Affinity DataIC50: 100nMAssay Description:Inhibition of recombinant SIRT1 using ZMAL substrate after 4 hrs by homogeneous fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of MDR1 (unknown origin) expressed in MDCK cells after 30 mins by Calcein-AM assayMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of recombinant SIRT1 using ZMAL substrate after 4 hrs by homogeneous fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 310nMAssay Description:Inhibition of MDR1 (unknown origin) expressed in MDCK cells after 30 mins by Calcein-AM assayMore data for this Ligand-Target Pair
Affinity DataIC50: 540nMAssay Description:Inhibition of MDR1 (unknown origin) expressed in MDCK cells after 30 mins by Calcein-AM assayMore data for this Ligand-Target Pair
Affinity DataIC50: 670nMAssay Description:Inhibition of MDR1 (unknown origin) expressed in MDCK cells after 30 mins by Calcein-AM assayMore data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Inhibition of recombinant SIRT2 using ZMAL substrate after 4 hrs by homogeneous fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 970nMAssay Description:Inhibition of MDR1 (unknown origin) expressed in MDCK cells after 30 mins by Calcein-AM assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of recombinant SIRT2 using ZMAL substrate after 4 hrs by homogeneous fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.02E+3nMAssay Description:Inhibition of MDR1 (unknown origin) expressed in MDCK cells after 30 mins by Calcein-AM assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of recombinant SIRT2 using ZMAL substrate after 4 hrs by homogeneous fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of recombinant SIRT2 using ZMAL substrate after 4 hrs by homogeneous fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.23E+3nMAssay Description:Inhibition of MDR1 (unknown origin) expressed in MDCK cells after 30 mins by Calcein-AM assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of MDR1 (unknown origin) expressed in MDCK cells after 30 mins by Calcein-AM assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of MRP1 (unknown origin) expressed in MDCK cells after 30 mins by Calcein-AM assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacylase sirtuin-5, mitochondrial(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of SIRT5 using ZK(suc)A substrate after 1 hr by homogeneous fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.76E+3nMAssay Description:Inhibition of MDR1 (unknown origin) expressed in MDCK cells after 30 mins by Calcein-AM assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.93E+3nMAssay Description:Inhibition of MDR1 (unknown origin) expressed in MDCK cells after 30 mins by Calcein-AM assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of MDR1 (unknown origin) expressed in MDCK cells after 30 mins by Calcein-AM assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of MDR1 (unknown origin) expressed in MDCK cells after 30 mins by Calcein-AM assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.38E+3nMAssay Description:Inhibition of MRP1 (unknown origin) expressed in MDCK cells after 30 mins by Calcein-AM assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of recombinant SIRT1 using ZMAL substrate after 4 hrs by homogeneous fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of recombinant SIRT2 using ZMAL substrate after 4 hrs by homogeneous fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of recombinant SIRT1 using ZMAL substrate after 4 hrs by homogeneous fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of MRP1 (unknown origin) expressed in MDCK cells after 30 mins by Calcein-AM assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacylase sirtuin-5, mitochondrial(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of SIRT5 using ZK(suc)A substrate after 1 hr by homogeneous fluorescence assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of recombinant SIRT3 using ZMAL substrate after 4 hrs by homogeneous fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.28E+3nMAssay Description:Inhibition of MRP1 (unknown origin) expressed in MDCK cells after 30 mins by Calcein-AM assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.34E+3nMAssay Description:Inhibition of MDR1 (unknown origin) expressed in MDCK cells after 30 mins by Calcein-AM assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.26E+3nMAssay Description:Inhibition of MDR1 (unknown origin) expressed in MDCK cells after 30 mins by Calcein-AM assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of recombinant SIRT1 using ZMAL substrate after 4 hrs by homogeneous fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of MRP1 (unknown origin) expressed in MDCK cells after 30 mins by Calcein-AM assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of recombinant SIRT1 using ZMAL substrate after 4 hrs by homogeneous fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of recombinant SIRT1 using ZMAL substrate after 4 hrs by homogeneous fluorescence assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacylase sirtuin-5, mitochondrial(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of SIRT5 using ZK(suc)A substrate after 1 hr by homogeneous fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.26E+3nMAssay Description:Inhibition of MRP1 (unknown origin) expressed in MDCK cells after 30 mins by Calcein-AM assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.66E+3nMAssay Description:Inhibition of MDR1 (unknown origin) expressed in MDCK cells after 30 mins by Calcein-AM assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of recombinant SIRT1 using ZMAL substrate after 4 hrs by homogeneous fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.50E+3nMAssay Description:Inhibition of recombinant SIRT2 using ZMAL substrate after 4 hrs by homogeneous fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.13E+3nMAssay Description:Inhibition of MRP1 (unknown origin) expressed in MDCK cells after 30 mins by Calcein-AM assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.21E+3nMAssay Description:Inhibition of MDR1 (unknown origin) expressed in MDCK cells after 30 mins by Calcein-AM assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.70E+3nMAssay Description:Inhibition of recombinant SIRT2 using ZMAL substrate after 4 hrs by homogeneous fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.92E+3nMAssay Description:Inhibition of MDR1 (unknown origin) expressed in MDCK cells after 30 mins by Calcein-AM assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9.20E+3nMAssay Description:Inhibition of MDR1 (unknown origin) expressed in MDCK cells after 30 mins by Calcein-AM assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9.70E+3nMAssay Description:Inhibition of recombinant SIRT2 using ZMAL substrate after 4 hrs by homogeneous fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9.80E+3nMAssay Description:Inhibition of recombinant SIRT2 using ZMAL substrate after 4 hrs by homogeneous fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9.90E+3nMAssay Description:Inhibition of recombinant SIRT1 using ZMAL substrate after 4 hrs by homogeneous fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant SIRT2 using ZMAL substrate after 4 hrs by homogeneous fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.04E+4nMAssay Description:Inhibition of recombinant SIRT2 using ZMAL substrate after 4 hrs by homogeneous fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.05E+4nMAssay Description:Inhibition of recombinant SIRT1 using ZMAL substrate after 4 hrs by homogeneous fluorescence assayMore data for this Ligand-Target Pair