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Found 39 with Last Name = 'slaninová' and Initial = 'j'
TargetOxytocin receptor(RAT)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50056796(CHEMBL435716 | DEAMINOOXYTOCIN)
Affinity DataKi:  0.900nMAssay Description:Binding affinity against Oxytocin receptor was determined in rat uterine membrane using radioligand [3H]-oxytocinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(RAT)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataKi:  1.70nMAssay Description:Binding affinity against Oxytocin receptor was determined in rat uterine membrane using radioligand [3H]-oxytocinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(RAT)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50056795(CHEMBL353396 | Deaminooxytocin Trisulfide)
Affinity DataKi:  3nMAssay Description:Binding affinity against Oxytocin receptor was determined in rat uterine membrane using radioligand [3H]-oxytocinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(RAT)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50056797(CHEMBL352836 | Oxytocin Trisulfide)
Affinity DataKi:  6nMAssay Description:Binding affinity against Oxytocin receptor was determined in rat uterine membrane using radioligand [3H]-oxytocinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataIC50:  2.70nMAssay Description:Displacement of [3H]OT from human OT receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50389547(CHEMBL2063984)
Affinity DataIC50:  3.47nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50389547(CHEMBL2063984)
Affinity DataIC50:  3.47nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM82258(CAS_114798-26-4 | Losartan | NSC_3961)
Affinity DataIC50:  5.62nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM82258(CAS_114798-26-4 | Losartan | NSC_3961)
Affinity DataIC50:  6nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50205997(CHEMBL395290 | [Pip7]OT)
Affinity DataIC50:  7nMAssay Description:Displacement of [3H]OT from human OT receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50389544(CHEMBL2063983)
Affinity DataIC50:  24.0nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50389544(CHEMBL2063983)
Affinity DataIC50:  24nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50205999(CHEMBL434193 | [Mpa1, D-Tyr(Et)2, D-Tic7, D-Tic9]O...)
Affinity DataIC50:  25nMAssay Description:Displacement of [3H]OT from human OT receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50389541(CHEMBL2063979)
Affinity DataIC50:  30nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50389541(CHEMBL2063979)
Affinity DataIC50:  30.2nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50205989(CHEMBL393020 | [Mpa1, D-Tyr(Et)2, Pip7]OT)
Affinity DataIC50:  40nMAssay Description:Displacement of [3H]OT from human OT receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50205986(CHEMBL233328 | [Mpa1, D-Tyr(Et)2, D-Tic7]OT)
Affinity DataIC50:  51nMAssay Description:Displacement of [3H]OT from human OT receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50206001(CHEMBL233080 | [Mpa1, D-Tyr(Et)2, Aib7, D-Tic9]OT)
Affinity DataIC50:  55nMAssay Description:Displacement of [3H]OT from human OT receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50206000(CHEMBL395430 | [Aib7]OT)
Affinity DataIC50:  75nMAssay Description:Displacement of [3H]OT from human OT receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50205987(CHEMBL438849 | [Mpa1, D-Tyr(Et)2, D-Tic7, Aib9]OT)
Affinity DataIC50:  80nMAssay Description:Displacement of [3H]OT from human OT receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50205992(CHEMBL415418 | [Mpa1, L-Tic7]OT)
Affinity DataIC50:  103nMAssay Description:Displacement of [3H]OT from human OT receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50389542(CHEMBL2063981)
Affinity DataIC50:  117nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50389542(CHEMBL2063981)
Affinity DataIC50:  117nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50205996(CHEMBL397407 | [L-Tic7]OT)
Affinity DataIC50:  130nMAssay Description:Displacement of [3H]OT from human OT receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50205995(CHEMBL234377 | [Mpa1, D-Tyr(Et)2, L-Tic7]OT)
Affinity DataIC50:  176nMAssay Description:Displacement of [3H]OT from human OT receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50389545(CHEMBL2063985)
Affinity DataIC50:  245nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50389545(CHEMBL2063985)
Affinity DataIC50:  245nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50205991(CHEMBL265630 | [Mpa1, D-Tic7]OT)
Affinity DataIC50:  380nMAssay Description:Displacement of [3H]OT from human OT receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50389543(CHEMBL2063982)
Affinity DataIC50:  446nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50389543(CHEMBL2063982)
Affinity DataIC50:  447nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50205988(CHEMBL393021 | [Mpa1, D-Tyr(Et)2, Aib7]OT)
Affinity DataIC50:  485nMAssay Description:Displacement of [3H]OT from human OT receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50389546(CHEMBL2063980)
Affinity DataIC50:  631nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50389546(CHEMBL2063980)
Affinity DataIC50:  634nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50205985(CHEMBL435159 | [D-Tic7]OT)
Affinity DataIC50:  730nMAssay Description:Displacement of [3H]OT from human OT receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50205993(CHEMBL441128 | [Mpa1, D-Tyr(Et)2, Gly(But)7]OT)
Affinity DataIC50:  1.00E+3nMAssay Description:Displacement of [3H]OT from human OT receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50205984(CHEMBL234363 | [Gly(But)7]OT)
Affinity DataIC50:  1.38E+3nMAssay Description:Displacement of [3H]OT from human OT receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50205994(CHEMBL232501 | [Mpa1, D-Tyr(Et)2, Gly(But)3, Gly(B...)
Affinity DataIC50:  7.85E+3nMAssay Description:Displacement of [3H]OT from human OT receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50205983(CHEMBL394268 | [Mpa1, D-Tic2, Aib7]OT)
Affinity DataIC50:  8.50E+3nMAssay Description:Displacement of [3H]OT from human OT receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50205998(CHEMBL415417 | [Gly(But)3, Gly(But)7]OT)
Affinity DataIC50:  5.17E+4nMAssay Description:Displacement of [3H]OT from human OT receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed