Compile Data Set for Download or QSAR
maximum 50k data
Found 247 with Last Name = 'soliman' and Initial = 'me'
TargetCarbonic anhydrase 7(Homo sapiens (Human))TBA
LigandPNGBDBM50612155(CHEMBL5288797)
Affinity DataKi:  0.280nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCarbonic anhydrase 7(Homo sapiens (Human))TBA
LigandPNGBDBM50612159(CHEMBL5266341)
Affinity DataKi:  0.350nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCarbonic anhydrase 7(Homo sapiens (Human))TBA
LigandPNGBDBM50612156(CHEMBL5288389)
Affinity DataKi:  0.390nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCarbonic anhydrase 7(Homo sapiens (Human))TBA
LigandPNGBDBM50612160(CHEMBL5289467)
Affinity DataKi:  0.470nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCarbonic anhydrase 7(Homo sapiens (Human))TBA
LigandPNGBDBM50612154(CHEMBL5286350)
Affinity DataKi:  0.960nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
University Of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50485187(CHEMBL2035872)
Affinity DataKi:  1.20nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 7(Homo sapiens (Human))TBA
LigandPNGBDBM50612152(CHEMBL5279810)
Affinity DataKi:  1.5nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCarbonic anhydrase 7(Homo sapiens (Human))TBA
LigandPNGBDBM50612158(CHEMBL5273629)
Affinity DataKi:  2.30nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCarbonic anhydrase 7(Homo sapiens (Human))TBA
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  2.5nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 7(Homo sapiens (Human))TBA
LigandPNGBDBM50612166(CHEMBL5284402)
Affinity DataKi:  2.80nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50612159(CHEMBL5266341)
Affinity DataKi:  3.10nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50612155(CHEMBL5288797)
Affinity DataKi:  3.80nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50612160(CHEMBL5289467)
Affinity DataKi:  4.20nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50612156(CHEMBL5288389)
Affinity DataKi:  5.10nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCarbonic anhydrase 7(Homo sapiens (Human))TBA
LigandPNGBDBM50612157(CHEMBL5265873)
Affinity DataKi:  5.80nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50612158(CHEMBL5273629)
Affinity DataKi:  5.90nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50612163(CHEMBL5268744)
Affinity DataKi:  6.10nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50612161(CHEMBL5273801)
Affinity DataKi:  8.80nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))TBA
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  12nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 7(Homo sapiens (Human))TBA
LigandPNGBDBM50612163(CHEMBL5268744)
Affinity DataKi:  14nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCarbonic anhydrase 7(Homo sapiens (Human))TBA
LigandPNGBDBM50612161(CHEMBL5273801)
Affinity DataKi:  16nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))TBA
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  26nMAssay Description:Binding affinity to human CA9 assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Birla Institute of Technology

LigandPNGBDBM15613(4-chloro-N-(2-morpholin-4-ylethyl)benzamide | 4-ch...)
Affinity DataKi:  30nMAssay Description:The activities of recombinant hMAO-A and hMAO-B were determined using p-tyramine as common substrate and calculated as 0.18 +/- 0.01 nmol/mg/min (n =...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))TBA
LigandPNGBDBM50612159(CHEMBL5266341)
Affinity DataKi:  35nMAssay Description:Binding affinity to human CA9 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCarbonic anhydrase 7(Homo sapiens (Human))TBA
LigandPNGBDBM50612164(CHEMBL5285561)
Affinity DataKi:  37nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCarbonic anhydrase 7(Homo sapiens (Human))TBA
LigandPNGBDBM50612167(CHEMBL5276437)
Affinity DataKi:  41nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))TBA
LigandPNGBDBM50612161(CHEMBL5273801)
Affinity DataKi:  45nMAssay Description:Binding affinity to human CA9 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50612166(CHEMBL5284402)
Affinity DataKi:  45nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))TBA
LigandPNGBDBM50612160(CHEMBL5289467)
Affinity DataKi:  47nMAssay Description:Binding affinity to human CA9 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50612152(CHEMBL5279810)
Affinity DataKi:  52nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50612157(CHEMBL5265873)
Affinity DataKi:  54nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCarbonic anhydrase 7(Homo sapiens (Human))TBA
LigandPNGBDBM50612165(CHEMBL5278830)
Affinity DataKi:  55nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCarbonic anhydrase 7(Homo sapiens (Human))TBA
LigandPNGBDBM50612162(CHEMBL5280008)
Affinity DataKi:  61nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50612154(CHEMBL5286350)
Affinity DataKi:  64nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCarbonic anhydrase 7(Homo sapiens (Human))TBA
LigandPNGBDBM50612153(CHEMBL5275945)
Affinity DataKi:  65nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCarbonic anhydrase 7(Homo sapiens (Human))TBA
LigandPNGBDBM50612169(CHEMBL5290815)
Affinity DataKi:  68nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCarbonic anhydrase 7(Homo sapiens (Human))TBA
LigandPNGBDBM50612168(CHEMBL5268000)
Affinity DataKi:  76nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50612160(CHEMBL5289467)
Affinity DataKi:  79nMAssay Description:Binding affinity to human CA1 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50612159(CHEMBL5266341)
Affinity DataKi:  82nMAssay Description:Binding affinity to human CA1 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50612154(CHEMBL5286350)
Affinity DataKi:  91nMAssay Description:Binding affinity to human CA1 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetGenome polyprotein(West Nile virus)
University Of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50030459(CHEMBL3344321)
Affinity DataKi:  130nMAssay Description:Inhibition of West Nile virus NS2B-NS3 proteaseMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Birla Institute of Technology

LigandPNGBDBM50420209(CHEMBL91153)
Affinity DataKi:  160nMAssay Description:The activities of recombinant hMAO-A and hMAO-B were determined using p-tyramine as common substrate and calculated as 0.18 +/- 0.01 nmol/mg/min (n =...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Birla Institute of Technology

LigandPNGBDBM15579(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Affinity DataKi:  160nMAssay Description:The activities of recombinant hMAO-A and hMAO-B were determined using p-tyramine as common substrate and calculated as 0.18 +/- 0.01 nmol/mg/min (n =...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50612162(CHEMBL5280008)
Affinity DataKi:  188nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))TBA
LigandPNGBDBM50612163(CHEMBL5268744)
Affinity DataKi:  199nMAssay Description:Binding affinity to human CA9 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Birla Institute of Technology

LigandPNGBDBM50011421(2-(4-Nitro-phenyl)-chromen-4-one | CHEMBL64780)
Affinity DataKi:  200nMAssay Description:The activities of recombinant hMAO-A and hMAO-B were determined using p-tyramine as common substrate and calculated as 0.18 +/- 0.01 nmol/mg/min (n =...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))TBA
LigandPNGBDBM50612164(CHEMBL5285561)
Affinity DataKi:  229nMAssay Description:Binding affinity to human CA9 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50612155(CHEMBL5288797)
Affinity DataKi:  250nMAssay Description:Binding affinity to human CA1 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))TBA
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  250nMAssay Description:Binding affinity to human CA1 assessed as inhibition constantMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50612168(CHEMBL5268000)
Affinity DataKi:  291nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
Displayed 1 to 50 (of 247 total ) | Next | Last >>
Jump to: