Affinity DataKi: 8nMAssay Description:Displacement of [3H]PT-1284 human muscarinic acetylcholine receptor M1 expressed in CHO cell membranes after 90 mins scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Displacement of [3H]PT-1284 human muscarinic acetylcholine receptor M1 expressed in CHO cell membranes after 90 mins scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Displacement of [3H]PT-1284 human muscarinic acetylcholine receptor M1 expressed in CHO cell membranes after 90 mins scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:In vitro inhibitory activity against [3H]- (+)-3-PPP binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against Caspase 1More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals
Curated by ChEMBL
Procter And Gamble Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Displacement of Fluormone from PPAR gammaMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against Caspase 1More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against Caspase 1More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against Caspase 1More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against Caspase 1More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against Caspase 1More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against Caspase 1More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against Caspase 1More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against Caspase 1More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against Caspase 1More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against Caspase 1More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant human MAGL using fluorogenic-7HCA as substrate preincubated for 30 mins followed by substrate addition measured after 60 mi...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against Caspase 1More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibitory activity against Caspase 1More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of caspase-1 using fluorogenic substrate and BMG Fluostar plate reader for 30 min at 37 degree CMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals
Curated by ChEMBL
Procter And Gamble Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Displacement of Fluormone from PPAR gammaMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against Caspase 1More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against Caspase 1More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against Caspase 1More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals
Curated by ChEMBL
Procter And Gamble Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Displacement of Fluormone from PPAR gammaMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of recombinant human MAGL using fluorogenic-7HCA as substrate preincubated for 30 mins followed by substrate addition measured after 60 mi...More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibitory activity against Caspase 8More data for this Ligand-Target Pair
TargetSodium/hydrogen exchanger 1(Homo sapiens (Human))
Pharmaceutical Research Institute
Curated by ChEMBL
Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 4.60nMAssay Description:Inhibition of human NHE1 expressed in Ap1 cell lineMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibitory activity against Caspase 1More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibitory activity against Caspase 1More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibitory activity against Caspase 8More data for this Ligand-Target Pair
TargetSodium/hydrogen exchanger 1(Homo sapiens (Human))
Pharmaceutical Research Institute
Curated by ChEMBL
Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 5.40nMAssay Description:Inhibition of human NHE1 expressed in Ap1 cell lineMore data for this Ligand-Target Pair
Affinity DataIC50: 5.60nMAssay Description:Inhibition of recombinant human MAGL using fluorogenic-7HCA as substrate preincubated for 30 mins followed by substrate addition measured after 60 mi...More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibitory activity against Caspase 1More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibitory activity against Caspase 1More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of recombinant human MAGL using fluorogenic-7HCA as substrate preincubated for 30 mins followed by substrate addition measured after 60 mi...More data for this Ligand-Target Pair
TargetSodium/hydrogen exchanger 1(Homo sapiens (Human))
Pharmaceutical Research Institute
Curated by ChEMBL
Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 6.5nMAssay Description:Inhibition of human NHE1 expressed in Ap1 cell lineMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals
Curated by ChEMBL
Procter And Gamble Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Displacement of Fluormone from PPAR gammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals
Curated by ChEMBL
Procter And Gamble Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Displacement of Fluormone from PPAR gammaMore data for this Ligand-Target Pair