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Found 116 with Last Name = 'upadhyay' and Initial = 's'
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))TBA
LigandPNGBDBM50110719(5-Methoxymethyl-3-pyrrol-1-yl-oxazolidin-2-one | C...)
Affinity DataKi:  4.90nMAssay Description:Inhibition of recombinant human MAO-A using kynuramine as substrate incubated for 20 mins by spectrophotometry analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))TBA
LigandPNGBDBM15611(N-Methyl,N-(propargyl),N-(pyrrol-2-ylmethyl)amine ...)
Affinity DataKi:  5.40nMAssay Description:Inhibition of MAO-A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))TBA
LigandPNGBDBM50028010(AD-810 | CHEBI:10127 | CI-912 | PD-110843 | Zonegr...)
Affinity DataKi:  2.90E+3nMAssay Description:Competitive inhibition of rat MAO-BMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))TBA
LigandPNGBDBM50028010(AD-810 | CHEBI:10127 | CI-912 | PD-110843 | Zonegr...)
Affinity DataKi:  3.10E+3nMAssay Description:Competitive inhibition of human MAO-BMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))TBA
LigandPNGBDBM50611766(CHEMBL5268461)
Affinity DataKi:  1.50E+4nMAssay Description:Irreversible inhibition of human recombinant MAO-BMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))TBA
LigandPNGBDBM50028010(AD-810 | CHEBI:10127 | CI-912 | PD-110843 | Zonegr...)
Affinity DataKi:  3.08E+4nMAssay Description:Inhibition of MAO-B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))TBA
LigandPNGBDBM50113840(4-Phenyl-butylamine | 4-phenylbutylamine | CHEMBL7...)
Affinity DataKi:  3.10E+4nMAssay Description:Competitive inhibition of human MAO-AMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50057302(C-(6-Phenyl-cuban-3-yl)-methylamine | CHEMBL17042)
Affinity DataKi:  1.20E+5nMAssay Description:Inhibition constant was evaluated against mitochondrial Monoamine oxidase BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50057301(C-Cuban-1-yl-methylamine | CHEMBL276317)
Affinity DataKi:  1.70E+5nMAssay Description:Inhibition constant was evaluated against mitochondrial Monoamine oxidase BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50057303(C-(6-Cyclopropyl-cuban-3-yl)-methylamine | CHEMBL1...)
Affinity DataKi:  2.60E+5nMAssay Description:Inhibition constant was evaluated against mitochondrial Monoamine oxidase BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))TBA
LigandPNGBDBM50611765(CHEMBL5283202)
Affinity DataKi:  2.68E+5nMAssay Description:Irreversible inhibition of human recombinant MAO-AMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))TBA
LigandPNGBDBM174835(US9114126, 2027BA1)
Affinity DataIC50:  0.220nMAssay Description:Inhibition of rat MAO-AMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))TBA
LigandPNGBDBM50029810(2-[5-(4-Benzyloxy-phenyl)-tetrazol-2-yl]-ethanol |...)
Affinity DataIC50:  2nMAssay Description:Inhibition of human MAO-BMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))TBA
LigandPNGBDBM50029819(2-{5-[4-(3-Chloro-benzyloxy)-phenyl]-tetrazol-2-yl...)
Affinity DataIC50:  2nMAssay Description:Inhibition of human MAO-BMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))TBA
LigandPNGBDBM50611768(CHEMBL292052)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant MAO-AMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))TBA
LigandPNGBDBM50038943(CHEMBL66260 | N-(7-Acetylamino-10-methyl-5,5-dioxo...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant MAO-AMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))TBA
LigandPNGBDBM50611769(CHEMBL65583)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant MAO-AMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))TBA
LigandPNGBDBM50038932(CHEMBL304069 | N-(9,10-Dioxo-9,10-dihydro-anthrace...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant MAO-AMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))TBA
LigandPNGBDBM50611770(CHEMBL304484)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant MAO-AMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))TBA
LigandPNGBDBM50611771(CHEMBL5270901)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant MAO-AMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))TBA
LigandPNGBDBM50261815(2-(3,4-dimethoxyphenyl)-3-fluoroprop-2-en-1-amine ...)
