:Displacement of H2K9(Ac)K13(Ac)K15(Ac) peptide from BRD9 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495425(CHEMBL3110353)
Affinity DataIC50:  631nMAssay Description:Displacement of H2K9(Ac)K13(Ac)K15(Ac) peptide from BRD9 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495430(CHEMBL3108803)
Affinity DataIC50:  631nMAssay Description:Displacement of H3K56(Ac) peptide from CREBBP bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495431(CHEMBL3108800)
Affinity DataIC50:  631nMAssay Description:Displacement of H3K56(Ac) peptide from CREBBP bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495425(CHEMBL3110353)
Affinity DataIC50:  794nMAssay Description:Displacement of H3K56(Ac) peptide from CREBBP bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495430(CHEMBL3108803)
Affinity DataIC50:  1.00E+3nMAssay Description:Displacement of H4Ac4 peptide from BRD4 bromodomain-1 (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495425(CHEMBL3110353)
Affinity DataIC50:  1.00E+3nMAssay Description:Displacement of H4Ac4 peptide from CECR2 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495430(CHEMBL3108803)
Affinity DataIC50:  1.00E+3nMAssay Description:Displacement of H2K9(Ac)K13(Ac)K15(Ac) peptide from BRD9 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495429(CHEMBL3108781)
Affinity DataIC50:  1.26E+3nMAssay Description:Displacement of H4Ac4 peptide from BRD4 bromodomain-1 (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495429(CHEMBL3108781)
Affinity DataIC50:  1.26E+3nMAssay Description:Displacement of H3K56(Ac) peptide from CREBBP bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495427(CHEMBL1513201)
Affinity DataIC50:  1.26E+3nMAssay Description:Displacement of H2K9(Ac)K13(Ac)K15(Ac) peptide from BRD9 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495427(CHEMBL1513201)
Affinity DataIC50:  1.59E+3nMAssay Description:Displacement of H3K56(Ac) peptide from CREBBP bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495429(CHEMBL3108781)
Affinity DataIC50:  1.59E+3nMAssay Description:Displacement of H2K9(Ac)K13(Ac)K15(Ac) peptide from BRD9 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495427(CHEMBL1513201)
Affinity DataIC50:  2.00E+3nMAssay Description:Displacement of H4Ac4 peptide from BRD4 bromodomain-1 (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495427(CHEMBL1513201)
Affinity DataIC50:  3.16E+3nMAssay Description:Displacement of H4Ac4 peptide from CECR2 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495428(CHEMBL3110357)
Affinity DataIC50:  5.01E+3nMAssay Description:Displacement of H4Ac4 peptide from BRD4 bromodomain-1 (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495432(CHEMBL3108806)
Affinity DataIC50:  5.01E+3nMAssay Description:Displacement of H4Ac4 peptide from CECR2 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495425(CHEMBL3110353)
Affinity DataIC50:  5.01E+3nMAssay Description:Displacement of H4Ac4 peptide from BRD4 bromodomain-1 (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495432(CHEMBL3108806)
Affinity DataIC50:  6.31E+3nMAssay Description:Displacement of H3K56(Ac) peptide from CREBBP bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495428(CHEMBL3110357)
Affinity DataIC50:  1.58E+4nMAssay Description:Displacement of H3K56(Ac) peptide from CREBBP bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495430(CHEMBL3108803)
Affinity DataIC50:  2.00E+4nMAssay Description:Displacement of H4Ac4 peptide from CECR2 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495432(CHEMBL3108806)
Affinity DataIC50:  2.00E+4nMAssay Description:Displacement of H4Ac4 peptide from BRD4 bromodomain-1 (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495426(CHEMBL3108801)
Affinity DataIC50:  2.51E+4nMAssay Description:Displacement of H4Ac4 peptide from CECR2 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495427(CHEMBL1513201)
Affinity DataIC50: <1.00E+5nMAssay Description:Displacement of H3K14(Ac) peptide from BAZ2B bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein polybromo-1(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495429(CHEMBL3108781)
Affinity DataIC50: <1.00E+5nMAssay Description:Displacement of H3K14(Ac) peptide from PB1-5 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495428(CHEMBL3110357)
Affinity DataIC50: <1.00E+5nMAssay Description:Displacement of H3K14(Ac) peptide from TIF1alpha bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495432(CHEMBL3108806)
Affinity DataIC50: <1.00E+5nMAssay Description:Displacement of H3K14(Ac) peptide from TIF1alpha bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495429(CHEMBL3108781)
Affinity DataIC50: <1.00E+5nMAssay Description:Displacement of H3K14(Ac) peptide from BAZ2B bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495432(CHEMBL3108806)
Affinity DataIC50: <1.00E+5nMAssay Description:Displacement of H3K14(Ac) peptide from BAZ2B bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein polybromo-1(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495432(CHEMBL3108806)
Affinity DataIC50: <1.00E+5nMAssay Description:Displacement of H3K14(Ac) peptide from PB1-5 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein polybromo-1(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495427(CHEMBL1513201)
Affinity DataIC50: <1.00E+5nMAssay Description:Displacement of H3K14(Ac) peptide from PB1-5 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein polybromo-1(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495428(CHEMBL3110357)
Affinity DataIC50: <1.00E+5nMAssay Description:Displacement of H3K14(Ac) peptide from PB1-5 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495427(CHEMBL1513201)
Affinity DataIC50: <1.00E+5nMAssay Description:Displacement of H3K14(Ac) peptide from TIF1alpha bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495429(CHEMBL3108781)
Affinity DataIC50: <1.00E+5nMAssay Description:Displacement of H3K14(Ac) peptide from TIF1alpha bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50495428(CHEMBL3110357)
Affinity DataIC50: <1.00E+5nMAssay Description:Displacement of H3K14(Ac) peptide from BAZ2B bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Oxford University

Curated by ChEMBL
LigandPNGBDBM3175(3-[1-[3-(Amidinothio)propyl]-3-indolyl]-4-(1-methy...)
Affinity DataKd:  8nMAssay Description:Binding affinity to non phosphorylated PIM1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Oxford University

Curated by ChEMBL
LigandPNGBDBM2583(3,4-Bis(3-indolyl)-1H-pyrrole-2,5-dione | 3,4-bis(...)
Affinity DataKd:  27nMAssay Description:Binding affinity to non phosphorylated PIM1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Oxford University

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataKd:  1.40nMAssay Description:Binding affinity to non phosphorylated PIM1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Oxford University

Curated by ChEMBL
LigandPNGBDBM11834(3-{2-[(dimethylamino)methyl]-1H,2H,3H,4H-pyrido[1,...)
Affinity DataKd:  250nMAssay Description:Binding affinity to non phosphorylated PIM1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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