Affinity DataKi: 0.0440nMAssay Description:Inhibition of Factor 10a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.0600nMAssay Description:Inhibition of Factor 10a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.0800nMAssay Description:Inhibition of Factor 10a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.105nMAssay Description:Inhibition of Factor 10a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.117nMAssay Description:Inhibition of Factor 10a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Binding affinity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Inhibition of Factor 10a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Binding affinity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Binding affinity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.540nMAssay Description:Displacement of [125I](+/-)DOI from human 5-HT2B receptor trasfected in CHO cell membrane after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:In vitro inhibitory activity against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Binding affinity for human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Binding affinity for human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Binding affinity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Binding affinity for human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.970nMAssay Description:Displacement of [125I](+/-)DOI from human 5-HT2B receptor trasfected in CHO cell membrane after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Displacement of [125I](+/-)DOI from human 5-HT2B receptor trasfected in CHO cell membrane after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity for human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Binding affinity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Binding affinity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Inhibitory concentration against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:In vitro inhibitory activity against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Displacement of [125I](+/-)DOI from human 5-HT2B receptor trasfected in CHO cell membrane after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Inhibition of Factor 10a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Binding affinity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Binding affinity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Binding affinity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Binding affinity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Inhibitory concentration against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Binding affinity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Binding affinity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Displacement of [125I](+/-)DOI from human 5-HT2B receptor trasfected in CHO cell membrane after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Inhibitory concentration against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Binding affinity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Inhibitory concentration against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Inhibitory concentration against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Binding affinity for human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Binding affinity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Binding affinity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 3.40nMAssay Description:Inhibitory concentration against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Binding affinity for human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Binding affinity for human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 4.10nMAssay Description:Binding affinity for human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 5.20nMAssay Description:In vitro inhibitory activity against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 7.10nMAssay Description:Displacement of [125I](+/-)DOI from human 5-HT2B receptor trasfected in CHO cell membrane after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Binding affinity for human Coagulation factor XMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:Inhibition of BI-BODIPY binding to BRD4 bromodomain 1 (42 to 168 residues)(unknown origin) expressed in Escherichia coli BL21(DE3) by fluorescence an...More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Millennium Pharmaceuticals
Curated by ChEMBL
Millennium Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 110nMAssay Description:Binding affinity to human ERGMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 110nMAssay Description:Inhibition of BI-BODIPY binding to BRD4 bromodomain 1 (42 to 168 residues)(unknown origin) expressed in Escherichia coli BL21(DE3) by fluorescence an...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 140nMAssay Description:Inhibition of BI-BODIPY binding to BRD4 bromodomain 1 (42 to 168 residues)(unknown origin) expressed in Escherichia coli BL21(DE3) by fluorescence an...More data for this Ligand-Target Pair