Affinity DataIC50:  10nMAssay Description:Inhibition of MAO-B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))TBA
LigandPNGBDBM50038934(CHEMBL65156 | N-(9,10,10-Trioxo-9,10-dihydro-10lam...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant MAO-AMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))TBA
LigandPNGBDBM50038942(CHEMBL63458 | N-(9,10,10-Trioxo-9,10-dihydro-10lam...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant MAO-AMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))TBA
LigandPNGBDBM50038941(CHEMBL63510 | N-(6-Methyl-9,10,10-trioxo-9,10-dihy...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant MAO-AMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))TBA
LigandPNGBDBM50038938(CHEMBL417566 | N-(6-Ethyl-9,10,10-trioxo-9,10-dihy...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant MAO-AMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))TBA
LigandPNGBDBM50038946(CHEMBL63141 | N-(9,10,10-Trioxo-6-propyl-9,10-dihy...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant MAO-AMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))TBA
LigandPNGBDBM50611767(CHEMBL63782)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant MAO-AMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))TBA
LigandPNGBDBM50038947(CHEMBL63934 | N-(10,10-Dioxo-10H-10lambda*6*-pheno...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant MAO-AMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))TBA
LigandPNGBDBM50038939(CHEMBL63678 | N-(5,5-Dioxo-5,10-dihydro-5lambda*6*...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant MAO-AMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))TBA
LigandPNGBDBM50428646(CHEMBL2332175)
Affinity DataIC50:  11nMAssay Description:Reversible inhibition of human MAO-BMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))TBA
LigandPNGBDBM50029816(5-Chloro-pyridine-2-carboxylic acid (2-amino-ethyl...)
Affinity DataIC50:  30nMAssay Description:Inhibition of human MAO-BMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM50294178(CHEMBL4160682)
Affinity DataIC50:  33nMAssay Description:Displacement of fluoromone TM from recombinant human ERalpha after 2 hrs by fluorescence polarization analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM50294174(CHEMBL4170939)
Affinity DataIC50:  47nMAssay Description:Displacement of fluoromone TM from recombinant human ERalpha after 2 hrs by fluorescence polarization analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMenin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50496327(CHEMBL3126198)
Affinity DataIC50:  56nMAssay Description:Inhibition of human His-tagged menin-biotinylated MLL (4 to 15) interaction after 1 hr by HTRF assayMore data for this Ligand-Target Pair
TargetMenin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50496346(CHEMBL3126196)
Affinity DataIC50:  67nMAssay Description:Inhibition of human His-tagged menin-biotinylated MLL (4 to 15) interaction after 1 hr by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetEstrogen receptor(Homo sapiens (Human))
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM50294181(CHEMBL4169456)
Affinity DataIC50:  74nMAssay Description:Displacement of fluoromone TM from recombinant human ERalpha after 2 hrs by fluorescence polarization analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM50294182(CHEMBL4161120)
Affinity DataIC50:  77nMAssay Description:Displacement of fluoromone TM from recombinant human ERalpha after 2 hrs by fluorescence polarization analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM50294175(CHEMBL4167567)
Affinity DataIC50:  80nMAssay Description:Displacement of fluoromone TM from recombinant human ERalpha after 2 hrs by fluorescence polarization analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMenin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50496331(CHEMBL3126197)
Affinity DataIC50:  81nMAssay Description:Inhibition of human His-tagged menin-biotinylated MLL (4 to 15) interaction after 1 hr by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMenin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50496354(CHEMBL3126194)
Affinity DataIC50:  90nMAssay Description:Inhibition of human His-tagged menin-biotinylated MLL (4 to 15) interaction after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))TBA
LigandPNGBDBM50031048(3-(4-(trifluoromethyl)phenyl)-5H-indeno[1,2-c]pyri...)
Affinity DataIC50:  90nMAssay Description:Inhibition of rat brain MAO-BMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMenin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50496330(CHEMBL3126199)
Affinity DataIC50:  114nMAssay Description:Inhibition of human His-tagged menin-biotinylated MLL (4 to 15) interaction after 1 hr by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetMenin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50496345(CHEMBL3126200)
Affinity DataIC50:  148nMAssay Description:Inhibition of human His-tagged menin-biotinylated MLL (4 to 15) interaction after 1 hr by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM50294185(CHEMBL4168369)
Affinity DataIC50:  192nMAssay Description:Displacement of fluoromone TM from recombinant human ERalpha after 2 hrs by fluorescence polarization analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMenin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50496329(CHEMBL3126201)
Affinity DataIC50:  195nMAssay Description:Inhibition of human His-tagged menin-biotinylated MLL (4 to 15) interaction after 1 hr by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetMenin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50496335(CHEMBL3126188)
Affinity DataIC50:  197nMAssay Description:Inhibition of human His-tagged menin-biotinylated MLL (4 to 15) interaction after 1 hr by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetEstrogen receptor(Homo sapiens (Human))
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM50294176(CHEMBL4164124)
Affinity DataIC50:  202nMAssay Description:Displacement of fluoromone TM from recombinant human ERalpha after 2 hrs by fluorescence polarization analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMenin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50496341(CHEMBL3126193)
Affinity DataIC50:  225nMAssay Description:Inhibition of human His-tagged menin-biotinylated MLL (4 to 15) interaction after 1 hr by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMenin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50496351(CHEMBL3126190)
Affinity DataIC50:  226nMAssay Description:Inhibition of human His-tagged menin-biotinylated MLL (4 to 15) interaction after 1 hr by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMenin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50496333(CHEMBL3126192)
Affinity DataIC50:  242nMAssay Description:Inhibition of human His-tagged menin-biotinylated MLL (4 to 15) interaction after 1 hr by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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