TargetCysteinyl leukotriene receptor 1(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
TargetCysteinyl leukotriene receptor 1(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
TargetCysteinyl leukotriene receptor 1(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
Affinity DataKi: 48nMAssay Description:Binding affinity to human NPSR by radioligand binding assayMore data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
Affinity DataIC50: 537nMAssay Description:Antagonist activity at mouse NPSR expressed in HEK293 cells assessed as inhibition of 10 nM hNPS-induced calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.62E+3nMAssay Description:Antagonist activity at mouse NPSR expressed in HEK293 cells assessed as inhibition of 100 nM hNPS-induced calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 562nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells assessed as increase in intracellular calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 372nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells assessed as increase in intracellular calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 32nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells assessed as increase in intracellular calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 1.55E+3nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells assessed as increase in intracellular calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 166nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells assessed as increase in intracellular calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 85nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells assessed as increase in intracellular calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 22nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells assessed as increase in intracellular calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 129nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells assessed as increase in intracellular calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 204nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells assessed as increase in intracellular calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 240nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells assessed as increase in intracellular calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 1.26E+3nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells assessed as increase in intracellular calcium mobilization by FLIPRMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Institute Of Neuroscienc
Curated by ChEMBL
National Institute Of Neuroscienc
Curated by ChEMBL
Affinity DataEC50: 1.90nMAssay Description:Antagonist activity at human recombinant delta opioid receptor expressed in CHO cells coexpressing alphaqi5 assessed as inhibition of DPDPE-induced i...More data for this Ligand-Target Pair
Affinity DataEC50: 0.389nMAssay Description:Antagonist activity at human recombinant NOP receptor expressed in CHO cells coexpressing alphaqi5 assessed as inhibition of N/OFQ-induced intracellu...More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Institute Of Neuroscienc
Curated by ChEMBL
National Institute Of Neuroscienc
Curated by ChEMBL
Affinity DataEC50: 3nMAssay Description:Antagonist activity at human recombinant delta opioid receptor expressed in CHO cells coexpressing alphaqi5 assessed as inhibition of DPDPE-induced i...More data for this Ligand-Target Pair
Affinity DataEC50: 70.8nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.24nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
Affinity DataEC50: 229nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
Affinity DataEC50: 66.1nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
Affinity DataEC50: 87.1nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
Affinity DataEC50: 13.8nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
Affinity DataEC50: 776nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.24nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.80nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.66E+3nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
Affinity DataEC50: 661nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.69E+3nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
Affinity DataEC50: 794nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0490nMAssay Description:Antagonist activity at human recombinant NK1 receptor expressed in CHO cells assessed as inhibition of NPS-induced intracellular calcium mobilizationMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
National Institute Of Neuroscienc
Curated by ChEMBL
National Institute Of Neuroscienc
Curated by ChEMBL
Affinity DataEC50: 0.0339nMAssay Description:Antagonist activity at human recombinant bradykinin 2 receptor expressed in CHO cells assessed as inhibition of bradykinin-induced intracellular calc...More data for this Ligand-Target Pair
Affinity DataEC50: 3.5nMAssay Description:Antagonist activity at human recombinant urotensin 2 receptor expressed in CHO cells assessed as inhibition of urotensin 2-induced intracellular calc...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
National Institute Of Neuroscienc
Curated by ChEMBL
National Institute Of Neuroscienc
Curated by ChEMBL
Affinity DataEC50: 11nMAssay Description:Antagonist activity at human recombinant mu opioid receptor expressed in CHO cells coexpressing alphaqi5 assessed as inhibition of dermorphin-induced...More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute Of Neuroscienc
Curated by ChEMBL
National Institute Of Neuroscienc
Curated by ChEMBL
Affinity DataEC50: 2.30nMAssay Description:Antagonist activity at human recombinant kappa opioid receptor expressed in CHO cells coexpressing alphaqi5 assessed as inhibition of dynorphin A-ind...More data for this Ligand-Target Pair
Affinity DataEC50: 0.282nMAssay Description:Antagonist activity at human recombinant NOP receptor expressed in CHO cells coexpressing alphaqi5 assessed as inhibition of N/OFQ-induced intracellu...More data for this Ligand-Target Pair
TargetProteinase-activated receptor 2(Homo sapiens (Human))
National Institute Of Neuroscienc
Curated by ChEMBL
National Institute Of Neuroscienc
Curated by ChEMBL
Affinity DataEC50: 3.16E+4nMAssay Description:Antagonist activity at human recombinant PAR2 expressed in A549 cells assessed as inhibition of SLIGKV-NH2-induced intracellular calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0575nMAssay Description:Antagonist activity at human recombinant NK1 receptor expressed in CHO cells assessed as inhibition of NPS-induced intracellular calcium mobilizationMore data for this Ligand-Target Pair
TargetProteinase-activated receptor 2(Homo sapiens (Human))
National Institute Of Neuroscienc
Curated by ChEMBL
National Institute Of Neuroscienc
Curated by ChEMBL
Affinity DataEC50: 2.82E+4nMAssay Description:Antagonist activity at human recombinant PAR2 expressed in A549 cells assessed as inhibition of SLIGKV-NH2-induced intracellular calcium mobilizationMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute Of Neuroscienc
Curated by ChEMBL
National Institute Of Neuroscienc
Curated by ChEMBL
Affinity DataEC50: 6.30nMAssay Description:Antagonist activity at human recombinant kappa opioid receptor expressed in CHO cells coexpressing alphaqi5 assessed as inhibition of dynorphin A-ind...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
National Institute Of Neuroscienc
Curated by ChEMBL
National Institute Of Neuroscienc
Curated by ChEMBL
Affinity DataEC50: 10nMAssay Description:Antagonist activity at human recombinant mu opioid receptor expressed in CHO cells coexpressing alphaqi5 assessed as inhibition of dermorphin-induced...More data for this Ligand-Target Pair
Affinity DataEC50: 4.10nMAssay Description:Antagonist activity at human recombinant urotensin 2 receptor expressed in CHO cells assessed as inhibition of urotensin 2-induced intracellular calc...More data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
National Institute Of Neuroscienc
Curated by ChEMBL
National Institute Of Neuroscienc
Curated by ChEMBL
Affinity DataEC50: 0.0490nMAssay Description:Antagonist activity at human recombinant bradykinin 2 receptor expressed in CHO cells assessed as inhibition of bradykinin-induced intracellular calc...More data for this Ligand-Target Pair