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Found 85 with Last Name = 'reinscheid' and Initial = 'rk'
TargetCysteinyl leukotriene receptor 1(Homo sapiens (Human))
University of California Irvine

Curated by PDSP Ki Database
LigandPNGBDBM50009073(4-(5-cyclopentyloxycarbonylamino-1-methyl-1H-indol...)
Affinity DataKi:  0.260nMMore data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 1(Homo sapiens (Human))
University of California Irvine

Curated by PDSP Ki Database
LigandPNGBDBM85673(CAS_5311297 | Montelukast | NSC_5311297)
Affinity DataKi:  2.30nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(Homo sapiens (Human))
University of California Irvine

Curated by PDSP Ki Database
LigandPNGBDBM50001285((E)-3-((3-(2-(7-chloroquinolin-2-yl)vinyl)phenyl)(...)
Affinity DataKi:  10.4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50443391(CHEMBL469695)
Affinity DataKi:  48nMAssay Description:Binding affinity to human NPSR by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine

Curated by PDSP Ki Database
LigandPNGBDBM85722(BAY u9773 | CAS_134733-55-4)
Affinity DataKi:  300nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine

Curated by PDSP Ki Database
LigandPNGBDBM50001285((E)-3-((3-(2-(7-chloroquinolin-2-yl)vinyl)phenyl)(...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine

Curated by PDSP Ki Database
LigandPNGBDBM50009073(4-(5-cyclopentyloxycarbonylamino-1-methyl-1H-indol...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine

Curated by PDSP Ki Database
LigandPNGBDBM85673(CAS_5311297 | Montelukast | NSC_5311297)
Affinity DataKi:  5.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50423102(CHEMBL267479)
Affinity DataIC50:  537nMAssay Description:Antagonist activity at mouse NPSR expressed in HEK293 cells assessed as inhibition of 10 nM hNPS-induced calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50423102(CHEMBL267479)
Affinity DataIC50:  1.62E+3nMAssay Description:Antagonist activity at mouse NPSR expressed in HEK293 cells assessed as inhibition of 100 nM hNPS-induced calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50479767(CHEMBL451444)
Affinity DataEC50:  562nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells assessed as increase in intracellular calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50479768(CHEMBL503441)
Affinity DataEC50:  372nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells assessed as increase in intracellular calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50479769(CHEMBL510338)
Affinity DataEC50:  32nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells assessed as increase in intracellular calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50479770(CHEMBL500802)
Affinity DataEC50:  1.55E+3nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells assessed as increase in intracellular calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50479771(CHEMBL447434)
Affinity DataEC50:  166nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells assessed as increase in intracellular calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50479772(CHEMBL525031)
Affinity DataEC50:  85nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells assessed as increase in intracellular calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50479773(CHEMBL524688)
Affinity DataEC50:  22nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells assessed as increase in intracellular calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50479774(CHEMBL506383)
Affinity DataEC50:  129nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells assessed as increase in intracellular calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50479775(CHEMBL510673)
Affinity DataEC50:  204nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells assessed as increase in intracellular calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50479776(CHEMBL505996)
Affinity DataEC50:  240nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells assessed as increase in intracellular calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50479777(CHEMBL499957)
Affinity DataEC50:  1.26E+3nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells assessed as increase in intracellular calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Institute Of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50413782(CHEMBL1627325)
Affinity DataEC50:  1.90nMAssay Description:Antagonist activity at human recombinant delta opioid receptor expressed in CHO cells coexpressing alphaqi5 assessed as inhibition of DPDPE-induced i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
National Institute Of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50004178(Nociceptin | Nociceptin/orphanin FQ | ORPHANIN FQ)
Affinity DataEC50:  0.389nMAssay Description:Antagonist activity at human recombinant NOP receptor expressed in CHO cells coexpressing alphaqi5 assessed as inhibition of N/OFQ-induced intracellu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Institute Of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50001683(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataEC50:  3nMAssay Description:Antagonist activity at human recombinant delta opioid receptor expressed in CHO cells coexpressing alphaqi5 assessed as inhibition of DPDPE-induced i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50412700(CHEMBL526492)
Affinity DataEC50:  70.8nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50412701(CHEMBL525809)
Affinity DataEC50:  2.24nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50412702(CHEMBL526323)
Affinity DataEC50:  229nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50412703(CHEMBL505657)
Affinity DataEC50:  66.1nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50412704(CHEMBL507881)
Affinity DataEC50:  87.1nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50412705(CHEMBL526355)
Affinity DataEC50:  13.8nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50412706(CHEMBL525398)
Affinity DataEC50:  776nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50412707(CHEMBL230333)
Affinity DataEC50:  2.24nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50412707(CHEMBL230333)
Affinity DataEC50:  4.80nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50413778(CHEMBL500443)
Affinity DataEC50:  1.66E+3nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50413779(CHEMBL500458)
Affinity DataEC50:  661nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50413780(CHEMBL507664)
Affinity DataEC50:  2.69E+3nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Mus musculus)
Istituto Di Chimica Biomolecolare

Curated by ChEMBL
LigandPNGBDBM50413781(CHEMBL509091)
Affinity DataEC50:  794nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
National Institute Of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50413782(CHEMBL1627325)
Affinity DataEC50:  0.0490nMAssay Description:Antagonist activity at human recombinant NK1 receptor expressed in CHO cells assessed as inhibition of NPS-induced intracellular calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
National Institute Of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50413782(CHEMBL1627325)
Affinity DataEC50:  0.0339nMAssay Description:Antagonist activity at human recombinant bradykinin 2 receptor expressed in CHO cells assessed as inhibition of bradykinin-induced intracellular calc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
National Institute Of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50413782(CHEMBL1627325)
Affinity DataEC50:  3.5nMAssay Description:Antagonist activity at human recombinant urotensin 2 receptor expressed in CHO cells assessed as inhibition of urotensin 2-induced intracellular calc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
National Institute Of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50413782(CHEMBL1627325)
Affinity DataEC50:  11nMAssay Description:Antagonist activity at human recombinant mu opioid receptor expressed in CHO cells coexpressing alphaqi5 assessed as inhibition of dermorphin-induced...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute Of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50413782(CHEMBL1627325)
Affinity DataEC50:  2.30nMAssay Description:Antagonist activity at human recombinant kappa opioid receptor expressed in CHO cells coexpressing alphaqi5 assessed as inhibition of dynorphin A-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
National Institute Of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50413782(CHEMBL1627325)
Affinity DataEC50:  0.282nMAssay Description:Antagonist activity at human recombinant NOP receptor expressed in CHO cells coexpressing alphaqi5 assessed as inhibition of N/OFQ-induced intracellu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 2(Homo sapiens (Human))
National Institute Of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50413782(CHEMBL1627325)
Affinity DataEC50:  3.16E+4nMAssay Description:Antagonist activity at human recombinant PAR2 expressed in A549 cells assessed as inhibition of SLIGKV-NH2-induced intracellular calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
National Institute Of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataEC50:  0.0575nMAssay Description:Antagonist activity at human recombinant NK1 receptor expressed in CHO cells assessed as inhibition of NPS-induced intracellular calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 2(Homo sapiens (Human))
National Institute Of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50413783(CHEMBL443719)
Affinity DataEC50:  2.82E+4nMAssay Description:Antagonist activity at human recombinant PAR2 expressed in A549 cells assessed as inhibition of SLIGKV-NH2-induced intracellular calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute Of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50010702(CHEMBL411557 | DYNORPHIN(1-17)-OH | Dynorphin A (1...)
Affinity DataEC50:  6.30nMAssay Description:Antagonist activity at human recombinant kappa opioid receptor expressed in CHO cells coexpressing alphaqi5 assessed as inhibition of dynorphin A-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
National Institute Of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50059841((S)-1-[(S)-2-[2-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hy...)
Affinity DataEC50:  10nMAssay Description:Antagonist activity at human recombinant mu opioid receptor expressed in CHO cells coexpressing alphaqi5 assessed as inhibition of dermorphin-induced...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
National Institute Of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50413784(UROTENSIN-II)
Affinity DataEC50:  4.10nMAssay Description:Antagonist activity at human recombinant urotensin 2 receptor expressed in CHO cells assessed as inhibition of urotensin 2-induced intracellular calc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
National Institute Of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50049949((BK) H-Arg-Pro-Pro-Gly-Phe-Ser-Pro-Phe-Arg-OH | (b...)
Affinity DataEC50:  0.0490nMAssay Description:Antagonist activity at human recombinant bradykinin 2 receptor expressed in CHO cells assessed as inhibition of bradykinin-induced intracellular calc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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